메뉴 건너뛰기




Volumn 33, Issue 5, 2006, Pages 599-605

Imaging of aromatase distribution in rat and rhesus monkey brains with [11C]vorozole

Author keywords

Amygdala; Aromatase; Hypothalamus; Positron emission tomography; Sex steroids; Vorozole

Indexed keywords

AROMATASE; AROMATASE INHIBITOR; RADIOPHARMACEUTICAL AGENT; UNCLASSIFIED DRUG; VOROZOLE; VOROZOLE C 11;

EID: 33745825511     PISSN: 09698051     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.nucmedbio.2006.03.009     Document Type: Article
Times cited : (43)

References (33)
  • 1
    • 0030174660 scopus 로고    scopus 로고
    • A review of brain aromatase cytochrome P450
    • Lephart E.D. A review of brain aromatase cytochrome P450. Brain Res Brain Res Rev 22 (1996) 1-26
    • (1996) Brain Res Brain Res Rev , vol.22 , pp. 1-26
    • Lephart, E.D.1
  • 2
    • 0031983425 scopus 로고    scopus 로고
    • Anatomic distribution and regulation of aromatase gene expression in the rat brain
    • Roselli C.E., Abdelgadir S.E., Ronnekleiv O.K., and Klosterman S.A. Anatomic distribution and regulation of aromatase gene expression in the rat brain. Biol Reprod 58 (1998) 79-87
    • (1998) Biol Reprod , vol.58 , pp. 79-87
    • Roselli, C.E.1    Abdelgadir, S.E.2    Ronnekleiv, O.K.3    Klosterman, S.A.4
  • 3
    • 0032507727 scopus 로고    scopus 로고
    • The effect of anabolic-androgenic steroids on aromatase activity and androgen receptor binding in the rat preoptic area
    • Roselli C.E. The effect of anabolic-androgenic steroids on aromatase activity and androgen receptor binding in the rat preoptic area. Brain Res 792 (1998) 271-276
    • (1998) Brain Res , vol.792 , pp. 271-276
    • Roselli, C.E.1
  • 4
    • 0029977498 scopus 로고    scopus 로고
    • Distribution and steroid hormone regulation of aromatase mRNA expression in the forebrain of adult male and female rats: a cellular-level analysis using in situ hybridization
    • Wagner C.K., and Morrell J.I. Distribution and steroid hormone regulation of aromatase mRNA expression in the forebrain of adult male and female rats: a cellular-level analysis using in situ hybridization. J Comp Neurol 370 (1996) 71-84
    • (1996) J Comp Neurol , vol.370 , pp. 71-84
    • Wagner, C.K.1    Morrell, J.I.2
  • 5
    • 0027175248 scopus 로고
    • Brain aromatase and the control of male sexual behavior
    • Balthazart J., and Foidart A. Brain aromatase and the control of male sexual behavior. J Steroid Biochem Mol Biol 44 (1993) 521-540
    • (1993) J Steroid Biochem Mol Biol , vol.44 , pp. 521-540
    • Balthazart, J.1    Foidart, A.2
  • 7
    • 0028047993 scopus 로고
    • Effects of steroidal and non steroidal aromatase inhibitors on sexual behavior and aromatase-immunoreactive cells and fibers in the quail brain
    • Foidart A., Harada N., and Balthazart J. Effects of steroidal and non steroidal aromatase inhibitors on sexual behavior and aromatase-immunoreactive cells and fibers in the quail brain. Brain Res 657 (1994) 105-123
    • (1994) Brain Res , vol.657 , pp. 105-123
    • Foidart, A.1    Harada, N.2    Balthazart, J.3
  • 8
    • 0029042444 scopus 로고
    • Aromatase-immunoreactive cells are present in mouse brain areas that are known to express high levels of aromatase activity
    • Foidart A., Harada N., and Balthazart J. Aromatase-immunoreactive cells are present in mouse brain areas that are known to express high levels of aromatase activity. Cell Tissue Res 280 (1995) 561-574
    • (1995) Cell Tissue Res , vol.280 , pp. 561-574
    • Foidart, A.1    Harada, N.2    Balthazart, J.3
  • 9
    • 0029872885 scopus 로고    scopus 로고
    • Effect of vorozole, an aromatase enzyme inhibitor, on sexual behavior, aromatase activity and neural immunoreactivity
    • Rissman E.F., Harada N., and Roselli C.E. Effect of vorozole, an aromatase enzyme inhibitor, on sexual behavior, aromatase activity and neural immunoreactivity. J Neuroendocrinol 8 (1996) 199-210
    • (1996) J Neuroendocrinol , vol.8 , pp. 199-210
    • Rissman, E.F.1    Harada, N.2    Roselli, C.E.3
  • 10
    • 0344795782 scopus 로고
    • Inhibitors of steroid biosynthesis
    • Sandler M., and Harold J. (Eds), Oxford University Press, Oxford
    • Brodie A.M.H. Inhibitors of steroid biosynthesis. In: Sandler M., and Harold J. (Eds). Design of enzyme inhibitors as drugs (1994), Oxford University Press, Oxford 503-522
