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Volumn 275, Issue 1-2, 2004, Pages 73-83

Microscopic molecular mobility of amorphous AG-041R measured by solid-state 13C NMR

Author keywords

Amorphous; Molecular mobility; Relaxation; Solid state 13C NMR

Indexed keywords

1 (2,2 DIETHOXYETHYL) 3 [(4 METHYLPHENYL)AMINOCARBONYLMETHYL] 3 (4 METHYLPHENYL)UREIDOINDOLIN 2 ONE; AG 041R; GASTRIN ANTAGONIST; UNCLASSIFIED DRUG;

EID: 1842638444     PISSN: 03785173     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ijpharm.2004.01.038     Document Type: Article
Times cited : (8)

References (15)
  • 2
    • 0030725409 scopus 로고    scopus 로고
    • Evaluation of three novel cholecystokinin-B/gastrin receptor antagonists: A study of their effects on rat stomach enterochromaffin-like cell activity
    • Ding X.Q., Lindstrom E., Hakanson R. Evaluation of three novel cholecystokinin-B/gastrin receptor antagonists: a study of their effects on rat stomach enterochromaffin-like cell activity. Phamacol. Toxicol. 81:1997;232-237.
    • (1997) Phamacol. Toxicol. , vol.81 , pp. 232-237
    • Ding, X.Q.1    Lindstrom, E.2    Hakanson, R.3
  • 3
    • 0031761368 scopus 로고    scopus 로고
    • Regeneration gene protein may mediate gastric mucosal proliferation induced by hypergastrinemia in rats
    • Fukui Y., Kinoshita T., Maekawa A., Okada S., Waki S., Hassan H., Okamoto H., Chiba T. Regeneration gene protein may mediate gastric mucosal proliferation induced by hypergastrinemia in rats. Gastroenterology. 115:1998;1483-1493.
    • (1998) Gastroenterology , vol.115 , pp. 1483-1493
    • Fukui, Y.1    Kinoshita, T.2    Maekawa, A.3    Okada, S.4    Waki, S.5    Hassan, H.6    Okamoto, H.7    Chiba, T.8
  • 4
    • 0032911447 scopus 로고    scopus 로고
    • Determination of the viscosity of an amorphous drug using thermomechanical analysis (TMA)
    • Hancock B.C., Dupuis Y., Thibert R. Determination of the viscosity of an amorphous drug using thermomechanical analysis (TMA). Pharm. Res. 16:1999a;672-675.
    • (1999) Pharm. Res. , vol.16 , pp. 672-675
    • Hancock, B.C.1    Dupuis, Y.2    Thibert, R.3
  • 5
    • 0029015405 scopus 로고    scopus 로고
    • Molecular mobility of amorphous pharmaceutical solids below their glass transition temperatures
    • Hancock B.C., Shamblin S.L., Zografi G. Molecular mobility of amorphous pharmaceutical solids below their glass transition temperatures. Pharm. Res. 12:1999b;799-805.
    • (1999) Pharm. Res. , vol.12 , pp. 799-805
    • Hancock, B.C.1    Shamblin, S.L.2    Zografi, G.3
  • 6
    • 0343953614 scopus 로고    scopus 로고
    • Oral bioavailability of a poorly water soluble HIV-1 protease inhibitor incorporated into pH-sensitive particles: Effect of the particle size and nutritional state
    • Jaeghere F.D., Allemann E., Kubel F., Galli B., Cozens R., Doelker E., Gruny R. Oral bioavailability of a poorly water soluble HIV-1 protease inhibitor incorporated into pH-sensitive particles: effect of the particle size and nutritional state. J. Control. Release. 68:2000;291-298.
    • (2000) J. Control. Release , vol.68 , pp. 291-298
    • Jaeghere, F.D.1    Allemann, E.2    Kubel, F.3    Galli, B.4    Cozens, R.5    Doelker, E.6    Gruny, R.7
  • 7
    • 0032756138 scopus 로고    scopus 로고
    • Physical properties of solid molecular dispersions of indomethacin with poly(vinylpyrrolidone) and poly(vinylpyrrolidone-co-vinyl-acetate) in relation to indomethacin crystallization
    • Matsumoto T., Zografi G. Physical properties of solid molecular dispersions of indomethacin with poly(vinylpyrrolidone) and poly(vinylpyrrolidone-co-vinyl-acetate) in relation to indomethacin crystallization. Pharm. Res. 16:1999;1728-1772.
    • (1999) Pharm. Res. , vol.16 , pp. 1728-1772
