Synthesis and antibacterial activity of novel bifunctional macrolides

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 14, 2004, Pages 3809-3813

  Akritopoulou Zanze, Irini ^a   Phelan, Kathleen M ^a   Marron, Thomas G ^a   Yong, Hong ^a   Ma, Zhenkun ^a,b   Stone, Greg G ^a,c   Daly, Melissa M ^a   Hensey, Dena M ^a   Nilius, Angela M ^a   Djuric, Stevan W ^a  

^a ABBOTT LABORATORIES   (United States)

^b Cumbre Inc   (United States)

^c PFIZER INC   (United States)

Author keywords

Bifunctional macrolides; Ketolides; Macrolide resistance

Indexed keywords

ANTIBIOTIC AGENT; ERYTHROMYCIN; MACROLIDE;

ANTIBACTERIAL ACTIVITY; ANTIBIOTIC RESISTANCE; ARTICLE; BACTERIAL STRAIN; CONTROLLED STUDY; DRUG SCREENING; DRUG SYNTHESIS; HAEMOPHILUS INFLUENZAE; METHICILLIN RESISTANT STAPHYLOCOCCUS AUREUS; NONHUMAN; STAPHYLOCOCCUS AUREUS; STREPTOCOCCUS PNEUMONIAE;

ANTI-BACTERIAL AGENTS; BACTERIA; CELL MEMBRANE; DRUG RESISTANCE; DRUG RESISTANCE, BACTERIAL; ERYTHROMYCIN; MACROLIDES; MICROBIAL SENSITIVITY TESTS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 2942558864     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.04.077     Document Type: Article

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