메뉴 건너뛰기




Volumn 131, Issue 2, 1996, Pages 117-129

A lamellar matrix model for stratum corneum intercellular lipids. II. Effect of geometry of the stratum corneum on permeation of model drugs 5-fluorouracil and oestradiol

Author keywords

5 Fluorouracil; Activation energy; Diffusion coefficient; Model human stratum corneum lipid; Oestradiol; Permeability coefficient

Indexed keywords

ESTRADIOL; FLUOROURACIL; SKIN LIPID;

EID: 0029917046     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/0378-5173(95)04307-1     Document Type: Article
Times cited : (42)

References (34)
  • 1
    • 0021152563 scopus 로고
    • An automated diffusion apparatus for studying skin penetration
    • Akhter, S.A., Bennett, S.L., Waller, I.L. and Barry, B.W., An automated diffusion apparatus for studying skin penetration. Int. J. Pharm., 21 (1984) 17-26.
    • (1984) Int. J. Pharm. , vol.21 , pp. 17-26
    • Akhter, S.A.1    Bennett, S.L.2    Waller, I.L.3    Barry, B.W.4
  • 2
    • 0018383835 scopus 로고
    • Percutaneous absorption: In vivo experiments
    • Albery, W.J. and Hadgraft, J., Percutaneous absorption: in vivo experiments. J. Pharm. Pharmacol., 31 (1979) 140-147.
    • (1979) J. Pharm. Pharmacol. , vol.31 , pp. 140-147
    • Albery, W.J.1    Hadgraft, J.2
  • 4
    • 0001239953 scopus 로고
    • Studies of diffusion of water through dead human skin: The effect of different environmental states and of chemical alterations of the epidermis
    • Berenson, G.S. and Burch, G.E., Studies of diffusion of water through dead human skin: the effect of different environmental states and of chemical alterations of the epidermis. Am. J. Trop. Med. Hyg., 31 (1951) 842-853.
    • (1951) Am. J. Trop. Med. Hyg. , vol.31 , pp. 842-853
    • Berenson, G.S.1    Burch, G.E.2
  • 5
    • 0025828769 scopus 로고
    • Visualization of in vitro percutaneous penetration of mercuric chloride; transport through intercellular space versus cellular uptake through desmosomes
    • Boddé, H.E., van den Brink, I., Koerten, H.K. and de Haan, F.H.N., Visualization of in vitro percutaneous penetration of mercuric chloride; transport through intercellular space versus cellular uptake through desmosomes. J. Controlled Release, 15 (1991) 227-236.
    • (1991) J. Controlled Release , vol.15 , pp. 227-236
    • Boddé, H.E.1    Van Den Brink, I.2    Koerten, H.K.3    De Haan, F.H.N.4
  • 7
    • 0027258908 scopus 로고
    • The routes of penetration of ions and 5-fluorouracil across human skin and the mechanisms of action of terpene skin penetration enhancers
    • Cornwell, P.A. and Barry, B.W., The routes of penetration of ions and 5-fluorouracil across human skin and the mechanisms of action of terpene skin penetration enhancers. Int. J. Pharm., 94 (1993) 189-194.
    • (1993) Int. J. Pharm. , vol.94 , pp. 189-194
    • Cornwell, P.A.1    Barry, B.W.2
  • 8
    • 0028314174 scopus 로고
    • Sesquiterpene components of volatile oils as skin penetration enhancers for the hydrophilic permeant 5-fluorouracil
    • Cornwell, P.A. and Barry, B.W., Sesquiterpene components of volatile oils as skin penetration enhancers for the hydrophilic permeant 5-fluorouracil. J. Pharm. Pharmacol., 46 (1994) 261-269.
    • (1994) J. Pharm. Pharmacol. , vol.46 , pp. 261-269
    • Cornwell, P.A.1    Barry, B.W.2
  • 9
    • 84991131535 scopus 로고
    • Epidermal lipids, membranes, and keratinization
    • Elias, P.M., Epidermal lipids, membranes, and keratinization. Int. J. Dermatol., 20 (1981) 1-19.
    • (1981) Int. J. Dermatol. , vol.20 , pp. 1-19
    • Elias, P.M.1
  • 10
    • 0018574988 scopus 로고
    • Localization and composition of lipids in neonatal mouse stratum granulosum and stratum corneum
    • Elias, P.M., Brown, B.E., Fritsch, P., Goerke, J., Gray, G.M. and White, R.J., Localization and composition of lipids in neonatal mouse stratum granulosum and stratum corneum. J. Invest. Dermatol., 73 (1979) 339-348.
    • (1979) J. Invest. Dermatol. , vol.73 , pp. 339-348
    • Elias, P.M.1    Brown, B.E.2    Fritsch, P.3    Goerke, J.4    Gray, G.M.5    White, R.J.6
  • 11
    • 0016608422 scopus 로고
