메뉴 건너뛰기




Volumn 19, Issue 1, 2005, Pages 9-30

Radiometallation of receptor-specific peptides for diagnosis and treatment of human cancer

Author keywords

Bombesin; Diagnosis; Peptides; Radionuclide; Review; Somatostatin; Therapy

Indexed keywords

ASTATINE 211; BISMUTH; BISMUTH 212; CADMIUM DERIVATIVE; COPPER 64; GALLIUM 67; GALLIUM 68; HOLMIUM; HOLMIUM 166; INDIUM; INDIUM 111; LUTETIUM; LUTETIUM 177; MOLYBDENUM; PENTETREOTIDE; PENTETREOTIDE IN 111; PEPTIDE DERIVATIVE; PROMETHIUM; PROMETHIUM 149; RADIOISOTOPE; RADIOPHARMACEUTICAL AGENT; RHENIUM 186; RHENIUM 188; RHODIUM; RHODIUM 105; SAMARIUM 153; TECHNETIUM 99M; UNCLASSIFIED DRUG; UNINDEXED DRUG; YTTRIUM; YTTRIUM 86; YTTRIUM 90;

EID: 16244378596     PISSN: 0258851X     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Review
Times cited : (32)

References (186)
  • 2
    • 2142784588 scopus 로고
    • Radiolabeling of antibodies for targeted diagnostics
    • Boca Raton, FL, CRC Press, Inc
    • Fritzberg AR and Wilbur DS: Radiolabeling of antibodies for targeted diagnostics. In: Targeted Delivery of Imaging Agents. Boca Raton, FL, CRC Press, Inc., 1995, pp 83-101.
    • (1995) Targeted Delivery of Imaging Agents , pp. 83-101
    • Fritzberg, A.R.1    Wilbur, D.S.2
  • 3
    • 0026648277 scopus 로고
    • Radioimmunodetection in cancer identification
    • Goldenberg DM and Larson SM: Radioimmunodetection in cancer identification. J Nucl Med 33: 803-814, 1992.
    • (1992) J. Nucl. Med. , vol.33 , pp. 803-814
    • Goldenberg, D.M.1    Larson, S.M.2
  • 5
    • 0024505574 scopus 로고
    • Delivery of novel therapeutic agents in tumors: Physiological barriers and strategies
    • Jain RK: Delivery of novel therapeutic agents in tumors: physiological barriers and strategies. J Natl Cancer Inst 81: 570-576, 1989.
    • (1989) J. Natl. Cancer Inst. , vol.81 , pp. 570-576
    • Jain, R.K.1
  • 7
    • 0000594222 scopus 로고
    • The design of site-directed radiopharmaceuticals for use in drug discovery
    • (Burns HD, Gibson RE, Dannals R and Siegl P, eds), Boston, Birkhauser
    • Eckelman, WC and Gibson RE: The design of site-directed radiopharmaceuticals for use in drug discovery. In: Nuclear Imaging in Drug Discovery, Development, and Approval (Burns HD, Gibson RE, Dannals R and Siegl P, eds), Boston, Birkhauser, 1993, pp 113-134.
    • (1993) Nuclear Imaging in Drug Discovery, Development, and Approval , pp. 113-134
    • Eckelman, W.C.1    Gibson, R.E.2
  • 8
  • 9
    • 0027197170 scopus 로고
    • Selective coupling of methotrexate to peptide hormone carriers through a gamma-carboxamide linkage of its glutamic acid moiety: Benzotriazol-1-yloxytris(dimethylamino)phosphonium hexafluorophosphate activation in salt coupling
    • Nagy A, Szoke B and Schally AV: Selective coupling of methotrexate to peptide hormone carriers through a gamma-carboxamide linkage of its glutamic acid moiety: benzotriazol-1-yloxytris(dimethylamino)phosphonium hexafluorophosphate activation in salt coupling. Proc Natl Acad Sci USA 90: 6373-6376, 1993.
