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Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 13, 2005, Pages 3302-3306

Carbonic anhydrase inhibitors. Synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with boron-containing sulfonamides, sulfamides, and sulfamates: Toward agents for boron neutron capture therapy of hypoxic tumors

(6) Winum, Jean Yves a,b Cecchi, Alessandro a Montero, Jean Louis b Innocenti, Alessio a Scozzafava, Andrea a Supuran, Claudiu T a

a UNIVERSITY OF FLORENCE (Italy)

b UNIV MONTPELLIER (France)

Author keywords

[No Author keywords available]

Indexed keywords

BORON DERIVATIVE; CARBONATE DEHYDRATASE; CARBONATE DEHYDRATASE I; CARBONATE DEHYDRATASE II; CARBONATE DEHYDRATASE INHIBITOR; SULFAMIDE DERIVATIVE; SULFONAMIDE;

ARTICLE; BINDING AFFINITY; CHEMICAL REACTION; DRUG DESIGN; DRUG SYNTHESIS; DRUG TARGETING; ENZYME INHIBITION; HUMAN; MINIMUM INHIBITORY CONCENTRATION; NEUTRON CAPTURE THERAPY;

ANTIGENS, NEOPLASM; BORON COMPOUNDS; BORON NEUTRON CAPTURE THERAPY; CARBONIC ANHYDRASE I; CARBONIC ANHYDRASE II; CARBONIC ANHYDRASE INHIBITORS; CARBONIC ANHYDRASES; HUMANS; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES; SULFONIC ACIDS;

EID: 20444409690 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2005.04.058 Document Type: Article

Times cited : (53)

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