    • The permeability barrier in mammalian epidermis
    • Elias, P.M. and Friend, D.S., The permeability barrier in mammalian epidermis. J. Cell Biol., 65 (1975) 180-191.
    • (1975) J. Cell Biol. , vol.65 , pp. 180-191
    • Elias, P.M.1    Friend, D.S.2
  • 12
    • 0024909221 scopus 로고
    • Water evaporation rates from a model of stratum corneum lipids
    • Friberg, S.E. and Kayali, I., Water evaporation rates from a model of stratum corneum lipids. J. Pharm. Sci., 78 (1989) 639-643.
    • (1989) J. Pharm. Sci. , vol.78 , pp. 639-643
    • Friberg, S.E.1    Kayali, I.2
  • 13
    • 0023680522 scopus 로고
    • Action of penetration enhancers on human skin as assessed by the permeation of model drugs 5-fluorouracil and estradiol. I. Infinite dose technique
    • Goodman, M. and Barry, B.W., Action of penetration enhancers on human skin as assessed by the permeation of model drugs 5-fluorouracil and estradiol. I. Infinite dose technique. J. Invest. Dermatol., 91 (1988) 323-327.
    • (1988) J. Invest. Dermatol. , vol.91 , pp. 323-327
    • Goodman, M.1    Barry, B.W.2
  • 14
    • 73049177744 scopus 로고
    • Analysis of data on the medicament release from ointments
    • Higuchi, W.I., Analysis of data on the medicament release from ointments. J. Pharm. Sci., 51 (1962) 802-804.
    • (1962) J. Pharm. Sci. , vol.51 , pp. 802-804
    • Higuchi, W.I.1
  • 15
    • 0025847626 scopus 로고
    • α-bisabolol, a possible safe penetration enhancer for dermal and transdermal therapeutics
    • Kadir, R. and Barry, B.W., α-Bisabolol, a possible safe penetration enhancer for dermal and transdermal therapeutics. Int. J. Pharm., 70 (1991) 87-94.
    • (1991) Int. J. Pharm. , vol.70 , pp. 87-94
    • Kadir, R.1    Barry, B.W.2
  • 16
    • 0026091719 scopus 로고
    • Lyotropic liquid crystals and the structural lipids of the stratum corneum
    • Kayali, I., Suhery, T., Friberg, S.E., Simion, F.A. and Rhein, L.D., Lyotropic liquid crystals and the structural lipids of the stratum corneum. J. Pharm. Sci., 80 (1991) 428-431.
    • (1991) J. Pharm. Sci. , vol.80 , pp. 428-431
    • Kayali, I.1    Suhery, T.2    Friberg, S.E.3    Simion, F.A.4    Rhein, L.D.5
  • 17
    • 0026763039 scopus 로고
    • Use of a model lipid matrix to demonstrate the dependence of the stratum corneum's barrier properties on its internal geometry
    • Lange-Lieckfeldt, R. and Lee, G., Use of a model lipid matrix to demonstrate the dependence of the stratum corneum's barrier properties on its internal geometry. J. Controlled Release, 20 (1992) 183-194.
    • (1992) J. Controlled Release , vol.20 , pp. 183-194
    • Lange-Lieckfeldt, R.1    Lee, G.2
  • 18
    • 0028906504 scopus 로고
    • Measuring the diffusional pathlength and area within membranes of excised human stratum corneum
    • Lieckfeldt, R. and Lee, G., Measuring the diffusional pathlength and area within membranes of excised human stratum corneum. J. Pharm. Pharmacol., 47 (1995) 26-29.
    • (1995) J. Pharm. Pharmacol. , vol.47 , pp. 26-29
    • Lieckfeldt, R.1    Lee, G.2
  • 20
    • 0016545625 scopus 로고
    • Drug permeation through human skin: Theory and in vitro experimental measurement
    • Michaels, A.S., Chandrasekaran, S.K. and Shaw, J.E., Drug permeation through human skin: theory and in vitro experimental measurement. AIChE J., 21 (1975) 985-996.
    • (1975) AIChE J. , vol.21 , pp. 985-996
    • Michaels, A.S.1    Chandrasekaran, S.K.2    Shaw, J.E.3
  • 21
    • 0029913714 scopus 로고    scopus 로고
    • A lamellar matrix model for stratum corneum intercellular lipids. I. Characterisation and comparison with stratum corneum intercellular structure
    • submitted
    • Moghimi, H.R., Williams, A.C. and Barry, B.W., A lamellar matrix model for stratum corneum intercellular lipids. I. Characterisation and comparison with stratum corneum intercellular structure. Int. J. Pharm., (1996) submitted.
    • (1996) Int. J. Pharm.
    • Moghimi, H.R.1    Williams, A.C.2    Barry, B.W.3
  • 22
    • 0015795402 scopus 로고
    • Phase transitions in phospholipid vesicles, fluorescence polarization and permeability measurements concerning the effect of temperature and cholesterol