    • (1993) Proc. Natl. Acad. Sci. USA , vol.90 , pp. 6373-6376
    • Nagy, A.1    Szoke, B.2    Schally, A.V.3
  • 10
    • 0028825878 scopus 로고
    • Neuropeptide receptors in health and disease: The molecular basis for in vivo imaging
    • Reubi JC: Neuropeptide receptors in health and disease: the molecular basis for in vivo imaging. J Nucl Med 36: 1825-1835, 1995.
    • (1995) J. Nucl. Med. , vol.36 , pp. 1825-1835
    • Reubi, J.C.1
  • 11
    • 0025851490 scopus 로고
    • Receptors on tumors studied with radionuclide scintigraphy
    • Larson S: Receptors on tumors studied with radionuclide scintigraphy. J Nucl Med 32: 1189-1191, 1991.
    • (1991) J. Nucl. Med. , vol.32 , pp. 1189-1191
    • Larson, S.1
  • 12
    • 0028071856 scopus 로고
    • Inhibitory effects of analogs of luteinizing hormone-releasing hormone on the growth of the androgen-independent Dunning R-3327-AT-1 rat prostate cancer
    • Pinski J, Reile H, Halmos G, Groot K and Schally AV: Inhibitory effects of analogs of luteinizing hormone-releasing hormone on the growth of the androgen-independent Dunning R-3327-AT-1 rat prostate cancer. Int J Cancer 59: 51-55, 1994.
    • (1994) Int. J. Cancer , vol.59 , pp. 51-55
    • Pinski, J.1    Reile, H.2    Halmos, G.3    Groot, K.4    Schally, A.V.5
  • 13
    • 0028889369 scopus 로고
    • In vitro identification of vasoactive intestinal peptide receptors in human tumors: Implications for tumor imaging
    • Reubi JC: In vitro identification of vasoactive intestinal peptide receptors in human tumors: implications for tumor imaging. J Nucl Med 36: 1846-1853, 1995.
    • (1995) J. Nucl. Med. , vol.36 , pp. 1846-1853
    • Reubi, J.C.1
  • 14
    • 0027995452 scopus 로고
    • Octreotide scintigraphy for small cell lung carcinoma: Past, present or future?
    • Stokkel MP and Pauwels EK: Octreotide scintigraphy for small cell lung carcinoma: past, present or future? Eur J Nucl Med 21: 1276-1278, 1994.
    • (1994) Eur. J. Nucl. Med. , vol.21 , pp. 1276-1278
    • Stokkel, M.P.1    Pauwels, E.K.2
  • 16
    • 0035155042 scopus 로고    scopus 로고
    • Bifunctional chelators for therapeutic lanthanide radiopharmaceuticals
    • Liu S and Edwards DS: Bifunctional chelators for therapeutic lanthanide radiopharmaceuticals. Bioconjugate Chem 12: 7-34, 2001.
    • (2001) Bioconjugate Chem. , vol.12 , pp. 7-34
    • Liu, S.1    Edwards, D.S.2
  • 17
    • 0032573089 scopus 로고    scopus 로고
    • Design and characterization of alpha-melanotropin peptide analogs cyclized through rhenium and technetium metal coordination
    • Giblin MF, Wang N, Hoffman TJ, Jurisson SS and Quinn TP: Design and characterization of alpha-melanotropin peptide analogs cyclized through rhenium and technetium metal coordination. Proc Natl Acad Sci USA 95: 12814-12818, 1998.
    • (1998) Proc. Natl. Acad. Sci. USA , vol.95 , pp. 12814-12818
    • Giblin, M.F.1    Wang, N.2    Hoffman, T.J.3    Jurisson, S.S.4    Quinn, T.P.5
  • 19
    • 0033594253 scopus 로고    scopus 로고
    • 64Cu-labeled somatostatin analogues in vitro and in a tumor-bearing rat model: Evaluation of new derivatives for positron emission tomography imaging and targeted radiotherapy
    • 64Cu-labeled somatostatin analogues in vitro and in a tumor-bearing rat model: evaluation of new derivatives for positron emission tomography imaging and targeted radiotherapy. J Med Chem 42: 1341-1347, 1999.
