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QSAR and Combinatorial Science

Volumn 24, Issue 4, 2005, Pages 458-469

Structure-based design of bacterial hyaluronan lyase inhibitors

(5) Botzki, Alexander a,b Salmen, Sunnhild a Bernhardt, Günther a Buschauer, Armin a Dove, Stefan a

a UNIVERSITY OF REGENSBURG (Germany)

b SANOFI (France)

Author keywords

Hyaluronidase inhibitors; LUDI; Property distribution; Structure based design

Indexed keywords

BACTERIA; CRYSTAL STRUCTURE; ENZYMES; HYALURONIC ACID;

EXTRACELLULAR MATRICES; HYALURONAN; HYALURONIDASE INHIBITOR; LUDI; POTENT INHIBITOR; PROPERTY; PROPERTY DISTRIBUTION; SELECTIVE INHIBITORS; STRUCTURE-BASED DESIGNS; TOOL DRUGS;

DATABASE SYSTEMS;

1,3 DIACETYLBENZIMIDAZOLE 2 THIONE; ENZYME INHIBITOR; HYALURONIDASE; HYALURONIDASE ANTIBODY; UNCLASSIFIED DRUG;

CONFERENCE PAPER; CRYSTAL STRUCTURE; DRUG DESIGN; DRUG SCREENING; DRUG STRUCTURE; MOLECULAR MODEL; MOLECULAR WEIGHT; PRIORITY JOURNAL; SCORING SYSTEM; STREPTOCOCCUS AGALACTIAE; STRUCTURAL HOMOLOGY;

EID: 20544455003 PISSN: 1611020X EISSN: None Source Type: Journal
DOI: 10.1002/qsar.200430930 Document Type: Conference Paper

Times cited : (11)

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