Microwave assisted synthesis of 2-(4-substituted piperazin-1-yl)-1,8- naphthyridine-3-carbonitrile as a new class of serotonin 5-HT 3 receptor antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 20, 2004, Pages 5179-5181

  Mahesh, Radhakrishnan ^a   Venkatesha Perumal, Ramachandran ^a   Vijaya Pandi, Pandi ^a  

^a BIRLA INSTITUTE OF TECHNOLOGY AND SCIENCE   (India)

Author keywords

1,8 Naphthyridine; Serotonin 5 HT3 antagonists

Indexed keywords

ALDEHYDE DERIVATIVE; CYANIDE; PIPERIDINE; SEROTONIN 3 ANTAGONIST;

ANIMAL TISSUE; ARTICLE; DRUG SYNTHESIS; GUINEA PIG; HEATING; ILEUM; MALE; MICROWAVE IRRADIATION; MYENTERIC PLEXUS; NONHUMAN;

ANIMALS; GUINEA PIGS; ILEUM; MALE; MICROWAVES; MUSCLE CONTRACTION; MUSCLE, SMOOTH; MYENTERIC PLEXUS; NAPHTHYRIDINES; NEUROMUSCULAR JUNCTION; NITRILES; PIPERAZINES; RECEPTORS, SEROTONIN, 5-HT3; SEROTONIN ANTAGONISTS; STRUCTURE-ACTIVITY RELATIONSHIP;

CAVIA PORCELLUS; SUS SCROFA;

EID: 4544258286     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.07.060     Document Type: Article

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