    • (1999) J. Med. Chem. , vol.42 , pp. 1341-1347
    • Lewis, J.S.1    Lewis, M.R.2    Srinivasan, A.3    Schmidt, M.A.4    Wang, J.5    Anderson, C.J.6
  • 22
    • 0033926430 scopus 로고    scopus 로고
    • Radio-labeled receptor-binding peptides: A new class of radiopharmaceuticals
    • Boerman OC, Oyen WJG and Corstens FHM: Radio-labeled receptor-binding peptides: a new class of radiopharmaceuticals. Sern Nucl Med 30: 195-208, 2000.
    • (2000) Sem. Nucl. Med. , vol.30 , pp. 195-208
    • Boerman, O.C.1    Oyen, W.J.G.2    Corstens, F.H.M.3
  • 23
    • 0033233437 scopus 로고    scopus 로고
    • 99mTc-labelled peptide-based radiopharmaceuticals: An overview
    • 99mTc-labelled peptide-based radiopharmaceuticals: an overview. Nuclear Med Commun 20 1093-1112, 1999.
    • (1999) Nuclear Med. Commun. , vol.20 , pp. 1093-1112
    • Okarvi, S.V.1
  • 27
    • 0001579481 scopus 로고    scopus 로고
    • Radiometal-labeled agents (non-technetium) for diagnostic imaging
    • Anderson CJ and Welch MJ: Radiometal-labeled agents (non-technetium) for diagnostic imaging. Chem Rev 99: 2219-2234, 1999.
    • (1999) Chem. Rev. , vol.99 , pp. 2219-2234
    • Anderson, C.J.1    Welch, M.J.2
  • 28
    • 11444251794 scopus 로고
    • Coordination compounds in nuclear medicine
    • Jurisson S, Berning D, Jia W and Ma D: Coordination compounds in nuclear medicine. Chem Rev 93: 1137-1156, 1993.
    • (1993) Chem. Rev. , vol.93 , pp. 1137-1156
    • Jurisson, S.1    Berning, D.2    Jia, W.3    Ma, D.4
  • 29
    • 0001294083 scopus 로고    scopus 로고
    • Potential technetium small molecule radiopharmaceuticals
    • Jurisson S and Lydon JD: Potential technetium small molecule radiopharmaceuticals. Chem Rev 99: 2205-2218, 1999.
    • (1999) Chem. Rev. , vol.99 , pp. 2205-2218
    • Jurisson, S.1    Lydon, J.D.2
  • 30
    • 0008883289 scopus 로고    scopus 로고
    • 99mTc-labeled small peptides as diagnostic radiopharmaceuticals
    • 99mTc-labeled small peptides as diagnostic radiopharmaceuticals. Chem Rev 99: 2235-2268, 1999.
    • (1999) Chem. Rev. , vol.99 , pp. 2235-2268
    • Liu, S.1    Edwards, D.S.2
  • 31
    • 0004045544 scopus 로고    scopus 로고
    • Fifteenth Edition. Copyright©1996, General Electric Co. and KAPL Inc.
    • Chart of the Nuclides, Fifteenth Edition. Copyright©1996, General Electric Co. and KAPL Inc..
    • Chart of the Nuclides
  • 32
    • 0345114077 scopus 로고
    • Hard and soft acids and bases
    • Pearson RG: Hard and soft acids and bases. J Am Chem Soc 22: 3533-3539, 1963.
