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Volumn 53, Issue 2, 1998, Pages 283-294

Ivermectin: A positive allosteric effector of the α7 neuronal nicotinic acetylcholine receptor

Author keywords

[No Author keywords available]

Indexed keywords

CHOLINERGIC RECEPTOR; IVERMECTIN; NICOTINIC RECEPTOR;

EID: 0031887759     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.53.2.283     Document Type: Article
Times cited : (285)

References (40)
  • 1
    • 0026450951 scopus 로고
    • Pharmacological properties of the homomeric alpha 7 receptor
    • Bertrand D, Bertrand S, and Ballivet M (1992) Pharmacological properties of the homomeric alpha 7 receptor. Neurosci Lett 146:87-90.
    • (1992) Neurosci Lett , vol.146 , pp. 87-90
    • Bertrand, D.1    Bertrand, S.2    Ballivet, M.3
  • 2
    • 0031032208 scopus 로고    scopus 로고
    • Electrophysiology: A method to investigate the functional properties of ligand-gated channels
    • Bertrand D, Buisson B, Krause RM, Hu H-Y, and Bertrand S (1997) Electrophysiology: a method to investigate the functional properties of ligand-gated channels. J Recept Signal Transd Res 17:227-242.
    • (1997) J Recept Signal Transd Res , vol.17 , pp. 227-242
    • Bertrand, D.1    Buisson, B.2    Krause, R.M.3    Hu, H.-Y.4    Bertrand, S.5
  • 3
    • 0029006150 scopus 로고
    • Nicotinic receptor: An allosteric protein specialized for intercellular communication
    • Bertrand D and Changeux JP (1995) Nicotinic receptor: an allosteric protein specialized for intercellular communication. Semin Neurosci 7:75-90.
    • (1995) Semin Neurosci , vol.7 , pp. 75-90
    • Bertrand, D.1    Changeux, J.P.2
  • 4
    • 85013526554 scopus 로고
    • Electrophysiology of neuronal nicotinic acetylcholine receptors expressed in Xenopus oocytes following nuclear injection of genes or cDNA
    • (Conn M, ed) Academic Press, New York
    • Bertrand D, Cooper E, Valera S, Rungger D, and Ballivet M (1991a) Electrophysiology of neuronal nicotinic acetylcholine receptors expressed in Xenopus oocytes following nuclear injection of genes or cDNA, in Methods in Neuroscience (Conn M, ed) pp 174-193, Academic Press, New York.
    • (1991) Methods in Neuroscience , pp. 174-193
    • Bertrand, D.1    Cooper, E.2    Valera, S.3    Rungger, D.4    Ballivet, M.5
  • 5
    • 0027214596 scopus 로고
    • Mutations at two distinct sites within the channel domain M2 alter calcium permeability of neuronal alpha 7 nicotinic receptor
    • Bertrand D, Galzi JL, Devillers-Thiéry A, Bertrand S, and Changeux JP (1993) Mutations at two distinct sites within the channel domain M2 alter calcium permeability of neuronal alpha 7 nicotinic receptor. Proc Natl Acad Sci USA 90:6971-6975.
    • (1993) Proc Natl Acad Sci USA , vol.90 , pp. 6971-6975
    • Bertrand, D.1    Galzi, J.L.2    Devillers-Thiéry, A.3    Bertrand, S.4    Changeux, J.P.5
  • 8
    • 2642614797 scopus 로고    scopus 로고
    • Steroid modulation of the nicotinic acetylcholine receptor
    • (Conn M, ed) Humana Press, Totowa, NJ
    • Buisson B and Bertrand D (1998) Steroid modulation of the nicotinic acetylcholine receptor, in Comparative Endocrinology (Conn M, ed) Humana Press, Totowa, NJ.
    • (1998) Comparative Endocrinology
    • Buisson, B.1    Bertrand, D.2
  • 11
    • 0025605864 scopus 로고
    • A neuronal nicotinic acetylcholine receptor subunit (alpha 7) is developmentally regulated and forms a homo-oligomeric channel blocked by alpha-BTX
    • Couturier S, Bertrand D, Matter JM, Hernandez MC, Bertrand S, Millar N, Valera S, Barkas T, and Ballivet M (1990) A neuronal nicotinic acetylcholine receptor subunit (alpha 7) is developmentally regulated and forms a homo-oligomeric channel blocked by alpha-BTX. Neuron 5:847-56.
    • (1990) Neuron , vol.5 , pp. 847-856
    • Couturier, S.1    Bertrand, D.2    Matter, J.M.3    Hernandez, M.C.4    Bertrand, S.5    Millar, N.6    Valera, S.7    Barkas, T.8    Ballivet, M.9
  • 13
    • 0031000154 scopus 로고    scopus 로고
    • Activation of the recombinant human alpha-7 nicotinic acetylcholine receptor significantly raises intracellular free calcium
