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Volumn 11, Issue 4, 2006, Pages 417-424

Effects of enantiomer and isomer permeation enhancers on transdermal delivery of ligustrazine hydrochloride

Author keywords

Apparent density; Enantiomer enhancers; Isomer enhancers; Permeation mechanism; Transdermal delivery

Indexed keywords

LIMONENE; PENETRATION ENHANCING AGENT; TERPINENE; TETRAMETHYLPYRAZINE;

EID: 33845218313     PISSN: 10837450     EISSN: 10979867     Source Type: Journal    
DOI: 10.1080/10837450600770163     Document Type: Article
Times cited : (19)

References (34)
  • 1
    • 0031930725 scopus 로고    scopus 로고
    • Cryo-electron diffraction as a tool to study local variations in the lipid organization of human stratum corneum
    • Pilgram, G.S.; Van Pelt, A.M.; Spies, F.; Bouwstra, J.A.; Koerten, H.K. Cryo-electron diffraction as a tool to study local variations in the lipid organization of human stratum corneum. J. Microsc. 1998, 189 (Pt. 1), 71-78.
    • (1998) J. Microsc. , vol.189 , Issue.PART 1 , pp. 71-78
    • Pilgram, G.S.1    Van Pelt, A.M.2    Spies, F.3    Bouwstra, J.A.4    Koerten, H.K.5
  • 2
    • 0014827372 scopus 로고
    • The role of lipids in the epidermal barrier to water diffusion
    • Sweeny, T.M.; Downing, D.T. The role of lipids in the epidermal barrier to water diffusion. J. Invest. Dermatol. 1970, 55 (2), 135-140.
    • (1970) J. Invest. Dermatol. , vol.55 , Issue.2 , pp. 135-140
    • Sweeny, T.M.1    Downing, D.T.2
  • 3
    • 0029917046 scopus 로고    scopus 로고
    • A lamellar matrix model for stratum corneum intercellular lipids. II. Effect of geometry of the stratum corneum on permeation of model drugs 5-fluorouracil and oestradiol
    • Moghimi, H.R.; Williams, A.C.; Barrry, B.W. A lamellar matrix model for stratum corneum intercellular lipids. II. Effect of geometry of the stratum corneum on permeation of model drugs 5-fluorouracil and oestradiol. Int. J. Pharm. 1996, 131 (2), 117-129.
    • (1996) Int. J. Pharm. , vol.131 , Issue.2 , pp. 117-129
    • Moghimi, H.R.1    Williams, A.C.2    Barrry, B.W.3
  • 4
    • 0025828769 scopus 로고
    • Visualization of in vitro percutaneous penetration of mercuric chloride transport through intercellular space versus cellular uptake through desmosomes
    • Boddé, H.E.; van den Brìnk, I.; Koerten, H.K.; de Haan, F.H.N. Visualization of in vitro percutaneous penetration of mercuric chloride transport through intercellular space versus cellular uptake through desmosomes. J. Control. Release 1991, 15 (3), 227-236.
    • (1991) J. Control. Release , vol.15 , Issue.3 , pp. 227-236
    • Boddé, H.E.1    Van Den Brìnk, I.2    Koerten, H.K.3    De Haan, F.H.N.4
  • 5
    • 0032764606 scopus 로고    scopus 로고
    • Effect of chiral enhancers on the permeability of optically active and racemic metoprolol across hairless mouse skin
    • Kommuru, T.R.; Khan, M.A.; Reddy, I.K. Effect of chiral enhancers on the permeability of optically active and racemic metoprolol across hairless mouse skin. Chirality 1999, 11 (7), 536-540.
    • (1999) Chirality , vol.11 , Issue.7 , pp. 536-540
    • Kommuru, T.R.1    Khan, M.A.2    Reddy, I.K.3
  • 6
    • 0028843878 scopus 로고
    • Does solute stereochemistry influence percutaneous penetration
    • Heard, C.M.; Brain, K.R. Does solute stereochemistry influence percutaneous penetration. Chirality 1995, 7 (4), 305-309.