    • (1963) J. Am. Chem. Soc. , vol.22 , pp. 3533-3539
    • Pearson, R.G.1
  • 36
    • 0027139813 scopus 로고
    • Measurement of pharmacokinetics of yttrium-86 radiopharmaceuticals with PET and radiation dose calculation of analogous yttrium-90 radiotherapeutics
    • Herzog H, Rosch F, Stocklin G, Lueders C, Qaim SM and Feinendegen LE: Measurement of pharmacokinetics of yttrium-86 radiopharmaceuticals with PET and radiation dose calculation of analogous yttrium-90 radiotherapeutics. J Nucl Med 34: 2222, 1993.
    • (1993) J. Nucl. Med. , vol.34 , pp. 2222
    • Herzog, H.1    Rosch, F.2    Stocklin, G.3    Lueders, C.4    Qaim, S.M.5    Feinendegen, L.E.6
  • 38
    • 0012725753 scopus 로고    scopus 로고
    • Therapeutic radiopharmaceuticals
    • Volkert WA and Hoffman TJ: Therapeutic radiopharmaceuticals. Chem Rev 99: 2269-2292, 1999.
    • (1999) Chem. Rev. , vol.99 , pp. 2269-2292
    • Volkert, W.A.1    Hoffman, T.J.2
  • 39
    • 0001630977 scopus 로고
    • Chemical and structural approaches to rational drug design
    • Weiner DB, Williams MV, eds. Boca Raton, FL, CRC Press
    • Fritzberg AR, Gustavson LM, Hylarides MD and Reno JM: Chemical and structural approaches to rational drug design. In: Weiner DB, Williams MV, eds. Boca Raton, FL, CRC Press, p 125, 1995.
    • (1995) , pp. 125
    • Fritzberg, A.R.1    Gustavson, L.M.2    Hylarides, M.D.3    Reno, J.M.4
  • 40
    • 0030111464 scopus 로고    scopus 로고
    • Vehicles, chelators, and radionuclides: Choosing the "building blocks" of an effective therapeutic radioimmunoconjugate
    • Schubiger PA, Alberto R and Smith A: Vehicles, chelators, and radionuclides: choosing the "building blocks" of an effective therapeutic radioimmunoconjugate. Bioconjugate Chem 7: 165-179, 1996.
    • (1996) Bioconjugate Chem. , vol.7 , pp. 165-179
    • Schubiger, P.A.1    Alberto, R.2    Smith, A.3
  • 41
  • 42
    • 0032053948 scopus 로고    scopus 로고
    • Reactor-produced radionuclides at the University of Missouri Research Reactor
    • Ehrhardt GJ, Ketring AR and Ayers LM: Reactor-produced radionuclides at the University of Missouri Research Reactor. Appl Radiat Isot 49: 295-297, 1998.
    • (1998) Appl. Radiat. Isot. , vol.49 , pp. 295-297
    • Ehrhardt, G.J.1    Ketring, A.R.2    Ayers, L.M.3
  • 44
    • 0028965789 scopus 로고
    • Radiolabeling with technetium-99m to study high-capacity and low-capacity biochemical systems
    • Eckelman WC: Radiolabeling with technetium-99m to study high-capacity and low-capacity biochemical systems. Eur J Nucl Med 22 249, 1995.
    • (1995) Eur. J. Nucl. Med. , vol.22 , pp. 249
    • Eckelman, W.C.1
  • 45
    • 0347991822 scopus 로고    scopus 로고
    • Gastrin releasing peptide (GRP) receptor targeted radiopharmaceuticals: A concise update
    • Smith CJ, Volkert WA and Hoffman TJ: Gastrin releasing peptide (GRP) receptor targeted radiopharmaceuticals: a concise update. Nucl Med Biol 30: 861-868, 2002.
    • (2002) Nucl. Med. Biol. , vol.30 , pp. 861-868
    • Smith, C.J.1    Volkert, W.A.2    Hoffman, T.J.3
  • 47
    • 0025198361 scopus 로고
    • Labeling of hematoporphyrin with Rhodium-105 and binding studies with human gamma globulin
    • Pillai MRA, Lo JM and Troutner DE: Labeling of hematoporphyrin with Rhodium-105 and binding studies with human gamma globulin. Appl Radiat Isot 41: 69-73, 1990.
