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Volumn 18, Issue 3, 2004, Pages 309-319

The evaluation of the N-type channel blocking properties of cilnidipine and other voltage-dependent calcium antagonists

Author keywords

1,4 dihydropyridine calcium 3H noradrenaline; Antagonist; Arteries; Cilnidipine; Heart; N type calcium channel

Indexed keywords

AMLODIPINE; CALCIUM CHANNEL N TYPE; CILNIDIPINE; MIBEFRADIL; NORADRENALIN; OMEGA CONOTOXIN GVIA; VOLTAGE GATED CALCIUM CHANNEL;

EID: 2942580721     PISSN: 07673981     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.1472-8206.2004.00236.x     Document Type: Article
Times cited : (22)

References (30)
  • 1
    • 0034780790 scopus 로고    scopus 로고
    • Calcium channel blockers in hypertension: Reappraisal after new trials and major meta-analyses
    • Opie L.H. Calcium channel blockers in hypertension: reappraisal after new trials and major meta-analyses. Am. J. Hypertens. (2001) 14 1074-1081.
    • (2001) Am. J. Hypertens. , vol.14 , pp. 1074-1081
    • Opie, L.H.1
  • 2
    • 0033850448 scopus 로고    scopus 로고
    • Calcium antagonists in the treatment of heart failure. Re-evaluation of therapeutic strategies
    • Gattis W., O'Connor C.M. Calcium antagonists in the treatment of heart failure. Re-evaluation of therapeutic strategies. Drugs (2000) 59 17-24.
    • (2000) Drugs , vol.59 , pp. 17-24
    • Gattis, W.1    O'Connor, C.M.2
  • 3
    • 0031912905 scopus 로고    scopus 로고
    • Calcium channel blockers in heart failure
    • Elkayam U. Calcium channel blockers in heart failure. Cardiology (1998) 89 (Suppl. 1) 38-46.
    • (1998) Cardiology , vol.89 , Issue.1 SUPPL. , pp. 38-46
    • Elkayam, U.1
  • 4
    • 0035212594 scopus 로고    scopus 로고
    • Calcium channel blockers in treatment of hypertension
    • Muntwyler J., Follath F. Calcium channel blockers in treatment of hypertension. Prog. Cardiovasc. Dis. (2001) 44 207-216.
    • (2001) Prog. Cardiovasc. Dis. , vol.44 , pp. 207-216
    • Muntwyler, J.1    Follath, F.2
  • 5
    • 0035988499 scopus 로고    scopus 로고
    • The effects of calcium channel blockers on cardiovascular outcomes: A review of randomised controlled trials
    • De Leeuw P.W., Birkenhager W.H. The effects of calcium channel blockers on cardiovascular outcomes: a review of randomised controlled trials. Blood Press. (2002) 11 71-78.
    • (2002) Blood Press. , vol.11 , pp. 71-78
    • De Leeuw, P.W.1    Birkenhager, W.H.2
  • 6
    • 0019415146 scopus 로고
    • Regional wall motion from radiopaque markers after intravenous and intracoronary injections of nifedipine
    • Serruys P.W., Brower R.W., ten Katen H.J., Bom A.H., Hugenholtz P.G. Regional wall motion from radiopaque markers after intravenous and intracoronary injections of nifedipine. Circulation (1981) 63 584-591.
    • (1981) Circulation , vol.63 , pp. 584-591
    • Serruys, P.W.1    Brower, R.W.2    Ten Katen, H.J.3    Bom, A.H.4    Hugenholtz, P.G.5
  • 8
    • 0028295970 scopus 로고
    • Unique pharmacologic properties of amlodipine
    • Burges R., Moisey D. Unique pharmacologic properties of amlodipine. Am. J. Cardiol. (1994) 73 2A-9A.
    • (1994) Am. J. Cardiol. , vol.73
    • Burges, R.1    Moisey, D.2
  • 9
    • 0025875513 scopus 로고
    • Pharmacology of lacidipine, a vascular-selective calcium antagonist
    • Micheli D., Ratti E., Toson G., Gaviraghi G. Pharmacology of lacidipine, a vascular-selective calcium antagonist. J. Cardiovasc. Pharmacol. (1991) 17 (Suppl. 4) S1-S8.