    • (1995) Chirality , vol.7 , Issue.4 , pp. 305-309
    • Heard, C.M.1    Brain, K.R.2
  • 7
    • 0035834175 scopus 로고    scopus 로고
    • Effect of melting point of chiral terpenes on human stratum corneum uptake
    • Mackay, K.M.; Williams, A.C.; Barry, B.W. Effect of melting point of chiral terpenes on human stratum corneum uptake. Int. J. Pharm. 2001, 228 (1-2), 89-97.
    • (2001) Int. J. Pharm. , vol.228 , Issue.1-2 , pp. 89-97
    • Mackay, K.M.1    Williams, A.C.2    Barry, B.W.3
  • 8
    • 0032723185 scopus 로고    scopus 로고
    • Differential permeation of propranolol enantiomers across human skin in vitro from formulations containing an enantioselective excipient
    • Suedee, R.; Brain, K.R.; Heard, C.M. Differential permeation of propranolol enantiomers across human skin in vitro from formulations containing an enantioselective excipient. Chirality 1999, 11 (9), 680-683.
    • (1999) Chirality , vol.11 , Issue.9 , pp. 680-683
    • Suedee, R.1    Brain, K.R.2    Heard, C.M.3
  • 10
    • 0028199842 scopus 로고
    • Chiral β-blockers for transdermal delivery
    • Touitou, E.; Chow, D.D.; Lawter, J.R. Chiral β-blockers for transdermal delivery. Int. J. Pharm. 1994, 104 (1), 19-28.
    • (1994) Int. J. Pharm. , vol.104 , Issue.1 , pp. 19-28
    • Touitou, E.1    Chow, D.D.2    Lawter, J.R.3
  • 11
    • 0029050101 scopus 로고
    • Permeability of pure enantiomers of ketorolac through human cadaer skin
    • Roy, S.D.; Chatterjee, D.J.; Manoukian, E.; Divor, A. Permeability of pure enantiomers of ketorolac through human cadaer skin. J. Pharm. Sci. 1995, 84 (8), 987-990.
    • (1995) J. Pharm. Sci. , vol.84 , Issue.8 , pp. 987-990
    • Roy, S.D.1    Chatterjee, D.J.2    Manoukian, E.3    Divor, A.4
  • 12
    • 0031874357 scopus 로고    scopus 로고
    • Racemate and enantiomers of ketoprofen: Phase diagram, thermodynamic studies, skin permeability, and use of chiral permeation enhancers
    • Kommuru, T.R.; Khan, M.A.; Reddy, I.K. Racemate and enantiomers of ketoprofen: phase diagram, thermodynamic studies, skin permeability, and use of chiral permeation enhancers. J. Pharm. Sci. 1998, 87 (7), 833-840.
    • (1998) J. Pharm. Sci. , vol.87 , Issue.7 , pp. 833-840
    • Kommuru, T.R.1    Khan, M.A.2    Reddy, I.K.3
  • 13
    • 0034867707 scopus 로고    scopus 로고
    • Pharmacokinetics of the R- and S-enantiomers of oxybutynin and N-desethyloxybutynin following oral and transdermal administration of the racemate in healthy volunteers
    • Zobrist, R.H.; Schmid, B.; Feick, A.; Quan, D.; Sanders, S.W. Pharmacokinetics of the R- and S-enantiomers of oxybutynin and N-desethyloxybutynin following oral and transdermal administration of the racemate in healthy volunteers. Pharm. Res. 2001, 18 (7), 1029-1034.
    • (2001) Pharm. Res. , vol.18 , Issue.7 , pp. 1029-1034
    • Zobrist, R.H.1    Schmid, B.2    Feick, A.3    Quan, D.4    Sanders, S.W.5
  • 14
    • 0024473801 scopus 로고
    • Effect of limonene and related compounds on the percutaneous absorption of indomethacin
    • Okabe, H.; Takayama, K.; Ogura, A.; Nagai, T. Effect of limonene and related compounds on the percutaneous absorption of indomethacin, Drug Des. Deliv. 1989, 4 (4) 313-321.
