The dopamine D3 receptor partial agonist, BP 897, is an antagonist at human dopamine D3 receptors and at rat somatodendritic dopamine D3 receptors

European Journal of Pharmacology

Volumn 424, Issue 2, 2001, Pages 85-90

  Wicke, Karsten ^a   Garcia Ladona, Javier ^a  

^a Knoll AG   (Germany)

Author keywords

BP 897; Dopamine; Dopamine D3 receptor; Drug dependence; Electrophysiology; Functional assay

Indexed keywords

2 DIPROPYLAMINO 7 HYDROXYTETRALIN; 3,4,4A,10B TETRAHYDRO 4 PROPYL 2H,5H [1]BENZOPYRANO[4,3 B][1,4]OXAZIN 9 OL; BP 897; BROMIDE; DOPAMINE; DOPAMINE 3 RECEPTOR; DOPAMINE 3 RECEPTOR BLOCKING AGENT; DOPAMINE 3 RECEPTOR STIMULATING AGENT; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); QUINPIROLE;

ANIMAL CELL; ANIMAL EXPERIMENT; ARTICLE; CHO CELL; CONTROLLED STUDY; DOPAMINE RECEPTOR BLOCKING; DOPAMINERGIC ACTIVITY; DOPAMINERGIC NERVE CELL; DOSE RESPONSE; DRUG ACTIVITY; DRUG ANTAGONISM; DRUG POTENCY; ELECTROPHYSIOLOGY; ENZYME ACTIVATION; EXPERIMENTAL MODEL; HUMAN; IC 50; IN VIVO STUDY; MALE; NERVE CONDUCTION; NONHUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION; RAT; RECEPTOR BINDING; SUBSTANTIA NIGRA;

ANIMALS; BENZOPYRANS; BINDING, COMPETITIVE; CHO CELLS; CRICETINAE; DENDRITES; DOPAMINE; DOPAMINE AGONISTS; DOPAMINE ANTAGONISTS; DOSE-RESPONSE RELATIONSHIP, DRUG; ELECTROPHYSIOLOGY; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); HUMANS; MALE; NEURONS; OXAZINES; PIPERAZINES; QUINPIROLE; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, DOPAMINE D2; RECEPTORS, DOPAMINE D3; SUBSTANTIA NIGRA; SULFUR RADIOISOTOPES; TETRAHYDRONAPHTHALENES;

EID: 0035919534     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(01)01054-8     Document Type: Article

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