Synthesis and antitrichinellosis activity of some 2-substituted-[1,3] thiazolo[3,2-a]benzimidazol-3(2H)-ones

Bioorganic and Medicinal Chemistry

Volumn 13, Issue 19, 2005, Pages 5550-5559

  Mavrova, Anelia Ts ^a   Anichina, Kamelya K ^a   Vuchev, Dimitar I ^b   Tsenov, Jordan A ^c   Kondeva, Magdalena S ^d   Micheva, Mitka K ^d  

^a UNIVERSITY OF CHEMICAL TECHNOLOGY AND METALLURGY   (Bulgaria)

^b NATIONAL CENTER OF INFECTIOUS AND PARASITIC DISEASES   (Bulgaria)

^c INSTITUTE OF ORGANIC CHEMISTRY   (Bulgaria)

^d UNIVERSITY OF SOFIA   (Bulgaria)

Author keywords

Ab initio; Antitrichinellosis activity; Benzimidazoles; Hepatotoxicity; Thiazolo 2,3 a benzimidazolones

Indexed keywords

2 (1,3 BENZODIOXOL 5 YLMETHYLENE)[1,3]THIAZOLO[3,2 A]BENZIMIDAZOL 3(2H) ONE; 2 (INDOL 3 YLMETHYLENE) 6(7) METHYL[1,3]THIAZOLO[3,2 A]BENZIMIDAZOL 3(2H) ONE; 2 (INDOL 3 YLMETHYLENE)[1,3]THIAZOLO[3,2 A]BENZIMIDAZOL 3(2H) ONE; ALBENDAZOLE; BENZIMIDAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

AB INITIO CALCULATION; ANIMAL CELL; ANTHELMINTIC ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG CYTOTOXICITY; DRUG EFFECT; DRUG EFFICACY; DRUG STRUCTURE; DRUG SYNTHESIS; INFRARED SPECTROSCOPY; LIVER TOXICITY; MASS SPECTROMETRY; NONHUMAN; PROTON NUCLEAR MAGNETIC RESONANCE; RAT; STRUCTURE ANALYSIS; TRICHINELLA SPIRALIS; TRICHINOSIS;

ANIMALS; BENZIMIDAZOLES; CELL SURVIVAL; DOSE-RESPONSE RELATIONSHIP, DRUG; HEPATOCYTES; MOLECULAR STRUCTURE; PARASITIC SENSITIVITY TESTS; RATS; THIAZOLES; TRICHINELLA SPIRALIS; TRICHINOSIS;

TRICHINELLA SPIRALIS;

EID: 23944520887     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2005.06.046     Document Type: Article

References (29)

