Characterization of peripheral human cannabinoid receptor (hCB2) expression and pharmacology using a novel radioligand, [35S]Sch225336

Journal of Biological Chemistry

Volumn 281, Issue 38, 2006, Pages 28143-28151

  Gonsiorek, Waldemar ^a   Hesk, David ^a   Chen, Shu Cheng ^a   Kinsley, David ^a   Fine, Jay S ^a   Jackson, James V ^a   Bober, Loretta A ^a   Deno, Gregory ^a   Bian, Hong ^a   Fossetta, James ^a   Lunn, Charles A ^a   Kozlowski, Joseph A ^a   Lavey, Brian ^a   Piwinski, John ^a   Narula, Satwant K ^a   Lundell, Daniel J ^a   Hipkin, R William ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AMINES; ANTIBODIES; BIOCHEMISTRY; CARBOXYLIC ACIDS; METHANE;

CANNABINOID RECEPTOR; HEMOPOIETIC CELLS; PHARMACOLOGY; PRIMARY AMINES;

CELLS;

CANNABINOID 1 RECEPTOR; CANNABINOID 2 RECEPTOR; N [1S [4 [[4 METHOXY 2 [(4 METHOXYPHENYL)SULFONYL]PHENYL]SULFONYL]ETHYL]METHANE SULFONAMIDE; RADIOLIGAND; SCH 225336; SULFONAMIDE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; AUTORADIOGRAPHY; BINDING AFFINITY; CONTROLLED STUDY; DRUG MECHANISM; DRUG SYNTHESIS; HUMAN; HUMAN CELL; HUMAN TISSUE; IMMUNOBLOTTING; NONHUMAN; PRIORITY JOURNAL; PROTEIN ANALYSIS; PROTEIN EXPRESSION;

ANIMALS; AUTORADIOGRAPHY; BLOTTING, WESTERN; CHO CELLS; CRICETINAE; HL-60 CELLS; HUMANS; LYMPHOCYTES; RADIOLIGAND ASSAY; RECEPTOR, CANNABINOID, CB2; SPLEEN; SULFONAMIDES;

EID: 33748780355     PISSN: 00219258     EISSN: 1083351X     Source Type: Journal    
DOI: 10.1074/jbc.M602364200     Document Type: Article

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