    • (1991) J. Cardiovasc. Pharmacol. , vol.17 , Issue.4 SUPPL.
    • Micheli, D.1    Ratti, E.2    Toson, G.3    Gaviraghi, G.4
  • 10
    • 0031739851 scopus 로고    scopus 로고
    • Lercanidipine: Short plasma half-life, long duration of action and high cholesterol tolerance. Updated molecular model to rationalize its pharmacokinetic properties
    • Herbette L.G., Vecchiarelli M., Sartani A., Leonardi A. Lercanidipine: short plasma half-life, long duration of action and high cholesterol tolerance. Updated molecular model to rationalize its pharmacokinetic properties. Blood Press. (1998) 2 10-17.
    • (1998) Blood Press. , vol.2 , pp. 10-17
    • Herbette, L.G.1    Vecchiarelli, M.2    Sartani, A.3    Leonardi, A.4
  • 11
    • 0036563247 scopus 로고    scopus 로고
    • N- and L-type calcium channel antagonist improves glomerular dynamics, reverses severe nephrosclerosis, and inhibits apoptosis and proliferation in an 1-NAME/SHR model
    • Zhou X., Ono H., Ono Y., Frohlich E.D. N- and L-type calcium channel antagonist improves glomerular dynamics, reverses severe nephrosclerosis, and inhibits apoptosis and proliferation in an 1-NAME/SHR model. J. Hypertens. (2002) 20 993-1000.
    • (2002) J. Hypertens. , vol.20 , pp. 993-1000
    • Zhou, X.1    Ono, H.2    Ono, Y.3    Frohlich, E.D.4
  • 12
    • 0033972645 scopus 로고    scopus 로고
    • Preferential inhibition of L- and N-type calcium channels in the rat hippocampal neurons by cilnidipine
    • Murai Y., Uneyama H., Ishibashi H., Takahama K., Akaike N. Preferential inhibition of L- and N-type calcium channels in the rat hippocampal neurons by cilnidipine. Brain Res. (2000) 854 6-10.
    • (2000) Brain Res. , vol.854 , pp. 6-10
    • Murai, Y.1    Uneyama, H.2    Ishibashi, H.3    Takahama, K.4    Akaike, N.5
  • 13
    • 0023874003 scopus 로고
    • Dominant role of N-type Ca2+ channels in evoked release of norepinephrine from sympathetic neurons
    • Hirning L.D., Fox A.P., McCleskey E.W. et al. Dominant role of N-type Ca2+ channels in evoked release of norepinephrine from sympathetic neurons. Science (1988) 239 57-61.
    • (1988) Science , vol.239 , pp. 57-61
    • Hirning, L.D.1    Fox, A.P.2    McCleskey, E.W.3
  • 14
    • 0029791654 scopus 로고    scopus 로고
    • Effects of N-, P- and Q-type neuronal calcium channel antagonists on mammalian peripheral neurotransmission
    • Wright C.E., Angus J.A. Effects of N-, P- and Q-type neuronal calcium channel antagonists on mammalian peripheral neurotransmission. Br. J. Pharmacol. (1996) 119 49-56.
    • (1996) Br. J. Pharmacol. , vol.119 , pp. 49-56
    • Wright, C.E.1    Angus, J.A.2
  • 15
    • 0030942404 scopus 로고    scopus 로고
    • Effect of cilnidipine, a novel dihydropyridine Ca++-channel antagonist, on N-type Ca++ channel in rat dorsal root ganglion neurons
    • Fujii S., Kameyama K., Hosono M., Hayashi Y., Kitamura K. Effect of cilnidipine, a novel dihydropyridine Ca++-channel antagonist, on N-type Ca++ channel in rat dorsal root ganglion neurons. J. Pharmacol. Exp. Ther. (1997) 280 1184-1191.
    • (1997) J. Pharmacol. Exp. Ther. , vol.280 , pp. 1184-1191
    • Fujii, S.1    Kameyama, K.2    Hosono, M.3    Hayashi, Y.4    Kitamura, K.5
  • 16
    • 0028865516 scopus 로고
    • Inhibitory effect of cilnidipine on pressor response to acute cold stress in spontaneously hypertensive rats