    • (1989) Drug Des. Deliv. , vol.4 , Issue.4 , pp. 313-321
    • Okabe, H.1    Takayama, K.2    Ogura, A.3    Nagai, T.4
  • 16
    • 1842484885 scopus 로고    scopus 로고
    • Formulation and in vitro evaluation of transdermal patches of melatonin
    • Kanikkannan, N.; Andega, S.; Burton, S.; Babu, R. J.; Singh, M. Formulation and in vitro evaluation of transdermal patches of melatonin. Drug Dev. Ind. Pharm. 2004, 30 (2), 205-212.
    • (2004) Drug Dev. Ind. Pharm. , vol.30 , Issue.2 , pp. 205-212
    • Kanikkannan, N.1    Andega, S.2    Burton, S.3    Babu, R.J.4    Singh, M.5
  • 17
    • 0033816053 scopus 로고    scopus 로고
    • Effect of formulation variables on the percutaneous permeation of ketoprofen from gel formulations
    • El-Kattan, A.F.; Asbill, C.S.; Kim, N.; Michniak, B.B. Effect of formulation variables on the percutaneous permeation of ketoprofen from gel formulations. Drug Deliv. 2000, 7 (3), 147-153.
    • (2000) Drug Deliv. , vol.7 , Issue.3 , pp. 147-153
    • El-Kattan, A.F.1    Asbill, C.S.2    Kim, N.3    Michniak, B.B.4
  • 18
    • 0032214492 scopus 로고    scopus 로고
    • Pre'atb. V. In vitro percutaneous penetration through hairless rat skin: Influence of temperature, vehicle and penetration enhancers
    • Clarysa, P.; Alewaetersa, K.; Jadoulb, A.; Barela, A.; Manadasb, R.O.; Pre'atb. V. In vitro percutaneous penetration through hairless rat skin: Influence of temperature, vehicle and penetration enhancers. Eur. J. Pharm. Biopharm. 1998, 46 (3), 279-283.
    • (1998) Eur. J. Pharm. Biopharm. , vol.46 , Issue.3 , pp. 279-283
    • Clarysa, P.1    Alewaetersa, K.2    Jadoulb, A.3    Barela, A.4    Manadasb, R.O.5
  • 19
    • 0000686969 scopus 로고
    • Ultrastructural evaluation of porcine integument
    • Tumbleson, M.E. (Ed.); Plenum Press: New York
    • Monteiro-Riviere, N. Ultrastructural evaluation of porcine integument. In Swine in Biomedical Research; Tumbleson, M.E. (Ed.); Plenum Press: New York, 1986, 641-655.
    • (1986) Swine in Biomedical Research , pp. 641-655
    • Monteiro-Riviere, N.1
  • 20
    • 0034607386 scopus 로고    scopus 로고
    • The effect of terpene enhancer lipophilicity on the percutaneous permeation of hydrocortisone formulated in HPMC gel systems
    • El-Kattan, A.F.; Asbill, C.S.; Michniak, B.B. The effect of terpene enhancer lipophilicity on the percutaneous permeation of hydrocortisone formulated in HPMC gel systems, Int. J. Pharm. 2000, 198 (2), 179-189.
    • (2000) Int. J. Pharm. , vol.198 , Issue.2 , pp. 179-189
    • El-Kattan, A.F.1    Asbill, C.S.2    Michniak, B.B.3
  • 21
    • 0037177466 scopus 로고    scopus 로고
    • Boldrini effect of different terpene-containing essential oils on permeation of estradiol through hairless mouse skin
    • Monti, D.P.; Chetoni, S.; Burgalassi, M.; Najarro, M.; Fabrizio Saettone, E. Boldrini effect of different terpene-containing essential oils on permeation of estradiol through hairless mouse skin. Int. J. Pharm. 2002, 237 (1-2), 209-214.
