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Volumn 19, Issue 6, 2006, Pages 336-342

Percutaneous absorption of steroids: Determination of in vitro permeability and tissue reservoir characteristics in human skin layers

Author keywords

Absorption kinetics, steroids; Maximum flux, steroids; Tissue accumulation, steroids; Topical steroids; Transdermal penetration, steroids

Indexed keywords

ALDOSTERONE; CORTICOSTERONE; HYDROCORTISONE; PROGESTERONE; STEROID; TESTOSTERONE;

EID: 33751336852     PISSN: 16605527     EISSN: None     Source Type: Journal    
DOI: 10.1159/000095254     Document Type: Article
Times cited : (51)

References (23)
  • 2
    • 0024803965 scopus 로고
    • Percutaneous absorption of steroids: Relative contributions of epidermal penetration and dermal clearance
    • Siddiqui O, Roberts MS, Polack AE: Percutaneous absorption of steroids: relative contributions of epidermal penetration and dermal clearance. J Pharmacokinet Biopharm 1989;17:405-424.
    • (1989) J Pharmacokinet Biopharm , vol.17 , pp. 405-424
    • Siddiqui, O.1    Roberts, M.S.2    Polack, A.E.3
  • 3
    • 1342272343 scopus 로고
    • Percutaneous absorption of hydrocortisone in two human subjects
    • Malkinson F, Ferguson E: Percutaneous absorption of hydrocortisone in two human subjects. J Invest Dermatol 1955;25:281-283.
    • (1955) J Invest Dermatol , vol.25 , pp. 281-283
    • Malkinson, F.1    Ferguson, E.2
  • 5
    • 0004652987 scopus 로고
    • The influence of solubility, protein binding, and percutaneous absorption on reservoir formation in skin
    • Miselnicky S, Lichtin J, Sakar A, Bronough RL: Th e influence of solubility, protein binding, and percutaneous absorption on reservoir formation in skin. J Soc Cosmet Chem 1988;39:169-177.
    • (1988) J Soc Cosmet Chem , vol.39 , pp. 169-177
    • Miselnicky, S.1    Lichtin, J.2    Sakar, A.3    Bronough, R.L.4
  • 6
    • 0034950532 scopus 로고    scopus 로고
    • An experimental approach to study the binding properties of vitamin e (alpha-tocopherol) during hairless mouse skin permeation
    • (Tokyo)
    • Lee A, Tojo K: An experimental approach to study the binding properties of vitamin E (alpha-tocopherol) during hairless mouse skin permeation. Chem Pharm Bull (Tokyo) 2001;49:659-663.
    • (2001) Chem Pharm Bull , vol.49 , pp. 659-663
    • Lee, A.1    Tojo, K.2
  • 7
    • 0016619618 scopus 로고
    • Comparative bioavailability and activity of proprietary topical corticosteroid preparations: Vasoconstrictor assays on thirty-one ointments
    • Barry BW, Woodford R: Comparative bioavailability and activity of proprietary topical corticosteroid preparations: vasoconstrictor assays on thirty-one ointments. Br J Dermatol 1975;93:63-71.
    • (1975) Br J Dermatol , vol.93 , pp. 63-71
    • Barry, B.W.1    Woodford, R.2
  • 8
    • 1342301603 scopus 로고    scopus 로고
    • Factors aff ecting the formation of a skin reservoir for topically applied solutes
    • Roberts MS, Cross SE, Anissimov YG: Factors aff ecting the formation of a skin reservoir for topically applied solutes. Skin Pharmacol Physiol 2004;17:3-16.
    • (2004) Skin Pharmacol Physiol , vol.17 , pp. 3-16
    • Roberts, M.S.1    Cross, S.E.2    Anissimov, Y.G.3
  • 9
    • 2342599148 scopus 로고    scopus 로고
    • Molecular size as the main determinant of solute maximum flux across the skin
    • Magnusson BM, Anissimov YG, Cross SE, Roberts MS: Molecular size as the main determinant of solute maximum flux across the skin. J Invest Dermatol 2004;122:993-999.
    • (2004) J Invest Dermatol , vol.122 , pp. 993-999
    • Magnusson, B.M.1    Anissimov, Y.G.2    Cross, S.E.3    Roberts, M.S.4
  • 11
    • 0032720217 scopus 로고    scopus 로고
    • Diffusion modelling of percutaneous absorption kinetics. 1. Effects of flow rate, receptor sampling rate and viable epidermal resistance for a constant donor concentration
    • Anissimov YG, Roberts MS: Diffusion modelling of percutaneous absorption kinetics. 1. Effects of flow rate, receptor sampling rate and viable epidermal resistance for a constant donor concentration. J Pharm Sci 1999;88:1201-1209.
    • (1999) J Pharm Sci , vol.88 , pp. 1201-1209
    • Anissimov, Y.G.1    Roberts, M.S.2
  • 12
    • 0032835415 scopus 로고    scopus 로고
    • A physiological pharmacokinetic model for solute disposition in tissues below a topical application site