    • Hosono M., Hiruma T., Watanabe K. et al. Inhibitory effect of cilnidipine on pressor response to acute cold stress in spontaneously hypertensive rats. Jpn. J. Pharmacol. (1995) 69 119-125.
    • (1995) Jpn. J. Pharmacol. , vol.69 , pp. 119-125
    • Hosono, M.1    Hiruma, T.2    Watanabe, K.3
  • 17
    • 0033051158 scopus 로고    scopus 로고
    • Effects of amlodipine and cilnidipine on cardiac sympathetic nervous system and neurohormonal status in essential hypertension
    • Sakata K., Shirotani M., Yoshida H. et al. Effects of amlodipine and cilnidipine on cardiac sympathetic nervous system and neurohormonal status in essential hypertension. Hypertension (1999) 33 1447-1452.
    • (1999) Hypertension , vol.33 , pp. 1447-1452
    • Sakata, K.1    Shirotani, M.2    Yoshida, H.3
  • 18
    • 0017702173 scopus 로고
    • Contractile properties of small arterial resistance vessels in spontaneously hypertensive and normotensive rats
    • Mulvany M.J., Halpern W. Contractile properties of small arterial resistance vessels in spontaneously hypertensive and normotensive rats. Circ. Res. (1977) 41 19-26.
    • (1977) Circ. Res. , vol.41 , pp. 19-26
    • Mulvany, M.J.1    Halpern, W.2
  • 19
    • 0033979505 scopus 로고    scopus 로고
    • Inhibitory effect of mibefradil on contractions induced by sympathetic neurotransmitter release in the rat tail artery
    • van der L.R., Pfaffendorf M., De Mey J.G., van Zwieten P.A. Inhibitory effect of mibefradil on contractions induced by sympathetic neurotransmitter release in the rat tail artery. Naunyn Schmiedebergs Arch. Pharmacol. (2000) 361 74-79.
    • (2000) Naunyn Schmiedebergs Arch. Pharmacol. , vol.361 , pp. 74-79
    • Van Der, L.R.1    Pfaffendorf, M.2    De Mey, J.G.3    Van Zwieten, P.A.4
  • 20
    • 0035502303 scopus 로고    scopus 로고
    • Characterisation of a modified approach to the study of sympathetic neurotransmission and its presynaptic modulation in the isolated rabbit thoracic aorta
    • Nap A., Pfaffendorf M., van Zwieten P. Characterisation of a modified approach to the study of sympathetic neurotransmission and its presynaptic modulation in the isolated rabbit thoracic aorta. J. Pharmacol Toxicol Methods (2001) 46 (3) 145-151.
    • (2001) J. Pharmacol. Toxicol. Methods , vol.46 , Issue.3 , pp. 145-151
    • Nap, A.1    Pfaffendorf, M.2    Van Zwieten, P.3
  • 21
    • 0028865517 scopus 로고
    • Inhibitory effect of cilnidipine on vascular sympathetic neurotransmission and subsequent vasoconstriction in spontaneously hypertensive rats
    • Hosono M., Fujii S., Hiruma T. et al. Inhibitory effect of cilnidipine on vascular sympathetic neurotransmission and subsequent vasoconstriction in spontaneously hypertensive rats. Jpn. J. Pharmacol. (1995) 69 127-134.
    • (1995) Jpn. J. Pharmacol. , vol.69 , pp. 127-134
    • Hosono, M.1    Fujii, S.2    Hiruma, T.3
  • 22
    • 0034141454 scopus 로고    scopus 로고
    • N-Type calcium channels control sympathetic neurotransmission in human heart atrium
    • Molderings G.J., Likungu J., Gothert M. N-Type calcium channels control sympathetic neurotransmission in human heart atrium. Circulation (2000) 101 403-407.
    • (2000) Circulation , vol.101 , pp. 403-407
    • Molderings, G.J.1    Likungu, J.2    Gothert, M.3
  • 23
    • 0036065892 scopus 로고    scopus 로고
    • Inhibitory effects of cilnidipine on peripheral and brain N-type Ca(2+) channels expressed in BHK cells