    • Delbono O, Gopalakrishnan M, Renganathan M, Monteggia LM, Messi ML, and Sullivan JP (1997) Activation of the recombinant human alpha-7 nicotinic acetylcholine receptor significantly raises intracellular free calcium. J Pharmacol Exp Ther 280:428-438.
    • (1997) J Pharmacol Exp Ther , vol.280 , pp. 428-438
    • Delbono, O.1    Gopalakrishnan, M.2    Renganathan, M.3    Monteggia, L.M.4    Messi, M.L.5    Sullivan, J.P.6
  • 15
    • 0029958046 scopus 로고    scopus 로고
    • Identification of calcium binding sites that regulate potentiation of a neuronal nicotinic acetylcholine receptor
    • Galzi JL, Bertrand S, Corringer PJ, Changeux JP, and Bertrand D (1996a) Identification of calcium binding sites that regulate potentiation of a neuronal nicotinic acetylcholine receptor. EMBO J 15:5824-5832.
    • (1996) EMBO J , vol.15 , pp. 5824-5832
    • Galzi, J.L.1    Bertrand, S.2    Corringer, P.J.3    Changeux, J.P.4    Bertrand, D.5
  • 16
    • 0026656037 scopus 로고
    • Mutations in the ion channel domain of a neuronal nicotinic receptor convert ion selectivity from cationic to anionic
    • Galzi JL, Devillers-Thiéry A, Hussy N, Bertrand S, Changeux JP, and Bertrand D (1992) Mutations in the ion channel domain of a neuronal nicotinic receptor convert ion selectivity from cationic to anionic. Nature (Lond) 359:500-505.
    • (1992) Nature (Lond) , vol.359 , pp. 500-505
    • Galzi, J.L.1    Devillers-Thiéry, A.2    Hussy, N.3    Bertrand, S.4    Changeux, J.P.5    Bertrand, D.6
  • 19
    • 0029805769 scopus 로고    scopus 로고
    • Hippocampal synaptic transmission enhanced by low concentrations of nicotine
    • Gray R, Rajan AS, Radcliffe KA, Yakehiro M, and Dani JA (1996) Hippocampal synaptic transmission enhanced by low concentrations of nicotine. Nature (Lond) 383:713-716.
    • (1996) Nature (Lond) , vol.383 , pp. 713-716
    • Gray, R.1    Rajan, A.S.2    Radcliffe, K.A.3    Yakehiro, M.4    Dani, J.A.5
  • 20
    • 0028174057 scopus 로고
    • Effect of ivermectin on γ-aminobutyric acid-induced chloride currents in mouse hippocampal embryonic neurones
    • Krusek J and Zemková H (1994) Effect of ivermectin on γ-aminobutyric acid-induced chloride currents in mouse hippocampal embryonic neurones. Eur J Pharmacol 259:121-128.
    • (1994) Eur J Pharmacol , vol.259 , pp. 121-128
    • Krusek, J.1    Zemková, H.2
  • 21
    • 0030611558 scopus 로고    scopus 로고
    • 2+; ions in nicotinic facilitation of GABA release in mouse thalamus
    • 2+; ions in nicotinic facilitation of GABA release in mouse thalamus. J Neurosci 17:576-585.
    • (1997) J Neurosci , vol.17 , pp. 576-585
    • Léna, C.1    Changeux, J.P.2
  • 22
    • 0029690580 scopus 로고    scopus 로고
    • Neuronal nicotinic acetylcholine receptors
    • (Narahashi T, ed) Plenum Press, New York
    • Lindstrom J (1996) Neuronal nicotinic acetylcholine receptors, in Ion Channels. (Narahashi T, ed) pp 377-450, Plenum Press, New York.
    • (1996) Ion Channels , pp. 377-450
    • Lindstrom, J.1
  • 24
    • 78651189765 scopus 로고
    • On the nature of allosteric transitions: A plausible model
    • Monod J, Wyman J, and Changeux JP (1965) On the nature of allosteric transitions: a plausible model. J Mol Biol 12:88-118.
    • (1965) J Mol Biol , vol.12 , pp. 88-118
    • Monod, J.1    Wyman, J.2    Changeux, J.P.3
  • 25
    • 0026716690 scopus 로고
    • Potentiation of nicotinic receptor response by external calcium in rat central neurons
    • Mulle C, Lêna C, and Changeux JP (1992) Potentiation of nicotinic receptor response by external calcium in rat central neurons. Neuron 8:937-945.
    • (1992) Neuron , vol.8 , pp. 937-945
    • Mulle, C.1    Lêna, C.2    Changeux, J.P.3
  • 27
    • 0026011670 scopus 로고
    • Community-based treatment of onchocerciasis with ivermectin: Safety, efficacy, and acceptability of yearly treatment
    • Pacqué M, Muñoz B, Greene BM, and Taylor HR (1991) Community-based treatment of onchocerciasis with ivermectin: safety, efficacy, and acceptability of yearly treatment. J Inf Dis 163:381-385.
    • (1991) J Inf Dis , vol.163 , pp. 381-385
    • Pacqué, M.1    Muñoz, B.2    Greene, B.M.3    Taylor, H.R.4
