HIV-1 integrase inhibition by pyrrole/imidazole-containing polyamides

Journal of Peptide Research

Volumn 66, Issue SUPPL. 1, 2005, Pages 138-145

  Zakharova, O D ^a   Baranova, S ^a   Parissi, V ^b,c,d   Ryabinin, V A ^a   Sinyakov, A N ^a   Litvak, S ^b,c,d   Litvak, L T ^b,c,d   Nevinsky, G A ^a  

^a INSTITUTE OF CHEMICAL BIOLOGY AND FUNDAMENTAL MEDICINE   (Russian Federation)

^b University Victor Segalen   (France)

^c UNIVERSITÉ DE BORDEAUX   (France)

^d IFR 66 Pathologies Infectieuses et Cancers   (France)

Author keywords

DNA minor groove binders; HIV 1; Inhibition; Integrase; Pyrrole imidazole containing polyamides

Indexed keywords

4 AMINOBUTYRIC ACID; BETA ALANINE; DISTAMYCIN A; DNA; GLYCINE; IMIDAZOLE DERIVATIVE; INTEGRASE; INTEGRASE INHIBITOR; POLYAMIDE; PYRROLE DERIVATIVE;

AMINO ACID SEQUENCE; AMINO TERMINAL SEQUENCE; ARTICLE; BINDING AFFINITY; CARBOXY TERMINAL SEQUENCE; DRUG MECHANISM; DRUG SYNTHESIS; ENZYME ACTIVITY; ENZYME INHIBITION; INHIBITION KINETICS; PRIORITY JOURNAL;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 33645060975     PISSN: 1397002X     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1747-0285.2006.00343.x     Document Type: Article

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