    • Roberts MS, Cross SE: A physiological pharmacokinetic model for solute disposition in tissues below a topical application site. Pharm Res 1999;16:1392-1398.
    • (1999) Pharm Res , vol.16 , pp. 1392-1398
    • Roberts, M.S.1    Cross, S.E.2
  • 13
    • 0037960270 scopus 로고    scopus 로고
    • Determination of the eff ect of lipophilicity on the in vitro permeability and tissue reservoir characteristics of topically applied solutes in human skin layers
    • Cross SE, Magnusson BM, Anissimov YG, Winckle G, Roberts MS: Determination of the eff ect of lipophilicity on the in vitro permeability and tissue reservoir characteristics of topically applied solutes in human skin layers. J Invest Dermatol 2003;120:759-764.
    • (2003) J Invest Dermatol , vol.120 , pp. 759-764
    • Cross, S.E.1    Magnusson, B.M.2    Anissimov, Y.G.3    Winckle, G.4    Roberts, M.S.5
  • 14
    • 0002246502 scopus 로고
    • Preparation of isolated sheets of human stratum corneum
    • Kligman A, Christophers E: Preparation of isolated sheets of human stratum corneum. Arch Dermatol 1963;88:702-704.
    • (1963) Arch Dermatol , vol.88 , pp. 702-704
    • Kligman, A.1    Christophers, E.2
  • 15
    • 0034868376 scopus 로고    scopus 로고
    • Probing the effect of vehicles on topical delivery: Understanding the basic relationship between solvent and solute penetration using silicone membranes
    • Cross SE, Pugh WJ, Hadgraft J, Roberts MS: Probing the effect of vehicles on topical delivery: understanding the basic relationship between solvent and solute penetration using silicone membranes. Pharm Res 2001;18:999-1005.
    • (2001) Pharm Res , vol.18 , pp. 999-1005
    • Cross, S.E.1    Pugh, W.J.2    Hadgraft, J.3    Roberts, M.S.4
  • 17
    • 0023819029 scopus 로고
    • 14C]diazepam across isolated hairless mouse stratum corneum/epidermal tissues
    • 14C]diazepam across isolated hairless mouse stratum corneum/epidermal tissues. J Invest Dermatol 1988;90:317-319.
    • (1988) J Invest Dermatol , vol.90 , pp. 317-319
    • Koch, R.1    Palicharla, P.2    Groves, M.J.3
  • 18
    • 0033995212 scopus 로고    scopus 로고
    • Epidermal permeability-penetrant structure relationships: 4, QSAR of permeant diff usion across human stratum corneum in terms of molecular weight, H-bonding and electronic charge
    • Pugh WJ, Degim IT, Hadgraft J: Epidermal permeability-penetrant structure relationships: 4, QSAR of permeant diff usion across human stratum corneum in terms of molecular weight, H-bonding and electronic charge. Int J Pharm 2000;197:203-211.
    • (2000) Int J Pharm , vol.197 , pp. 203-211
    • Pugh, W.J.1    Degim, I.T.2    Hadgraft, J.3
  • 19
    • 0023701378 scopus 로고
    • Heterogeneity effects on permeability-partition coefficient relationships in human stratum corneum
    • Anderson B, Higuchi W, Raykar PV: Heterogeneity effects on permeability-partition coefficient relationships in human stratum corneum. Pharm Res 1988;5:566-573.
    • (1988) Pharm Res , vol.5 , pp. 566-573
    • Anderson, B.1    Higuchi, W.2    Raykar, P.V.3
  • 20
    • 0017332794 scopus 로고
    • The binding of topically applied glucocorticoids to rat skin
    • Baker J, Christian R, Simpson P: The binding of topically applied glucocorticoids to rat skin. Br J Dermatol 1977;96:171-178.
    • (1977) Br J Dermatol , vol.96 , pp. 171-178
    • Baker, J.1    Christian, R.2    Simpson, P.3
  • 21
    • 0028006643 scopus 로고
    • Transport of beta-estradiol in freshly excised human skin in vitro: Diffusion and metabolism in each skin layer
    • Liu P, Higuchi W, Ghanem AH, Good WR: Transport of beta-estradiol in freshly excised human skin in vitro: diffusion and metabolism in each skin layer. Pharm Res 1994;11:1777-1784.
    • (1994) Pharm Res , vol.11 , pp. 1777-1784
    • Liu, P.1    Higuchi, W.2    Ghanem, A.H.3    Good, W.R.4
  • 22
  • 23
    • 0030440956 scopus 로고    scopus 로고
    • Local deep tissue penetration of compounds after dermal application: Structure-tissue penetration relationships
    • Singh P, Roberts MS: Local deep tissue penetration of compounds after dermal application: structure-tissue penetration relationships. J Pharmacol Exp Ther 1996;279:908-917.
    • (1996) J Pharmacol Exp Ther , vol.279 , pp. 908-917
    • Singh, P.1    Roberts, M.S.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.