1. L.X. Liu, and P.F. Weller Drug Therapy 334 1996 1178 1196
2. J. Dupouy-Camet, W. Kociecka, F. Brushi, Bolas-Fernandez, and E. Pozio Expert. Opin. Pharmacother. 3 2002 14
3. W.C. Campbell, and D.A. Denham W.C. Campbell Trichinella and Trichinosis 1983 Plenum Press USA and London, UK 340 355
4. W.C. Campbell, and R.S. Rew R. Rew Chemotherapy of Parasitic Diseases 1986 Plenum Press New York 282 283 302
5. W. Kociecka, L. Gustowska, and B. Morozewicz Effect of Early Prophylactic Therapy in Patients Infected with T. spiralis G. Ortega-Pierres R. Gambel F. Van Knapen D. Wakelin Trichinellosis. Proceedings of the 9th International Conference on Trichinellosis 1996 German Press Nonoalco Tlarecolo, Mexico 635 641
6. M.L. Lopez-Garcia, S. Torrado-Susana, S. Torrado-Santiago, A.R. Martinez, and F. Bolas Vet. Parasitol. 75 1998 209 219
7. T. Bera, and D.P. Belsarem Ind. J. Chem 31B 1992 370 372
8. W.C. Campbell Parasitol. Today 1 1985 10 176
9. L.X. Liu, and P.F. Weller New Eng. J. Med. 334 1996 1178 1184
10. A. Harder Parasitol. Res 88 2001 272 277
11. A. Criado-Fornelio, F. Rodrigues-Caabeiro, and A. Jimenez-Gonzalez Rev. Iber. Parasitol. 46 1986 326 332
12. R.M. Ros-Moreno, M.J. Moreno-Guzman, and A. Jimenez-Gonzalez Parasitol. Res. 85 1999 320 323
13. W.J. Blackhall, R.K. Prichard, and R.N. Beech Mol. Biochem. Parasitol. 131 2003 137 145
14. A. Mavrova, K. Anichina, and D. Vuchev J. Chem. Tech. Metal XXXVIII 2003 251 256
15. D. Davyt, W. Entz, R. Fernandes, and R. Mariezcurrena J. Nat. Prod. 61 1998 1560 1563
16. M. Khan J. Environ. Health B 18 1983 1223 1236
17. S.K. Srivastava, A. Agarwal, P.M. Chanhan, and S.K. Agarwal Bioorg. Med. Chem. 7 1999 1223 1236
18. S. Kapoor, and K.S. Singhal Indian J. Exp. Biol. 36 1998 887 890
19. W. Chengde, M.F. Chan, and F. Stavros J. Med. Chem. 40 1997 1690 1697
20. R.J. Barst, S. Rich, and E.M. Horn Circulation 102 2000 Abst 2076
21. Kim, B. M.; Vacca, J. P. G.B. Patent 2, 292, 246, 1996.
22. J.A. Van Allan, and B.D. Deacon Org. Synth. 4 1963 569
23. S. Narayan, V. Kumar, and H.K. Pujary Indian J. Chem. B 25 1986 267 270
24. Frisch, M. J.; Trucks, G. W.; Schlegel, H. B.; Scuseria, G. E.; Robb, M. A.; Cheeseman, J. R.; Zakrzewski, V. G.; Montgomery, J. A., Jr.; Stratmann, R. E.; Burant, J. C.; Dapprich, S.; Millam, J. M.; Daniels, A. D.; Kudin, K. N.; Strain, M. C.; Farkas, O.; Tomasi, J.; Barone, V.; Cossi, M.; Cammi, R.; Mennucci, B.; Pomelli, C.; Adamo, C.; Clifford, S.; Ochterski, J.; Petersson, G. A.; Ayala, P. Y.; Cui, Q.; Morokuma, K.; Malick, D. K.; Rabuck, A. D.; Raghavachari, K.; Foresman, J. B.; Cioslowski, J.; Ortiz, J. V.; Baboul, A. G.; Stefanov, B. B.; Liu, G.; Liashenko, A.; Piskorz, P.; Komaromi, I.; Gomperts, R.; Martin, R. L.; Fox, D. J.; Keith, T.; Al-Laham, M. A.; Peng, C. Y.; Nanayakkara, A.; Gonzalez, C.; Challacombe, M.; Gill, P. M. W.; Johnson, B.; Chen, W.; Wong, M. W.; Andres, J. L.; Gonzalez, C.; Head-Gordon, M.; Replogle, E. S.; Pople, J.A. Gaussian 98, Revision A.7, Gaussian, Inc., Pittsburgh, PA, 1998.
25. R.O. McCracken J. Parasitolog. 64 1978 214 219
26. X. Rey Grobellet, N. Ferre, and C. Eeckhoute Biochem. Biophys. Res. Commun. 220 1996 789 790
27. D. Fau, D. Eugene, and A. Berson J. Pharmacol. Exp. Therap. 269 1994 954 962
28. A. Mifrazaelian, M.R. Rouini, and S. Dadashzadeh Biopharm. Drug Dispos. 23 2002 379 383
29. D. Fau, A. Berson, and D. Eugene J. Pharmacol. Exp. Therap. 263 1992 67 69