    • Papahadjopoulos, D., Jacobson, K., Nir, S. and Isac, T., Phase transitions in phospholipid vesicles, fluorescence polarization and permeability measurements concerning the effect of temperature and cholesterol. Biochim. Biophys. Acta, 311 (1973) 330-348.
    • (1973) Biochim. Biophys. Acta , vol.311 , pp. 330-348
    • Papahadjopoulos, D.1    Jacobson, K.2    Nir, S.3    Isac, T.4
  • 23
    • 0025851987 scopus 로고
    • The influence of stratum corneum morphology on water permeability
    • Potts, R.O. and Francoeur, M.L., The influence of stratum corneum morphology on water permeability. J. Invest. Dermatol., 96 (1991) 495-499.
    • (1991) J. Invest. Dermatol. , vol.96 , pp. 495-499
    • Potts, R.O.1    Francoeur, M.L.2
  • 24
    • 0039520410 scopus 로고
    • The prediction of percutaneous penetration: A mechanistic model
    • Gurny, R. and Teubner, A. (Eds.), Wissenschaftliche Verlagsgesellschaft mbH, Stuttgart
    • Potts, R.O. and Guy, R.H., The prediction of percutaneous penetration: a mechanistic model. In Gurny, R. and Teubner, A. (Eds.), Dermal and Transdermal Drug Delivery, New Insights and Perspectives, Wissenschaftliche Verlagsgesellschaft mbH, Stuttgart, 1993, pp. 153-160.
    • (1993) Dermal and Transdermal Drug Delivery, New Insights and Perspectives , pp. 153-160
    • Potts, R.O.1    Guy, R.H.2
  • 25
    • 0023982575 scopus 로고
    • The role of protein and lipid domains in the uptake of solutes by human stratum corneum
    • Raykar, P.V., Fung, M.-C. and Anderson, B.D., The role of protein and lipid domains in the uptake of solutes by human stratum corneum. Pharm. Res., 5 (1988) 140-150.
    • (1988) Pharm. Res. , vol.5 , pp. 140-150
    • Raykar, P.V.1    Fung, M.-C.2    Anderson, B.D.3
  • 29
    • 85023279147 scopus 로고
    • Permeability of lipophilic molecules
    • Bonting, S.L. and de Pont, J.J.H.H.M. (Eds.), Elsevier/North-Holland Biomedical Press, Amsterdam
    • Stein, W.D., Permeability of lipophilic molecules. In Bonting, S.L. and de Pont, J.J.H.H.M. (Eds.), Membrane Transport, Elsevier/North-Holland Biomedical Press, Amsterdam, 1981, pp. 1-28. Tojo, K., Random brick model for drug transport across stratum corneum. J. Pharm. Sci., 76 (1987) 889-891.
    • (1981) Membrane Transport , pp. 1-28
    • Stein, W.D.1
  • 30
    • 0023513926 scopus 로고
    • Random brick model for drug transport across stratum corneum
    • Stein, W.D., Permeability of lipophilic molecules. In Bonting, S.L. and de Pont, J.J.H.H.M. (Eds.), Membrane Transport, Elsevier/North-Holland Biomedical Press, Amsterdam, 1981, pp. 1-28. Tojo, K., Random brick model for drug transport across stratum corneum. J. Pharm. Sci., 76 (1987) 889-891.
    • (1987) J. Pharm. Sci. , vol.76 , pp. 889-891
    • Tojo, K.1
  • 31
    • 0025858199 scopus 로고
    • The enhancement index concept applied to terpene penetration enhancers for human skin and model lipophilic (oestradiol) and hydrophilic (5-fluorouracil) drugs
    • Williams, A.C. and Barry, B.W., The enhancement index concept applied to terpene penetration enhancers for human skin and model lipophilic (oestradiol) and hydrophilic (5-fluorouracil) drugs. Int. J. Pharm., 74 (1991a) 157-168.
    • (1991) Int. J. Pharm. , vol.74 , pp. 157-168
    • Williams, A.C.1    Barry, B.W.2
  • 32
    • 0025961840 scopus 로고
    • Terpenes and the lipid-protein-partitioning theory of skin penetration enhancement
    • Williams, A.C. and Barry, B.W., Terpenes and the lipid-protein-partitioning theory of skin penetration enhancement. Pharm. Res., 8 (1991b) 17-24.
    • (1991) Pharm. Res. , vol.8 , pp. 17-24
    • Williams, A.C.1    Barry, B.W.2
  • 33
    • 0026743238 scopus 로고
    • On the non-Gaussian distribution of human skin permeabilities
    • Williams, A.C., Cornwell, P.A. and Barry, B.W., On the non-Gaussian distribution of human skin permeabilities. Int. J. Pharm., 86 (1992) 69-77.
    • (1992) Int. J. Pharm. , vol.86 , pp. 69-77
    • Williams, A.C.1    Cornwell, P.A.2    Barry, B.W.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.