    • (1990) Appl. Radiat. Isot. , vol.41 , pp. 69-73
    • Pillai, M.R.A.1    Lo, J.M.2    Troutner, D.E.3
  • 49
    • 0001311976 scopus 로고    scopus 로고
    • Rhodium (III) complexes with acyclic tetrathioether ligands. Effects of backbone chain length on the conjugation of the Rh. (III)complex
    • Goswami M, Alberto R, Barnes CL and Jurisson S: Rhodium (III) complexes with acyclic tetrathioether ligands. Effects of backbone chain length on the conjugation of the Rh (III)complex. Inorg Chem 35: 7546-755, 1996.
    • (1996) Inorg. Chem. , vol.35 , pp. 7546-8755
    • Goswami, M.1    Alberto, R.2    Barnes, C.L.3    Jurisson, S.4
  • 51
    • 0028217085 scopus 로고
    • Relative biological effectiveness of alpha-particle emitters in vivo at low doses
    • Howell RW, Azure MT, Narra VR and Rao DV: Relative biological effectiveness of alpha-particle emitters in vivo at low doses. Radiat Res 137: 352-360, 1994.
    • (1994) Radiat. Res. , vol.137 , pp. 352-360
    • Howell, R.W.1    Azure, M.T.2    Narra, V.R.3    Rao, D.V.4
  • 52
    • 0011736580 scopus 로고
    • Bismuth-212-labeled anti-TAC monoclonal antibody: Alpha-particle-emitting radionuclides as modalities for radiommumotherapy
    • Kozak RW, Atcher RW, Gansow OA, Friedman AM, Hines JJ and Waldman TA: Bismuth-212-labeled anti-TAC monoclonal antibody: alpha-particle-emitting radionuclides as modalities for radiommumotherapy. Proc Natl Acad Sci USA 83 (2): 474-478, 1986.
    • (1986) Proc. Natl. Acad. Sci. USA , vol.83 , Issue.2 , pp. 474-478
    • Kozak, R.W.1    Atcher, R.W.2    Gansow, O.A.3    Friedman, A.M.4    Hines, J.J.5    Waldman, T.A.6
  • 53
    • 0030013280 scopus 로고    scopus 로고
    • Radioimmunotherapy with alpha-particle emitting radioimmunoconjugates
    • Zalutsky MR and Bigner DD: Radioimmunotherapy with alpha-particle emitting radioimmunoconjugates. Acta Oncol 35: 373-379, 1996.
    • (1996) Acta Oncol. , vol.35 , pp. 373-379
    • Zalutsky, M.R.1    Bigner, D.D.2
  • 56
    • 0033233437 scopus 로고    scopus 로고
    • 99mTc-labelled peptide-based radiopharmaceuticals
    • 99mTc-labelled peptide-based radiopharmaceuticals. Nucl Med Commun 20: 1093-1112, 1999.
    • (1999) Nucl. Med. Commun. , vol.20 , pp. 1093-1112
    • Okarvi, S.V.1
  • 59
    • 0027389181 scopus 로고
    • Rhenium-186-labeled monoclonal antibodies for radioimmunotherapy: Preparation and evaluation
    • John E, Thakur ML, DeFulvio J, McDevitt MR and Damjanov I: Rhenium-186-labeled monoclonal antibodies for radioimmunotherapy: preparation and evaluation. J Nucl Med 34: 260-267, 1993.
    • (1993) J. Nucl. Med. , vol.34 , pp. 260-267
    • John, E.1    Thakur, M.L.2    DeFulvio, J.3    McDevitt, M.R.4    Damjanov, I.5
  • 61
    • 34249288481 scopus 로고
    • Antibody radiolabeling, problems and promises
    • Hnatowich DJ: Antibody radiolabeling, problems and promises. Nucl Med Biol 17: 49-55, 1990.
