Novel cyclopentane dicarboxamide sodium channel blockers as a potential treatment for chronic pain

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 7, 2005, Pages 1901-1907

  Shao, Pengchang P ^a   Ok, Dong ^a   Fisher, Michael H ^a   Garcia, Maria L ^a   Kaczorowski, Gregory J ^a   Li, Chunshi ^a   Lyons, Kathryn A ^a   Martin, William J ^a   Meinke, Peter T ^a   Priest, Birgit T ^a   Smith, McHardy M ^a   Wyvratt, Matthew J ^a   Ye, Feng ^a   Parsons, William H ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

Author keywords

Chronic pain; Neuropathic pain; Sodium channel blocker

Indexed keywords

AMIDE; BIPHENYL DERIVATIVE; CARBAMAZEPINE; CYCLOPENTANE DERIVATIVE; LIDOCAINE; MEXILETINE; SODIUM CHANNEL BLOCKING AGENT; SUCCINIMIDE; VOLTAGE GATED SODIUM CHANNEL;

ARTICLE; CHRONIC PAIN; DRUG CLEARANCE; DRUG SCREENING; ELECTROPHYSIOLOGY; METHYLATION; REDUCTION; STOICHIOMETRY; STRUCTURE ACTIVITY RELATION;

EID: 20144383383     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.02.002     Document Type: Article

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