Application of multi-component reactions to antimalarial drug discovery. Part 1: Parallel synthesis and antiplasmodial activity of new 4-aminoquinoline Ugi adducts

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 15, 2004, Pages 3901-3905

  Musonda, Chitalu C ^a   Taylor, Dale ^b   Lehman, Julie ^c   Gut, Jiri ^c   Rosenthal, Philip J ^c   Chibale, Kelly ^a  

^a UNIVERSITY OF CAPE TOWN   (South Africa)

^b UNIVERSITY OF CAPE TOWN   (South Africa)

^c UNIVERSITY OF CALIFORNIA   (United States)

Author keywords

4 Aminoquinolines; Malaria; Ugi isocyanide multi component reactions

Indexed keywords

4 AMINOQUINOLINE; ANTIMALARIAL AGENT;

ANTIMALARIAL ACTIVITY; ARTICLE; DRUG ACTIVITY; DRUG SYNTHESIS; NONHUMAN; PLASMODIUM FALCIPARUM; REACTION ANALYSIS;

PLASMODIUM FALCIPARUM;

EID: 3042545687     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.05.063     Document Type: Article

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