    • (2002) Int. J. Pharm. , vol.237 , Issue.1-2 , pp. 209-214
    • Monti, D.P.1    Chetoni, S.2    Burgalassi, M.3    Najarro, M.4    Fabrizio Saettone, E.5
  • 22
    • 0036430094 scopus 로고    scopus 로고
    • Enhancement effects of (R) and (S) enantiomers and the racemate of a model enhancer on permeation of theophylline through human skin
    • Vavrova, K.; Hrabalek, A.; Dolezal, P. Enhancement effects of (R) and (S) enantiomers and the racemate of a model enhancer on permeation of theophylline through human skin. Arch. Dermatol. Res. 2002, 294 (8), 383-385.
    • (2002) Arch. Dermatol. Res. , vol.294 , Issue.8 , pp. 383-385
    • Vavrova, K.1    Hrabalek, A.2    Dolezal, P.3
  • 23
    • 0030057728 scopus 로고    scopus 로고
    • Modes of action of terpene penetration enhancers in human corneum skin; differential scanning calorimetry, small-angle X-ray: Diffraction and enhancer uptake studies
    • Cornwell, P.A.; Barry, B.W.; Bouwstra, J.A.; Gooris, G.S. Modes of action of terpene penetration enhancers in human corneum skin; differential scanning calorimetry, small-angle X-ray:diffraction and enhancer uptake studies. Int. J. Pharm. 1996, 127 (1), 9-26
    • (1996) Int. J. Pharm. , vol.127 , Issue.1 , pp. 9-26
    • Cornwell, P.A.1    Barry, B.W.2    Bouwstra, J.A.3    Gooris, G.S.4
  • 24
    • 0028351443 scopus 로고
    • Comparative analysis of percutaneous absorption enhancement by d-limonene and oleic acid based on a skin diffusion model
    • Koyama, Y.; Bando, H.; Yamashita, F.; Takakura, Y.; Sezaki, H.; Hashida, M. Comparative analysis of percutaneous absorption enhancement by d-limonene and oleic acid based on a skin diffusion model. Pharm. Res. 1994, 11 (3), 377-383.
    • (1994) Pharm. Res. , vol.11 , Issue.3 , pp. 377-383
    • Koyama, Y.1    Bando, H.2    Yamashita, F.3    Takakura, Y.4    Sezaki, H.5    Hashida, M.6
  • 25
    • 0031722003 scopus 로고    scopus 로고
    • Mechanisms of percutaneous absorption of tamoxifen by terpenes: Eugenol, D-limonene and menthone
    • Zhao, K.; Singh, J. Mechanisms of percutaneous absorption of tamoxifen by terpenes: Eugenol, D-limonene and menthone. J. Control. Release 1998, 55 (2-3), 253-260.
    • (1998) J. Control. Release , vol.55 , Issue.2-3 , pp. 253-260
    • Zhao, K.1    Singh, J.2
  • 26
    • 0000460590 scopus 로고
    • Infrared spectroscopy of stratum corneum lipids: In vitro results and their relevance to permeability
    • Walters, K.A., Hadgraft, J. (Eds.); Marcel Dekker: New York
    • Potts and Francoeur. Infrared spectroscopy of stratum corneum lipids: In vitro results and their relevance to permeability. In Pharmaceutical Skin Permeation Enhancement; Walters, K.A., Hadgraft, J. (Eds.); Marcel Dekker: New York, 1993, 269-291.
    • (1993) Pharmaceutical Skin Permeation Enhancement , pp. 269-291
    • Potts1    Francoeur2
  • 27
    • 0021755229 scopus 로고
    • Polymorphic phase behaviour of phospholipids membranes studied by infrared spectroscopy
    • Casal, H.L.; Mantsch, H.H. Polymorphic phase behaviour of phospholipids membranes studied by infrared spectroscopy. Biochim. Biophys. Acta. 1984, 779 (4), 381-401.