    • Matsumoto, T.1    Zografi, G.2
  • 8
    • 9544227573 scopus 로고
    • Dependence of the glass transition temperature on heating and cooling rate
    • Moynihan C.T., Easteal A.J., Wilder J., Tucker J. Dependence of the glass transition temperature on heating and cooling rate. J. Phys. Chem. 78:1974;2673-2677.
    • (1974) J. Phys. Chem. , vol.78 , pp. 2673-2677
    • Moynihan, C.T.1    Easteal, A.J.2    Wilder, J.3    Tucker, J.4
  • 9
    • 0033004759 scopus 로고    scopus 로고
    • Nucleation and crystallization kinetics of hydrated amorphous lactose above the glass transition temperature
    • Schmitt E.A., Law D., Zhang G.G. Nucleation and crystallization kinetics of hydrated amorphous lactose above the glass transition temperature. J. Pharm. Sci. 83:1999;291-296.
    • (1999) J. Pharm. Sci. , vol.83 , pp. 291-296
    • Schmitt, E.A.1    Law, D.2    Zhang, G.G.3
  • 10
    • 0034019632 scopus 로고    scopus 로고
    • Interpretation of relaxation time constants for amorphous pharmaceutical systems
    • Shamblin S.L., Hancock B.C., Duplix Y., Pikal M.J. Interpretation of relaxation time constants for amorphous pharmaceutical systems. Int. J. Pharm. Sci. 89:2000;417-427.
    • (2000) Int. J. Pharm. Sci. , vol.89 , pp. 417-427
    • Shamblin, S.L.1    Hancock, B.C.2    Duplix, Y.3    Pikal, M.J.4
  • 11
    • 1842756433 scopus 로고    scopus 로고
    • Glass and crystal formation in binary aromatic mixtures: A mechanism for reducing spin-lattice relaxation times
    • Wang W., Ronald J.P., Grant D.M. Glass and crystal formation in binary aromatic mixtures: a mechanism for reducing spin-lattice relaxation times. J. Phys. Chem. 100:1996;18550-18553.
    • (1996) J. Phys. Chem. , vol.100 , pp. 18550-18553
    • Wang, W.1    Ronald, J.P.2    Grant, D.M.3
  • 12
    • 0014699523 scopus 로고
    • Non-symmetrical dielectric relaxation behavior arising from a simple empirical decay function
    • Williams G., Watts D.C. Non-symmetrical dielectric relaxation behavior arising from a simple empirical decay function. Trans. Faraday Soc. 66:1970;80-85.
    • (1970) Trans. Faraday Soc. , vol.66 , pp. 80-85
    • Williams, G.1    Watts, D.C.2
  • 13
    • 0026761653 scopus 로고
    • Glass formation of 4′′-O-(4-methoxyphenyl) acetylosin and physicochemical stability of the amorphous solid
    • Yamaguchi T., Nishimura M., Okamoto R., Takeuchi T., Yamamoto K. Glass formation of 4′′-O-(4-methoxyphenyl) acetylosin and physicochemical stability of the amorphous solid. Int. J. Pharm. 85:1992;87-96.
    • (1992) Int. J. Pharm. , vol.85 , pp. 87-96
    • Yamaguchi, T.1    Nishimura, M.2    Okamoto, R.3    Takeuchi, T.4    Yamamoto, K.5
  • 14
    • 0028597539 scopus 로고
    • Crystallization of indomethacin from the amorphous state below and above its glass transition temperature
    • Yoshioka M., Hancock B.C., Zografi G. Crystallization of indomethacin from the amorphous state below and above its glass transition temperature. J. Pharm. Sci. 83:1994;1700-1705.
    • (1994) J. Pharm. Sci. , vol.83 , pp. 1700-1705
    • Yoshioka, M.1    Hancock, B.C.2    Zografi, G.3
  • 15
    • 0032960417 scopus 로고    scopus 로고
    • The effect of excipients on the molecular mobility of lyophilized formulations, as measured by glass transition temperature and NMR relaxation-based critical mobility temperature
    • Yoshioka S., Aso Y., Kojima S. The effect of excipients on the molecular mobility of lyophilized formulations, as measured by glass transition temperature and NMR relaxation-based critical mobility temperature. Pharm. Res. 16:1999;135-140.
    • (1999) Pharm. Res. , vol.16 , pp. 135-140
    • Yoshioka, S.1    Aso, Y.2    Kojima, S.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.