  • 28
    • 0029670737 scopus 로고    scopus 로고
    • Neuronal nicotinic α7 receptor expressed in Xenopus oocytes presents five putative binding sites for methyllycaconitine
    • Palma E, Bertrand S, Binzoni T, and Bertrand D (1996) Neuronal nicotinic α7 receptor expressed in Xenopus oocytes presents five putative binding sites for methyllycaconitine. J Physiol (Lond) 491:151-161.
    • (1996) J Physiol (Lond) , vol.491 , pp. 151-161
    • Palma, E.1    Bertrand, S.2    Binzoni, T.3    Bertrand, D.4
  • 29
    • 0028176058 scopus 로고
    • Human α7 acetylcholine receptor: Cloning of the α7 subunit from the SH-SY5Y cell line and determination of pharmacological properties of native receptors and functional α7 homomers expressed in Xenopus oocytes
    • Peng X, Katz M, Gerzanich V, Anand R, and Lindstrom J (1994) Human α7 acetylcholine receptor: cloning of the α7 subunit from the SH-SY5Y cell line and determination of pharmacological properties of native receptors and functional α7 homomers expressed in Xenopus oocytes. Mol Pharmacol 45:546-554.
    • (1994) Mol Pharmacol , vol.45 , pp. 546-554
    • Peng, X.1    Katz, M.2    Gerzanich, V.3    Anand, R.4    Lindstrom, J.5
  • 30
    • 0022634647 scopus 로고
    • Hemoglobin as a receptor of drugs and peptides: X-ray studies of the stereochemistry of binding
    • Perutz MF, Fermi G, Abraham G, Poyart C, and Bursaux E (1986) Hemoglobin as a receptor of drugs and peptides: x-ray studies of the stereochemistry of binding. J Am Chem Soc 108:1064-1078.
    • (1986) J Am Chem Soc , vol.108 , pp. 1064-1078
    • Perutz, M.F.1    Fermi, G.2    Abraham, G.3    Poyart, C.4    Bursaux, E.5
  • 34
    • 0014014862 scopus 로고
    • On the nature of allosteric transitions: Implications of nonexclusive ligand binding
    • Rubin MM and Changeux JP (1966) On the nature of allosteric transitions: implications of nonexclusive ligand binding. J Mol Biol 21:265-274.
    • (1966) J Mol Biol , vol.21 , pp. 265-274
    • Rubin, M.M.1    Changeux, J.P.2
  • 35
    • 0027787864 scopus 로고
    • - channels by avermectin in rat cultured hippocampal neurons
    • - channels by avermectin in rat cultured hippocampal neurons. Arch Pharm 348:628-632.
    • (1993) Arch Pharm , vol.348 , pp. 628-632
    • Schönrock, B.1    Bormann, J.2
  • 36
    • 0023508151 scopus 로고
    • Effect of Avermectin B1a on chick neuronal γ-aminobutyrate receptor channels expressed in Xenopus oocytes
    • Sigel E and Baur R (1987) Effect of Avermectin B1a on chick neuronal γ-aminobutyrate receptor channels expressed in Xenopus oocytes. Mol Pharmacol 32:749-752.
    • (1987) Mol Pharmacol , vol.32 , pp. 749-752
    • Sigel, E.1    Baur, R.2
  • 37
    • 0026738827 scopus 로고
    • Progesterone modulates a neuronal nicotinic acetylcholine receptor
    • Valera S, Ballivet M, and Bertrand D (1992) Progesterone modulates a neuronal nicotinic acetylcholine receptor. Proc Natl Acad Sci USA 89:9949-9953.
    • (1992) Proc Natl Acad Sci USA , vol.89 , pp. 9949-9953
    • Valera, S.1    Ballivet, M.2    Bertrand, D.3
  • 38
    • 0029586823 scopus 로고
    • Epibatidine and ABT 418 reveal selective losses of alpha4 beta2 nicotinic receptors in Alzheimer brains
    • Warpman U and Nordberg A (1995) Epibatidine and ABT 418 reveal selective losses of alpha4 beta2 nicotinic receptors in Alzheimer brains. Neuroreport 6:2419-2423.
    • (1995) Neuroreport , vol.6 , pp. 2419-2423
    • Warpman, U.1    Nordberg, A.2
  • 39
    • 0028883671 scopus 로고
    • Cellular distribution of the mRNA for the alpha 7 subunit of the nicotinic acetylcholine receptor in the human cerebral cortex
    • Wevers A, Sullivan JP, Giordano T, Birtsch C, Monteggia LM, Nowacki S, Arneric S, and Schroder H (1995) Cellular distribution of the mRNA for the alpha 7 subunit of the nicotinic acetylcholine receptor in the human cerebral cortex. Drug Dev Res 36:103-110.
    • (1995) Drug Dev Res , vol.36 , pp. 103-110
    • Wevers, A.1    Sullivan, J.P.2    Giordano, T.3    Birtsch, C.4    Monteggia, L.M.5    Nowacki, S.6    Arneric, S.7    Schroder, H.8


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.