    • (1984) Biochim. Biophys. Acta , vol.779 , Issue.4 , pp. 381-401
    • Casal, H.L.1    Mantsch, H.H.2
  • 28
    • 0032443395 scopus 로고    scopus 로고
    • Mechanism of transport enhancement of LHRH through porcine epidermis by terpenes and iontophoresis: Permeability and lipid extraction studies
    • Bhatia, K.S.; Singh. J. Mechanism of transport enhancement of LHRH through porcine epidermis by terpenes and iontophoresis: permeability and lipid extraction studies. Pharm. Res. 1998, 15 (12), 1857-1862.
    • (1998) Pharm. Res. , vol.15 , Issue.12 , pp. 1857-1862
    • Bhatia, K.S.1    Singh, J.2
  • 29
    • 0035850210 scopus 로고    scopus 로고
    • Characterization of the influence of polyol fatty acid esters on the permeation of diclofenac through rat skin
    • Takahashi, K.; Sakano, H.; Yoshida, M.; Numata, N.; Mizuno, N. Characterization of the influence of polyol fatty acid esters on the permeation of diclofenac through rat skin. J. Control. Release 2001, 73 (2-3), 351-358.
    • (2001) J. Control. Release , vol.73 , Issue.2-3 , pp. 351-358
    • Takahashi, K.1    Sakano, H.2    Yoshida, M.3    Numata, N.4    Mizuno, N.5
  • 30
    • 0029826157 scopus 로고    scopus 로고
    • Effects of phospholipids on the in vitro percutaneous penetration of prednisolone and analysis of mechanism by using attenuated total reflectance-Fourier transform infrared spectroscopy
    • Yokomizo, Y.; Sagitani, H. Effects of phospholipids on the in vitro percutaneous penetration of prednisolone and analysis of mechanism by using attenuated total reflectance-Fourier transform infrared spectroscopy. J. Pharm. Sci. 1996, 85 (11), 1220-1226.
    • (1996) J. Pharm. Sci. , vol.85 , Issue.11 , pp. 1220-1226
    • Yokomizo, Y.1    Sagitani, H.2
  • 31
    • 0346104840 scopus 로고    scopus 로고
    • Role of solvent in interactions between fatty acids-based formulations and lipids in porcine stratum corneum
    • Wang, M.Y.; Yang, Y.Y.; Heng, P.W.S. Role of solvent in interactions between fatty acids-based formulations and lipids in porcine stratum corneum. J. Control. Release 2004, 94 (1) 207-216
    • (2004) J. Control. Release , vol.94 , Issue.1 , pp. 207-216
    • Wang, M.Y.1    Yang, Y.Y.2    Heng, P.W.S.3
  • 32
    • 0015134929 scopus 로고
    • Permeablity of the skin
    • Scheuplein, R.J., Blank, I.H., Permeablity of the skin. Physiol. Rev. 1971, 51 (4), 702-747
    • (1971) Physiol. Rev. , vol.51 , Issue.4 , pp. 702-747
    • Scheuplein, R.J.1    Blank, I.H.2
  • 33
    • 0042768142 scopus 로고    scopus 로고
    • Oxide terpenes as human skin penetration enhancers of haloperidol from ethanol and propylene glycol and their modes of action on stratum corneum
    • Vaddi, H.K.; Ho, P.C.; Chan, Y.W.; Chan, S.Y. Oxide terpenes as human skin penetration enhancers of haloperidol from ethanol and propylene glycol and their modes of action on stratum corneum. Biol. Pharm. Bull. 2003, 26 (2), 220-228.
    • (2003) Biol. Pharm. Bull. , vol.26 , Issue.2 , pp. 220-228
    • Vaddi, H.K.1    Ho, P.C.2    Chan, Y.W.3    Chan, S.Y.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.