SCOPUS 정보 검색 플랫폼

Volumn 58, Issue 2, 2006, Pages 209-218

Synthesis and binding profile of constrained analogues of N-[4-(4-arylpiperazin-1-yl)butyl]-3-methoxybenzamides, a class of potent dopamine D3 receptor ligands

(5) Leopoldo, Marcello a Lacivita, Enza a Colabufo, Nicola A a Berardi, Francesco a Perrone, Roberto a

a UNIVERSITY OF BARI (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

BENZAMIDE DERIVATIVE; DOPAMINE 3 RECEPTOR STIMULATING AGENT; GUANOSINE TRIPHOSPHATE; N [4 [4 (2,3 DICHLOROPHENYL) 1 PIPERAZINYL]CYCLOHEXYL] 3 METHOXYBENZAMIDE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING ASSAY; CELL LINE; CHO CELL; CIS ISOMER; COLUMN CHROMATOGRAPHY; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; NONHUMAN; PROTON NUCLEAR MAGNETIC RESONANCE; RAT; RECEPTOR AFFINITY; STRUCTURE ANALYSIS; TRANS ISOMER;

ANIMALS; BENZAMIDES; BINDING, COMPETITIVE; CELL LINE; CEREBRAL CORTEX; CHO CELLS; CRICETINAE; CRICETULUS; GUANOSINE TRIPHOSPHATE; HIPPOCAMPUS; HUMANS; LIGANDS; MALE; RADIOLIGAND ASSAY; RATS; RATS, WISTAR; RECEPTORS, DOPAMINE D3; SPIPERONE;

EID: 31544444193 PISSN: 00223573 EISSN: None Source Type: Journal
DOI: 10.1211/jpp.58.2.0008 Document Type: Article

Times cited : (13)

References (19)

1
- 0038579160
- 3 receptor function
- 3 receptor function. Nat. Med. 9: 762-767
- (2003) Nat. Med. , vol.9 , pp. 762-767
- Bezard, E.¹ Ferry, S.² Mach, U.³ Stark, H.⁴ Leriche, L.⁵ Boraud, T.⁶ Gross, C.⁷ Sokoloff, P.⁸

2
- 0036170920
- A review of pramipexole and its clinical utility in Parkinson's disease
- Biglan, K. M., Holloway, R. G. (2002) A review of pramipexole and its clinical utility in Parkinson's disease. Expert Opin. Pharmacother. 3: 197-210
- (2002) Expert Opin. Pharmacother. , vol.3 , pp. 197-210
- Biglan, K.M.¹ Holloway, R.G.²

3
- 0028978621
- 1A receptor full agonist in rat cerebral cortex
- 1A receptor full agonist in rat cerebral cortex. Naunyn Schmiedebergs Arch. Pharmacol. 352: 276-282
- (1995) Naunyn Schmiedebergs Arch. Pharmacol. , vol.352 , pp. 276-282
- Borsini, F.¹ Giraldo, E.² Monferini, E.³ Antonini, G.⁴ Parenti, M.⁵ Bietti, G.⁶ Donetti, A.⁷

4
- 15844382453
- 4 antagonists
- 4 antagonists. J. Med. Chem. 39: 1946-1948
- (1996) J. Med. Chem. , vol.39 , pp. 1946-1948
- Boyfield, I.¹ Brown, T.H.² Coldwell, M.C.³ Cooper, D.G.⁴ Hadley, M.S.⁵ Hagan, J.J.⁶ Healy, M.A.⁷ Jones, A.⁸ King, R.J.⁹ Middlemiss, D.N.¹⁰ Nash, D.J.¹¹ Riley, G.J.¹² Scott, E.E.¹³ Smith, S.A.¹⁴ Stemp, G.¹⁵

5
- 0015861774
- 50) of an enzymatic reaction
- 50) of an enzymatic reaction. Biochem. Pharmacol. 22: 3099-3108
- (1973) Biochem. Pharmacol. , vol.22 , pp. 3099-3108
- Cheng, Y.C.¹ Prusoff, W.H.²

6
- 4344614482
- Nonradioactive GTP binding assay to monitor activation of G protein-coupled receptors
- Frang, H., Mukkala, V.-M., Syystö, R., Ollikka, P., Hurskainen, P., Scheinin, M., Hemmilä, I. (2003) Nonradioactive GTP binding assay to monitor activation of G protein-coupled receptors. Assay Drug Dev. Technol. 1: 275-280
- (2003) Assay Drug Dev. Technol. , vol.1 , pp. 275-280
- Frang, H.¹ Mukkala, V.-M.² Syystö, R.³ Ollikka, P.⁴ Hurskainen, P.⁵ Scheinin, M.⁶ Hemmilä, I.⁷

7
- 0018835131
- α-adrenoceptors in rat brain: Sodium changes the affinity of agonists for prazosin sites
- Glossmann, H., Hornung, R. (1980) α-Adrenoceptors in rat brain: sodium changes the affinity of agonists for prazosin sites. Eur. J. Pharmacol. 61: 407-408
- (1980) Eur. J. Pharmacol. , vol.61 , pp. 407-408
- Glossmann, H.¹ Hornung, R.²