    • (1990) Nucl. Med. Biol. , vol.17 , pp. 49-55
    • Hnatowich, D.J.1
  • 62
    • 0016290352 scopus 로고
    • Selective binding of metal ions to macromolecules using bifunctional analogs of EDTA
    • Sundberg MW, Meares CF, Goodwin DA and Diamanti CI: Selective binding of metal ions to macromolecules using bifunctional analogs of EDTA. J Med Chem 17: 1304, 1974.
    • (1974) J. Med. Chem. , vol.17 , pp. 1304
    • Sundberg, M.W.1    Meares, C.F.2    Goodwin, D.A.3    Diamanti, C.I.4
  • 64
    • 0028327118 scopus 로고
    • Synthesis, radiochemistry and biological evaluation of a new somatostatin analogue(SDZ 219-387) labeled with technetium-99m
    • Maina T, Stolz B, Albert R, Bruns C, Koch P and Macke H: Synthesis, radiochemistry and biological evaluation of a new somatostatin analogue(SDZ 219-387) labeled with technetium-99m. Eur J Nucl Med 21 437, 1994.
    • (1994) Eur. J. Nucl. Med. , vol.21 , pp. 437
    • Maina, T.1    Stolz, B.2    Albert, R.3    Bruns, C.4    Koch, P.5    Macke, H.6
  • 66
    • 0001279485 scopus 로고
    • Technetium (V) and rhenium (V) complexes of 2,3-bis (mercaptoacetamido)propanoate. Chelate ring stereochemistry and influence on chemical and biological properties
    • Rao TN, Adhikesavalu D, Camerman A and Fritzberg AR: Technetium (V) and rhenium (V) complexes of 2,3-bis (mercaptoacetamido)propanoate. Chelate ring stereochemistry and influence on chemical and biological properties. J Am Chem Soc 112: 5798, 1990.
    • (1990) J. Am. Chem. Soc. , vol.112 , pp. 5798
    • Rao, T.N.1    Adhikesavalu, D.2    Camerman, A.3    Fritzberg, A.R.4
  • 67
    • 0023205303 scopus 로고
    • Animal evaluation of technetium-99m triamide mercaptide complexes as potential renal imaging agents
    • Eshima D, Taylor A, Fritzberg AR, Kasina S, Hansen L and Sorenson JF: Animal evaluation of technetium-99m triamide mercaptide complexes as potential renal imaging agents. J Nucl Med 28: 1180, 1987.
    • (1987) J. Nucl. Med. , vol.28 , pp. 1180
    • Eshima, D.1    Taylor, A.2    Fritzberg, A.R.3    Kasina, S.4    Hansen, L.5    Sorenson, J.F.6
  • 70
    • 0000962810 scopus 로고
    • Synthesis, characterization, and x-ray structural determinations of technetium(V)-oxo-tetradentate amine oxime complexes
    • Jurisson S, Schlemper EO, Troutner DE, Canning LR, Nowotnik DP and Neirinckx RD: Synthesis, characterization, and x-ray structural determinations of technetium(V)-oxo-tetradentate amine oxime complexes. Inorg Chem 25(4): 543-549, 1986.
    • (1986) Inorg. Chem. , vol.25 , Issue.4 , pp. 543-549
    • Jurisson, S.1    Schlemper, E.O.2    Troutner, D.E.3    Canning, L.R.4    Nowotnik, D.P.5    Neirinckx, R.D.6
  • 76
    • 0028815077 scopus 로고
    • 99mTc-labeled hydrazino nicotinic acid derivatized chemotactic peptides
    • 99mTc-labeled hydrazino nicotinic acid derivatized chemotactic peptides. Nucl Med Biol 22: 25-30, 1995.
    • (1995) Nucl. Med. Biol. , vol.22 , pp. 25-30
    • Babich, J.W.1    Fischman, A.J.2
  • 77
    • 0032766066 scopus 로고    scopus 로고
    • Technetium-99m somatostatin analogues: Effect of labelling methods and peptide sequence
    • Decristoforo C and Mather SJ: Technetium-99m somatostatin analogues: effect of labelling methods and peptide sequence. Eur J Nucl Med 26: 869-876, 1999.