    • (1994) Design of enzyme inhibitors as drugs , pp. 503-522
    • Brodie, A.M.H.1
  • 11
    • 0027983894 scopus 로고
    • Vorozole, a specific non-steroidal aromatase inhibitor
    • Wouters W., Snoeck E., and De Coster R. Vorozole, a specific non-steroidal aromatase inhibitor. Breast Cancer Res Treat 30 (1994) 89-94
    • (1994) Breast Cancer Res Treat , vol.30 , pp. 89-94
    • Wouters, W.1    Snoeck, E.2    De Coster, R.3
  • 13
    • 0029560237 scopus 로고
    • In vivo measurement of aromatase inhibition by letrozole (CGS 20267) in postmenopausal patients with breast cancer
    • Dowsett M., Jones A., Johnston S.R., Jacobs S., Trunet P., and Smith I.E. In vivo measurement of aromatase inhibition by letrozole (CGS 20267) in postmenopausal patients with breast cancer. Clin Cancer Res 1 (1995) 1511-1515
    • (1995) Clin Cancer Res , vol.1 , pp. 1511-1515
    • Dowsett, M.1    Jones, A.2    Johnston, S.R.3    Jacobs, S.4    Trunet, P.5    Smith, I.E.6
  • 17
    • 10044226276 scopus 로고    scopus 로고
    • Diminished aromatase immunoreactivity in the hypothalamus, but not in the basal forebrain nuclei in Alzheimer's disease
    • Ishunina T.A., van Beurden D., van der Meulen G., Unmehopa U.A., Hol E.M., Huitinga I., et al. Diminished aromatase immunoreactivity in the hypothalamus, but not in the basal forebrain nuclei in Alzheimer's disease. Neurobiol Aging 26 (2005) 173-194
    • (2005) Neurobiol Aging , vol.26 , pp. 173-194
    • Ishunina, T.A.1    van Beurden, D.2    van der Meulen, G.3    Unmehopa, U.A.4    Hol, E.M.5    Huitinga, I.6
  • 18
    • 0032808422 scopus 로고    scopus 로고
    • Quantitative autoradiography with short-lived positron emission tomography tracers: a study on muscarinic acetylcholine receptors with N-[(11)C]methyl-4-piperidylbenzilate
    • Sihver S., Sihver W., Bergström M., Höglund A.U., Sjöberg P., Långström B., et al. Quantitative autoradiography with short-lived positron emission tomography tracers: a study on muscarinic acetylcholine receptors with N-[(11)C]methyl-4-piperidylbenzilate. J Pharmacol Exp Ther 290 (1999) 917-922
    • (1999) J Pharmacol Exp Ther , vol.290 , pp. 917-922
    • Sihver, S.1    Sihver, W.2    Bergström, M.3    Höglund, A.U.4    Sjöberg, P.5    Långström, B.6
  • 20
    • 0031120073 scopus 로고    scopus 로고
    • Neuroanatomical distribution of aromatase mRNA in the rat brain: indications of regional regulation
    • Wagner C.K., and Morrell J.I. Neuroanatomical distribution of aromatase mRNA in the rat brain: indications of regional regulation. J Steroid Biochem Mol Biol 61 (1997) 307-314
    • (1997) J Steroid Biochem Mol Biol , vol.61 , pp. 307-314
    • Wagner, C.K.1    Morrell, J.I.2
  • 21
    • 0022348964 scopus 로고
    • Distribution and regulation of aromatase activity in the rat hypothalamus and limbic system
    • Roselli C.E., Horton L.E., and Resko J.A. Distribution and regulation of aromatase activity in the rat hypothalamus and limbic system. Endocrinology 117 (1985) 2471-2477
    • (1985) Endocrinology , vol.117 , pp. 2471-2477
    • Roselli, C.E.1    Horton, L.E.2    Resko, J.A.3
  • 22
    • 0021335635 scopus 로고
    • Regulation of brain aromatase activity in rats
    • Roselli C.E., Ellinwood W.E., and Resko J.A. Regulation of brain aromatase activity in rats. Endocrinology 114 (1984) 192-200
    • (1984) Endocrinology , vol.114 , pp. 192-200
    • Roselli, C.E.1    Ellinwood, W.E.2    Resko, J.A.3
  • 23
    • 0023512293 scopus 로고
    • The distribution and regulation of aromatase activity in the central nervous system
    • Roselli C.E., and Resko J.A. The distribution and regulation of aromatase activity in the central nervous system. Steroids 50 (1987) 495-508
    • (1987) Steroids , vol.50 , pp. 495-508
    • Roselli, C.E.1    Resko, J.A.2
  • 24
    • 0025797245 scopus 로고
    • Sex differences in androgen receptors and aromatase activity in microdissected regions of the rat brain
    • Roselli C.E. Sex differences in androgen receptors and aromatase activity in microdissected regions of the rat brain. Endocrinology 128 (1991) 1310-1316
    • (1991) Endocrinology , vol.128 , pp. 1310-1316
    • Roselli, C.E.1
  • 25
    • 0030726669 scopus 로고    scopus 로고