8
- 0037019828
- 3 receptor ligands with antagonistic properties
- 3 receptor ligands with antagonistic properties. ChemBioChem 3: 946-961
- (2002) ChemBioChem , vol.3 , pp. 946-961
- Hackling, A.E.¹ Stark, H.²

9
- 20444378913
- 3 receptors in drug addiction: A review of pharmacological evidence
- 3 receptors in drug addiction: a review of pharmacological evidence. Brain Res. Rev. 49: 77-105
- (2005) Brain Res. Rev. , vol.49 , pp. 77-105
- Heidbreder, C.A.¹ Gardner, E.L.² Xi, Z.-X.³ Thanos, P.K.⁴ Mugnaini, M.⁵ Hagan, J.J.⁶ Ashby, C.R.⁷

10
- 0037137596
- 3 receptor ligands
- 3 receptor ligands. J. Med. Chem. 45: 5727-5735
- (2002) J. Med. Chem. , vol.45 , pp. 5727-5735
- Leopoldo, M.¹ Berardi, F.² Colabufo, N.A.³ De Giorgio, P.⁴ Lacivita, E.⁵ Perrone, R.⁶ Tortorella, V.⁷

11
- 0030610305
- 3 dopamine receptor: Neurobiology and potential clinical relevance
- 3 dopamine receptor: neurobiology and potential clinical relevance. Pharmacol. Rev. 49: 231-252
- (1997) Pharmacol. Rev. , vol.49 , pp. 231-252
- Levant, B.¹

12
- 0037278185
- 3 dopamine receptor ligands as potential therapeutic agents for neurological and neuropsychiatric disorders
- 3 dopamine receptor ligands as potential therapeutic agents for neurological and neuropsychiatric disorders. Curr. Pharm. Des. 9: 643-671
- (2003) Curr. Pharm. Des. , vol.9 , pp. 643-671
- Luedtke, R.R.¹ Mach, R.H.²

13
- 0038548068
- 3 receptor antagonists
- 3 receptor antagonists. Bioorg. Med. Chem. Lett. 13: 2179-2183
- (2003) Bioorg. Med. Chem. Lett. , vol.13 , pp. 2179-2183
- Newman, A.H.¹ Cao, J.² Bennett, C.J.³ Robarge, M.J.⁴ Freeman, R.A.⁵ Luedtke, R.R.⁶

14
- 0032969297
- 1D receptors
- 1D receptors. Naunyn Schmiedebergs Arch. Pharmacol. 359: 447-453
- (1999) Naunyn Schmiedebergs Arch. Pharmacol. , vol.359 , pp. 447-453
- Newman-Tancredi, A.¹ Cussac, D.² Audinot, V.³ Millan, M.J.⁴

15
- 0030043026
- Effect of linking bridge modifications on the antipsychotic profile of some phthalimide and isoindolinone derivatives
- Norman, M. H., Minick, D. J., Rigdon, G. C. (1996) Effect of linking bridge modifications on the antipsychotic profile of some phthalimide and isoindolinone derivatives. J. Med. Chem. 39: 149-157
- (1996) J. Med. Chem. , vol.39 , pp. 149-157
- Norman, M.H.¹ Minick, D.J.² Rigdon, G.C.³

16
- 37049150114
- Aryl-2-haloalkylamines. I
- Ross, W. C. J. (1949) Aryl-2-haloalkylamines. I. J. Chem. Soc. 183-191
- (1949) J. Chem. Soc. , pp. 183-191
- Ross, W.C.J.¹

17
- 0025179967
- 3) as a target of neuroleptics
- 3) as a target of neuroleptics. Nature 347: 72-76
- (1990) Nature , vol.347 , pp. 72-76
- Sokoloff, P.¹ Giros, B.² Martres, M.P.³ Bouthenet, M.L.⁴ Schwarz, J.C.⁵

18
- 0028179609
- 4, dopamine receptors revealed in transfected neuronal cell lines
- 4, dopamine receptors revealed in transfected neuronal cell lines. Proc. Natl. Acad. Sci. USA 91: 649-653
- (1994) Proc. Natl. Acad. Sci. USA , vol.91 , pp. 649-653
- Swarzenski, B.C.¹ Tang, L.² Oh, Y.J.³ O'Malley, K.L.⁴ Todd, R.D.⁵

19
- 0035919534
- The dopamine D3 receptor partial agonist, BP 897, is an antagonist at human dopamine D3 receptors and at rat somatodendritic dopamine D3 receptors
- Wicke, K., Javier Garcia-Ladona, J. (2001) The dopamine D3 receptor partial agonist, BP 897, is an antagonist at human dopamine D3 receptors and at rat somatodendritic dopamine D3 receptors. Eur. J. Pharmacol. 424: 85-90
- (2001) Eur. J. Pharmacol. , vol.424 , pp. 85-90
- Wicke, K.¹ Javier Garcia-Ladona, J.²

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.