    • (1999) Eur. J. Nucl. Med. , vol.26 , pp. 869-876
    • Decristoforo, C.1    Mather, S.J.2
  • 80
    • 0032588840 scopus 로고    scopus 로고
    • 99mTc-HYNIC-folate: A novel receptor-based targeted radiopharmaceutical for tumor imaging
    • 99mTc-HYNIC-folate: A novel receptor-based targeted radiopharmaceutical for tumor imaging. J Nucl Med 40: 1563-1569, 1999.
    • (1999) J. Nucl. Med. , vol.40 , pp. 1563-1569
    • Guo, W.1    Hinkle, G.H.2    Lee, R.J.3
  • 81
    • 0032984811 scopus 로고    scopus 로고
    • 99mTc-technetium-labelled peptide-HYNIC conjugates: Effects of lipophilicity and stability on biodistribution
    • 99mTc-technetium-labelled peptide-HYNIC conjugates: effects of lipophilicity and stability on biodistribution. Nucl Med Biol 26: 389-396, 1999.
    • (1999) Nucl. Med. Biol. , vol.26 , pp. 389-396
    • Decristoforo, C.1    Mather, S.2
  • 82
    • 0037262667 scopus 로고    scopus 로고
    • Synthesis of target-specific radiolabeled peptides for diagnostic imaging
    • Fichna J and Janecka A: Synthesis of target-specific radiolabeled peptides for diagnostic imaging. Bioconj Chem 14: 3-17, 2003.
    • (2003) Bioconj. Chem. , vol.14 , pp. 3-17
    • Fichna, J.1    Janecka, A.2
  • 84
    • 0345055302 scopus 로고    scopus 로고
    • 99mTc-labeling of hydrazino nicotinamide-modified biologically active molecules using imine-N-containing heterocycles as coligands
    • 99mTc-labeling of hydrazino nicotinamide-modified biologically active molecules using imine-N-containing heterocycles as coligands. Bioconj Chem 9: 583-595, 1998.
    • (1998) Bioconj. Chem. , vol.9 , pp. 583-595
    • Liu, S.1    Edwards, D.S.2    Harris, A.R.3
  • 86
    • 0023906928 scopus 로고
    • Radiohalogenation of a monoclonal antibody using an N-succinimidyl 3-(tri-n-butylstannyl) benzoate intermediate
    • Zalutsky MR and Narula AS: Radiohalogenation of a monoclonal antibody using an N-succinimidyl 3-(tri-n-butylstannyl) benzoate intermediate. Cancer Res 48: 1446-1450, 1988.
    • (1988) Cancer Res. , vol.48 , pp. 1446-1450
    • Zalutsky, M.R.1    Narula, A.S.2
  • 92
    • 0000704180 scopus 로고    scopus 로고
    • 3]2-. Synthesis, characterization, and structures of rhenium(I) tricarbonyl complexes with thiourea and thiourea derivatives
    • 3]2-. Synthesis, characterization, and structures of rhenium(I) tricarbonyl complexes with thiourea and thiourea derivatives. Inorg Chem Acta 248: 193-202, 1996.
    • (1996) Inorg. Chem. Acta , vol.248 , pp. 193-202
    • Abram, U.1    Abram, S.2    Alberto, R.3    Schibli, R.4
  • 96
    • 0026161977 scopus 로고
    • A convenient synthesis of bifunctional chelating agents based on diethylenetriaminepentaacetic acid and their coordination chemistry with yttrium (III)
    • Cummins CH, Rutter EW Jr and Fordyce WA: A convenient synthesis of bifunctional chelating agents based on diethylenetriaminepentaacetic acid and their coordination chemistry with yttrium (III). Bioconj Chem 2: 18-186, 1991.
