The synthesis of triazolothiadiazines and thiadiazoles from 1,2-bis-(4-amino-5-mercapto-1,2,4-triazol-3-yl)-ethanol and ethane

Phosphorus, Sulfur and Silicon and the Related Elements

Volumn 181, Issue 10, 2006, Pages 2361-2371

  Moustafa, A H ^a   Haggam, R A ^a   Younes, M E ^a   El Ashry, E S H ^b  

^a Zagazig University   (Egypt)

^b Alexandria University Faculty Of Science   (Egypt)

Author keywords

1,2,4 Triazole; Antimicrobial activity; Malic acid; seco C nucleosides; Succinic acid; Triazolo 3,4 b 1,3,4 thiadiazole; Triazolo 3,4 b 1,3,4 thiadiazine

Indexed keywords

EID: 33748639896     PISSN: 10426507     EISSN: 15635325     Source Type: Journal    
DOI: 10.1080/10426500600634681     Document Type: Article

References (34)

1. (a) K. A. Watanabe, In Chemistry of nucleosides and nucleotides, Ed. L. B. Townsend (Plenum Press, New York, Vol. 3, p. 421, 1994);
2. (b) S. Hanessian and A. G. Pernet, Adv. Carbohydr. Chem. Biochem., 33 111 (1976);
3. (c) U. Hacksell and G. D. Daves, Progr. Med. Chem., 22, 2 (1985);
4. (d) C. K. Chu, P. M. El-Kabbani, and B. B. Thompson, Nucleosides Nucleotides, 3, 1 (1984).
5. (a) E. S. H. El Ashry and Y. El Kilany, Adv. Heterocycl. Chem., 67, 391 (1995);
6. (b) E. S. H. El Ashry, and Y. El Kilany, Adv. Heterocycl. Chem., 68, 1 (1997);
7. (c) E. S. H. El Ashry, and Y. El Kilany, Adv. Heterocycl. Chem., 69, 1295 (1998).
8. (a) J. T. Witkowski, R. K. Robins, R. W. Sidwell, and L. N. Simon, J. Med. Chem., 15, 1150 (1972);
9. (b) R. W. Sidwell, J. H. Huffman, G. P. Khare, L. B. Allen, J. T. Witkowski and R. K. Robins, Science, 177, 705 (1972).
10. B. W. Dymock, P. S. Jones, and F. X. Wilson, Antiviral Chem., Chemotherapy, 11(2), 79 (2000).
11. (a) G. Just and M. Ramjeesingh, Tetrahedron Lett., 985 (1975);
12. (b) T. Huynh-Dinh, J. Igolen, E. Bisagni, J. P. Marquet, and A. Civier, J. Chem. Soc. Perkin Trans 1, 1, 761 (1977);
13. (c) M. S. Poonian, and E. F. Vowoswiat, J. Org. Chem., 45, 203 (1980);
14. (d) M. S. Poonian and E. F. Vowoswiat, J. Org. Chem., 42, 1109 (1977).
15. (a) E. S. H. El Ashry, N. Rashed, M. Taha, and E. Ramadan, Adv. Heterocycl. Chem., 59, 39 (1994);
16. (b) E. S. H. El Ashry, N. Rashed, A. Mousaad, and E. Ramadan, Adv. Heterocycl. Chem., 61, 207 (1994)
17. (c) M. A. El-Saadani, B. A. B. El-Gamal, G. I. El Kholy, M. El Sayed, and E. S. H. El Ashry, J. Med. Res. Inst., 14, 293 (1993);
18. (d) B. A. B. El-Gamal, M. A. El-Saadani, E. K. A. El Sayed, M. M. El Sayed, and E. S. H. El Ashry, J. Med. Res. Inst., 15, 119 (1994);
19. (e) A. Mousaad, H. Abdel Hamid, A. El Nemer, and E. S. H. El Ashry, Bull. Chem. Soc. Jap., 65, 546 (1992);
20. (f) N. Rashed, A. El Nemer, and E. S. H. El Ashry, Arch. Pharm., 326, 153 (1992).
21. (a) S. Bala, R. P. Gupta, M. L. Sachdeva, A. Singh, and H. K. Puraji, Indian J. Chem., 16B, 481 (1978);
22. (b) S. W. Xiao, X.-P. Hu, C. H. Chu, and Z.-Y. Zhang, Indian J. Chem., 39B, 779 (2000).
23. (a) M. M. Ghorab, A.M. Sh. El-Sharief, Y. A. Ammar, and Sh. I. Mohamed, Farmaco, 55, 354 (2000);
24. (b) B. S. Holla, R. Gonsalves, and S. Shenoy, Farmaco, 53, 574 (1998).
25. L. F. Awad and E. S. H. El Ashry, Carbohydr. Res., 312, 9 (1998).
26. E. S. H. El Ashry, and L. F. Awad, Nucleosides, Nucleotides, and Nucleic Acids, 20, 901 (2001).
27. (a) E. S. H. El Ashry and L. F. Awad, Nucleosides, Nucleotides, and Nucleic Acids 20, 103 (2001);
28. (b) E. S. H. El Ashry, L. F. Awad, H. M. Abdel-Hamid, and A. I. Atta, In Int. Soc. for Nucleosides, Nucleotides, and Nucleic Acids, XVI Int. Round Table 5, Minneapolis, Minnesota, USA (2004).
29. E. S. H. El Ashry, N. Rashed, and A. H. Shobier, Pharmazie, 55, 251 (2000).
30. E. S. H. El Ashry, N. Rashed, and A. H. Shobier, Pharmazie 55, 331 (2000).
31. E. S. H. El Ashry, N. Rashed, N and A. H. Shobier, Pharmazie, 56, 403 (2000).
32. M. Balbaa, H. Mansour, H. El-Sawy, and E. S. H. El Ashry, Nucleosides, Nucleotides, and Nucleic Acids, 21, 695 (2002).
33. A. H. Moustafa, R. A. Haggam, M. E. Younes, and E. S. H. El Ashry, Nucleosides, Nucleotides, and Nucleic Acids, 24, 1885 (2005).
34. D. S. Reeves, and L. O. White, Principles methods of assaying antibiotic in pharmaceutical microbiology, 3rd ed., p. 140 (Blackwell Scientific, Oxford, 1983).