Synthesis of novel 10-deoxoartemisinins

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 10, 2005, Pages 2629-2631

  Khac, Vu Tran ^a   Van, Tuyen Nguyen ^a   Van, Sung Tran ^a  

^a INSTITUTE OF CHEMISTRY   (Viet Nam)

Author keywords

[No Author keywords available]

Indexed keywords

10 DEOXOARTEMISININ DERIVATIVE; ANTIMALARIAL AGENT; ARTEMISININ DERIVATIVE; UNCLASSIFIED DRUG;

ANTIBIOTIC RESISTANCE; ANTIMALARIAL ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG POTENCY; DRUG SYNTHESIS; IC 50; NONHUMAN; PLASMODIUM FALCIPARUM;

EID: 18144427876     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.03.050     Document Type: Article

References (24)

1. News from the WHO Division of Control of Tropical Diseases. TDR News 46 1994 5
2. M. Foely, and L. Tillely Int. J. Parasitol. 27 1997 213 240
3. J. Fishwick, W.G. McClean, G. Edwards, and S.A. Ward Chem. Biol. Interact. 96 1995 263 271
4. J.M. Grace, A.J. Anguilar, K.M. Trotman, and T.G. Brewer Drug Metab. Dispos. 26 1998 313 317
5. S.R. Meshnick, T.E. Taylor, and S. Kamchongwongpaisan Microbiol. Rev. 60 1996 301 315
6. G.H. Posner, and P.M. O'Neill J. Med. Chem. 47 2004 2945 2964
7. M. Jung, X. Li, D.A. Bustos, H.N. Elsohly, and J.D. McChesney Tetrahedron Lett. 30 1989 5973 5976
8. M. Jung, D.A. Bustos, H.N. Elsohly, and J.D. McChesney Synlett 1990 743 744
9. M. Jung, and S. Lee Heterocycles 45 1997 1055 1058
10. R.K. Haynes, and S.C. Vonwiller Synlett 1992 481 483
11. S.H. Woo, M.H. Parker, P. Ploypradith, J. Northrop, and G.H. Posner Tetrahedron Lett. 39 1998 1533 1536
12. M. Jung, and S. Lee Bioorg. Med. Chem. Lett. 7 1997 1091 1094
13. Tri, M. V.; Vu, T. K; Cuong. P. V. Synthesis of New 12- Aryldeoxoartemsinins. The Ninth Asian Symposium on Medicinal Plants, Spices and other Natural Products, (ASOMPS IX), Hanoi, Vietnam, September, 1998; pp 132-135
14. M.V. Tri, N.V. Tuyen, and P.V. Cuong Synthesis of new artemisinin derivatives containing C-C bond at 12 position Vietnamese J. Chem. 35 1997 11 14
15. M. Jung, and S. Lee Bioorg. Med. Chem. Lett. 8 1998 1003 1006
16. N.V. Tuyen, T.K. Vu, T.V. Sung, and P.V. Cuong Discovery of the antimalarial activity of new derivatives of artemisinin Vietnamese J. Chem. 40 2002 124 126
17. Y.M. Pu, and H. Ziffer J. Med. Chem. 38 1995 613 616
18. S. Hindley, S.A. Ward, R.C. Storr, N.L. Searle, P.G. Bray, B.K. Park, J. Davies, and P.M. O'Neill J. Med. Chem. 45 2002 1052 1063
19. P.M. O'Neill, N.L. Searle, K.W. Kan, R.C. Storr, J.L. Maggs, S.A. Ward, and B.K. Park J. Med. Chem. 42 1999 5487 5493
20. J. Ma, E. Katz, D.E. Kyle, and H. Ziffer J. Med. Chem. 43 2000 4228 4232
21. W. Trager, and J.B. Jensen Science 193 1976 673 677
22. Makler Am. J. Trop. Med. Hyg. 48 1993 7339 7341
23. +
24. +