Structure-activity relationships of a novel series of melanin-concentrating hormone (MCH) receptor antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 15, 2004, Pages 4099-4102

  Arienzo, Rosa ^a   Clark, David E ^a   Cramp, Sue ^a   Daly, Stephen ^a   Dyke, Hazel J ^a   Lockey, Peter ^a   Norman, Dennis ^a   Roach, Alan G ^a   Stuttle, Keith ^a   Tomlinson, Maxine ^a   Wong, Melanie ^a   Wren, Stephen P ^a  

^a Argenta Discovery Ltd   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

2 AMINOQUINOLINE; HORMONE RECEPTOR BLOCKING AGENT; MELANIN CONCENTRATING HORMONE RECEPTOR ANTAGONIST; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL REACTION; DRUG ACTIVITY; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; IC 50; REACTION ANALYSIS; STRUCTURE ACTIVITY RELATION;

HUMANS; KINETICS; MOLECULAR CONFORMATION; PIPERAZINES; PIPERIDINES; RECEPTORS, PITUITARY HORMONE; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 3042642750     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.05.051     Document Type: Article

References (11)

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