Multiple receptor states are required to describe both kinetic binding and activation of neutrophils via N-formyl peptide receptor ligands

Cellular Signalling

Volumn 18, Issue 10, 2006, Pages 1732-1747

  Kinzer Ursem, Tamara L ^a   Sutton, Karyn L ^a,b   Waller, Anna ^a   Omann, Geneva M ^b,c   Linderman, Jennifer J ^a  

^a UNIVERSITY OF MICHIGAN   (United States)

^b UNIVERSITY OF MICHIGAN MEDICAL SCHOOL   (United States)

^c VETERANS AFFAIRS MEDICAL CENTER   (United States)

Author keywords

Actin; Agonism; fMLP receptor; Internalization; Kinetic rate constants; Leukocyte; Mathematical model; Oxidant; Potency; Upregulation

Indexed keywords

FORMYLPEPTIDE RECEPTOR; GUANINE NUCLEOTIDE BINDING PROTEIN; LIGAND;

ACTIN POLYMERIZATION; ARTICLE; CONFORMATIONAL TRANSITION; CONTROLLED STUDY; HUMAN; INTERNALIZATION; LEUKOCYTE ACTIVATION; MATHEMATICAL MODEL; MOLECULAR DYNAMICS; OXIDATION KINETICS; PRIORITY JOURNAL; RECEPTOR AFFINITY; RECEPTOR BINDING; RECEPTOR INTRINSIC ACTIVITY; RECEPTOR OCCUPANCY; UPREGULATION;

ACTINS; HUMANS; KINETICS; LIGANDS; N-FORMYLMETHIONINE LEUCYL-PHENYLALANINE; NEUTROPHIL ACTIVATION; NEUTROPHILS; PROTEIN BINDING; PROTEIN CONFORMATION; PROTEIN TRANSPORT; RECEPTORS, FORMYL PEPTIDE; SIGNAL TRANSDUCTION; TEMPERATURE; TIME FACTORS;

EID: 33747213361     PISSN: 08986568     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.cellsig.2006.01.014     Document Type: Article

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