    • Kato K., Wakamori M., Mori Y., Imoto K., Kitamura K. Inhibitory effects of cilnidipine on peripheral and brain N-type Ca(2+) channels expressed in BHK cells. Neuropharmacology (2002) 42 1099-1108.
    • (2002) Neuropharmacology , vol.42 , pp. 1099-1108
    • Kato, K.1    Wakamori, M.2    Mori, Y.3    Imoto, K.4    Kitamura, K.5
  • 24
    • 0030766439 scopus 로고    scopus 로고
    • Blockade of N-type Ca2+ current by cilnidipine (FRC-8653) in acutely dissociated rat sympathetic neurones
    • Uneyama H., Takahara A., Dohmoto H., Yoshimoto R., Inoue K., Akaike N. Blockade of N-type Ca2+ current by cilnidipine (FRC-8653) in acutely dissociated rat sympathetic neurones. Br. J. Pharmacol. (1997) 122 37-42.
    • (1997) Br. J. Pharmacol. , vol.122 , pp. 37-42
    • Uneyama, H.1    Takahara, A.2    Dohmoto, H.3    Yoshimoto, R.4    Inoue, K.5    Akaike, N.6
  • 25
    • 0025076265 scopus 로고
    • Apparent vascular to cardiac sympatholytic selectivity of omega-conotoxin GVIA in the pithed rat
    • Pruneau D., Angus J.A. Apparent vascular to cardiac sympatholytic selectivity of omega-conotoxin GVIA in the pithed rat. Eur. J. Pharmacol. (1990) 184 127-133.
    • (1990) Eur. J. Pharmacol. , vol.184 , pp. 127-133
    • Pruneau, D.1    Angus, J.A.2
  • 26
    • 0035830609 scopus 로고    scopus 로고
    • Effects of a dual L/N-type Ca(2+) channel blocker cilnidipine on neurally mediated chronotropic response in anesthetized dogs
    • Konda T., Takahara A., Maeda K., Dohmoto H., Yoshimoto R. Effects of a dual L/N-type Ca(2+) channel blocker cilnidipine on neurally mediated chronotropic response in anesthetized dogs. Eur. J. Pharmacol. (2001) 413 117-120.
    • (2001) Eur. J. Pharmacol. , vol.413 , pp. 117-120
    • Konda, T.1    Takahara, A.2    Maeda, K.3    Dohmoto, H.4    Yoshimoto, R.5
  • 27
    • 0033847605 scopus 로고    scopus 로고
    • The sinoatrial node, a heterogeneous pacemaker structure
    • Boyett M.R., Honjo H., Kodama I. The sinoatrial node, a heterogeneous pacemaker structure. Cardiovasc. Res. (2000) 47 658-687.
    • (2000) Cardiovasc. Res. , vol.47 , pp. 658-687
    • Boyett, M.R.1    Honjo, H.2    Kodama, I.3
  • 28
    • 0032955695 scopus 로고    scopus 로고
    • Contribution of L-type Ca2+ current to electrical activity in sinoatrial nodal myocytes of rabbits
    • Verheijck E.E., van Ginneken A.C., Wilders R., Bouman L.N. Contribution of L-type Ca2+ current to electrical activity in sinoatrial nodal myocytes of rabbits. Am. J. Physiol. (1999) 276 H1064-H1077.
    • (1999) Am. J. Physiol. , vol.276
    • Verheijck, E.E.1    Van Ginneken, A.C.2    Wilders, R.3    Bouman, L.N.4
  • 29
    • 0034725972 scopus 로고    scopus 로고
    • Mibefradil, an I(Ca,T) blocker, effectively blocks I(Ca,L) in rabbit sinus node cells
    • Protas L., Robinson R.B. Mibefradil, an I(Ca,T) blocker, effectively blocks I(Ca,L) in rabbit sinus node cells. Eur. J. Pharmacol. (2000) 401 27-30.
    • (2000) Eur. J. Pharmacol. , vol.401 , pp. 27-30
    • Protas, L.1    Robinson, R.B.2
  • 30
    • 0035068015 scopus 로고    scopus 로고
    • State-dependent inhibition of L-type Ca2+ channels in A7r5 cells by cilnidipine and its derivatives
    • Uchida R., Yamazaki J., Ozeki S., Kitamura K. State-dependent inhibition of L-type Ca2+ channels in A7r5 cells by cilnidipine and its derivatives. Jpn. J. Pharmacol. (2001) 85 260-270.
    • (2001) Jpn. J. Pharmacol. , vol.85 , pp. 260-270
    • Uchida, R.1    Yamazaki, J.2    Ozeki, S.3    Kitamura, K.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.