Decrease in skin permeation and antibacterial effect of parabens by a polymeric additive, poly(2-methacryloyloxyethyl phosphorylcholine-co- butylmetacrylate)

Chemical and Pharmaceutical Bulletin

Volumn 53, Issue 3, 2005, Pages 271-276

  Hasegawa, Tetsuya ^a,b   Kim, Soan ^a   Tsuchida, Mamoru ^c   Issiki, Yasunori ^a   Kondo, Seiichi ^a   Sugibayashi, Kenji ^a  

^a JOSAI UNIVERSITY   (Japan)

^b JOSAI INTERNATIONAL UNIVERSITY   (Japan)

^c NOF Corporation   (Japan)

Author keywords

Antibacterial effect; Paraben; Poly(2 methacryloyloxyethyl phosphorylcholine co burylmetacrylate); Polymeric additive; Skin permeation

Indexed keywords

4 HYDROXYBENZOIC ACID ESTER; BUTYL PARABEN; DRUG ADDITIVE; ETHYL PARABEN; METHYL PARABEN; POLY(2 METHACRYLOYLOXYETHYLPHOSPHORYLCHOLINE CO BUTYL METHACRYLATE); POLYMER; PROPYL PARABEN; UNCLASSIFIED DRUG; WATER;

ANIMAL TISSUE; ANTIBACTERIAL ACTIVITY; AQUEOUS SOLUTION; ARTICLE; BACTERIAL MEMBRANE; CONCENTRATION (PARAMETERS); CONTROLLED STUDY; DRUG FORMULATION; DRUG SOLUBILITY; ESCHERICHIA COLI; HYDROPHILICITY; IN VITRO STUDY; LIPOPHILICITY; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; RAT; SKIN PENETRATION; STAPHYLOCOCCUS AUREUS;

ANIMALS; ANTI-BACTERIAL AGENTS; ANTI-INFECTIVE AGENTS, LOCAL; DIFFUSION; METHACRYLATES; PARABENS; PERMEABILITY; PHOSPHORYLCHOLINE; POLYMERS; RATS; SKIN; SOLUTIONS; WATER;

EID: 21144447619     PISSN: 00092363     EISSN: None     Source Type: Journal    
DOI: 10.1248/cpb.53.271     Document Type: Article

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