Synthesis and biological evaluation of a novel structural type of serotonin 5-HT3 receptor antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 16, Issue 10, 2006, Pages 2769-2772

  Venkatesha Perumal, Ramachandran ^a   Mahesh, Radhakrishnan ^b  

^a Periyar College of Pharmaceutical Sciences for Girls   (India)

^b BIRLA INSTITUTE OF TECHNOLOGY AND SCIENCE   (India)

Author keywords

5 HT3 receptor antagonist; Quinoxalin 2 carboxamides

Indexed keywords

AMIDE; MORPHOLINE DERIVATIVE; N [3 [(4 METHYLPIPERAZIN 1 YL)METHYL] 4 HYDROXYPHENYL] 3 METHOXYQUINOXALIN 2 CARBOXAMIDE; PIPERAZINE DERIVATIVE; PIPERIDINE DERIVATIVE; PYRROLIDINE DERIVATIVE; QUINOXALINE DERIVATIVE; SEROTONIN 3 ANTAGONIST; SEROTONIN 3 RECEPTOR; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DRUG PURITY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; GUINEA PIG; ILEUM; INFRARED SPECTROSCOPY; MALE; MASS SPECTROMETRY; MICROANALYSIS; MICROWAVE IRRADIATION; MYENTERIC PLEXUS; NONHUMAN; PROTON NUCLEAR MAGNETIC RESONANCE; SUBSTITUTION REACTION;

ANIMALS; GUINEA PIGS; MALE; RECEPTORS, SEROTONIN, 5-HT3; SEROTONIN ANTAGONISTS; SPECTRUM ANALYSIS;

ANIMALIA; CAVIA PORCELLUS;

EID: 33645891154     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2006.02.006     Document Type: Article

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