    • Regulation of aromatase gene expression in the adult rat brain
    • Roselli C.E., Abdelgadir S.E., and Resko J.A. Regulation of aromatase gene expression in the adult rat brain. Brain Res Bull 44 (1997) 351-357
    • (1997) Brain Res Bull , vol.44 , pp. 351-357
    • Roselli, C.E.1    Abdelgadir, S.E.2    Resko, J.A.3
  • 26
    • 0029056146 scopus 로고
    • A molecular model for the interaction between vorozole and other non-steroidal inhibitors and human cytochrome P450 19 (P450 aromatase)
    • Koymans L.M., Moereels H., and Vanden Bossche H. A molecular model for the interaction between vorozole and other non-steroidal inhibitors and human cytochrome P450 19 (P450 aromatase). J Steroid Biochem Mol Biol 53 (1995) 191-197
    • (1995) J Steroid Biochem Mol Biol , vol.53 , pp. 191-197
    • Koymans, L.M.1    Moereels, H.2    Vanden Bossche, H.3
  • 27
    • 0025257480 scopus 로고
    • Aromatase inhibition by R 76 713: a kinetic analysis in rat ovarian homogenates
    • Krekels M.D., Wouters W., and De Coster R. Aromatase inhibition by R 76 713: a kinetic analysis in rat ovarian homogenates. Steroids 55 (1990) 69-73
    • (1990) Steroids , vol.55 , pp. 69-73
    • Krekels, M.D.1    Wouters, W.2    De Coster, R.3
  • 28
    • 0025727599 scopus 로고
    • Aromatase in the human choriocarcinoma JEG-3: inhibition by R 76 713 in cultured cells and in tumors grown in nude mice
    • Krekels M.D., Wouters W., De Coster R., Van Ginckel R., Leonaers A., and Janssen P.A. Aromatase in the human choriocarcinoma JEG-3: inhibition by R 76 713 in cultured cells and in tumors grown in nude mice. J Steroid Biochem Mol Biol 38 (1991) 415-422
    • (1991) J Steroid Biochem Mol Biol , vol.38 , pp. 415-422
    • Krekels, M.D.1    Wouters, W.2    De Coster, R.3    Van Ginckel, R.4    Leonaers, A.5    Janssen, P.A.6
  • 29
    • 0025168832 scopus 로고
    • R 76713 and enantiomers: selective, nonsteroidal inhibitors of the cytochrome P450-dependent oestrogen synthesis
    • Vanden Bossche H., Willemsens G., Roels I., Bellens D., Moereels H., Coene M.C., et al. R 76713 and enantiomers: selective, nonsteroidal inhibitors of the cytochrome P450-dependent oestrogen synthesis. Biochem Pharmacol 40 (1990) 1707-1718
    • (1990) Biochem Pharmacol , vol.40 , pp. 1707-1718
    • Vanden Bossche, H.1    Willemsens, G.2    Roels, I.3    Bellens, D.4    Moereels, H.5    Coene, M.C.6
  • 30
    • 0025296956 scopus 로고
    • Potency and selectivity of the aromatase inhibitor R 76,713. A study in human ovarian, adipose stromal, testicular and adrenal cells
    • Wouters W., De Coster R., Beerens D., Doolaege R., Gruwez J.A., Van Camp K., et al. Potency and selectivity of the aromatase inhibitor R 76,713. A study in human ovarian, adipose stromal, testicular and adrenal cells. J Steroid Biochem 36 (1990) 57-65
    • (1990) J Steroid Biochem , vol.36 , pp. 57-65
    • Wouters, W.1    De Coster, R.2    Beerens, D.3    Doolaege, R.4    Gruwez, J.A.5    Van Camp, K.6
  • 31
    • 0030930389 scopus 로고    scopus 로고
    • Distribution of aromatase cytochrome P450 messenger ribonucleic acid in adult rhesus monkey brains
    • Abdelgadir S.E., Roselli C.E., Choate J.V., and Resko J.A. Distribution of aromatase cytochrome P450 messenger ribonucleic acid in adult rhesus monkey brains. Biol Reprod 57 (1997) 772-777
    • (1997) Biol Reprod , vol.57 , pp. 772-777
    • Abdelgadir, S.E.1    Roselli, C.E.2    Choate, J.V.3    Resko, J.A.4
  • 32
    • 0027269413 scopus 로고
    • Aromatase activity in the rat brain: hormonal regulation and sex differences
    • Roselli C.E., and Resko J.A. Aromatase activity in the rat brain: hormonal regulation and sex differences. J Steroid Biochem Mol Biol 44 (1993) 499-508
    • (1993) J Steroid Biochem Mol Biol , vol.44 , pp. 499-508
    • Roselli, C.E.1    Resko, J.A.2
  • 33
    • 0023546559 scopus 로고
    • Genetic evidence for androgen-dependent and independent control of aromatase activity in the rat brain
    • Roselli C.E., Salisbury R.L., and Resko J.A. Genetic evidence for androgen-dependent and independent control of aromatase activity in the rat brain. Endocrinology 121 (1987) 2205-2210
    • (1987) Endocrinology , vol.121 , pp. 2205-2210
    • Roselli, C.E.1    Salisbury, R.L.2    Resko, J.A.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.