    • (1991) Bioconj. Chem. , vol.2 , pp. 18-186
    • Cummins, C.H.1    Rutter Jr., E.W.2    Fordyce, W.A.3
  • 100
    • 0001353258 scopus 로고    scopus 로고
    • 2 conjugate for specific targeting of tumors expressing gastrin releasing peptide receptors (GRP-R)
    • 2 conjugate for specific targeting of tumors expressing gastrin releasing peptide receptors (GRP-R). J Nucl Med (Supplement) 41(5): 119P, 2000.
    • (2000) J. Nucl. Med. , vol.41 , Issue.5 SUPPL.
    • Gali, H.1    Hoffman, T.J.2    Owen, N.K.3    Sieckman, G.L.4    Volkert, W.A.5
  • 102
    • 0034976943 scopus 로고    scopus 로고
    • Radiometallated receptor-avid peptide conjugates for specific in vivo targeting of cancer cells
    • Hoffman TJ, Quinn TP and Volkert WA: Radiometallated receptor-avid peptide conjugates for specific in vivo targeting of cancer cells. Nucl Med Biol 28: 527-539, 2001.
    • (2001) Nucl. Med. Biol. , vol.28 , pp. 527-539
    • Hoffman, T.J.1    Quinn, T.P.2    Volkert, W.A.3
  • 106
    • 0042854927 scopus 로고    scopus 로고
    • Peptide receptors as molecular targets for cancer diagnosis and therapy
    • Reubi JC: Peptide receptors as molecular targets for cancer diagnosis and therapy. Endocrine Rev 24: 389-427, 2003.
    • (2003) Endocrine Rev. , vol.24 , pp. 389-427
    • Reubi, J.C.1
  • 108
    • 1542472268 scopus 로고    scopus 로고
    • Molecular targeting with radionuclides: State of the science
    • Britz-Cunningham SH and Adelstein SJ: Molecular targeting with radionuclides: state of the science. J Nucl Med 44: 1945-1961, 2003.
    • (2003) J. Nucl. Med. , vol.44 , pp. 1945-1961
    • Britz-Cunningham, S.H.1    Adelstein, S.J.2
  • 111
    • 0036415073 scopus 로고    scopus 로고
    • Somatostatin analogs and radiopeptides in cancer therapy
    • Froidevaux S and Eberle AN: Somatostatin analogs and radiopeptides in cancer therapy. Biopolymers 66: 161-183, 2002.
    • (2002) Biopolymers , vol.66 , pp. 161-183
    • Froidevaux, S.1    Eberle, A.N.2
  • 121
    • 0034790290 scopus 로고    scopus 로고
    • Between the Scylla and Charybdis of peptide radionuclide therapy: Hitting the tumor and saving the kidney
    • Boerman OC, Oyen WJG and Corstens FHM: Between the Scylla and Charybdis of peptide radionuclide therapy: hitting the tumor and saving the kidney. Eur J Nucl Med 28: 1447-1449, 2001.
    • (2001) Eur. J. Nucl. Med. , vol.28 , pp. 1447-1449
    • Boerman, O.C.1    Oyen, W.J.G.2    Corstens, F.H.M.3
  • 123
    • 0015296908 scopus 로고
    • Isolation and amino acid sequences of alytesin and bombesin, two analogous active tetradecapeptides from the skin of european discoglossid frogs
    • Anastasi A, Erspamer V and Nucci M: Isolation and amino acid sequences of alytesin and bombesin, two analogous active tetradecapeptides from the skin of european discoglossid frogs. Arch Biochem Biophys 148: 443-446, 1972.
    • (1972) Arch. Biochem. Biophys. , vol.148 , pp. 443-446
    • Anastasi, A.1    Erspamer, V.2    Nucci, M.3
  • 124
    • 0021244729 scopus 로고
    • The contractile effect of bombesin, gastrin releasing peptide and various fragments in the rat stomach strip
    • Girard F, Bachelard H, St-Pierre S and Rioux F: The contractile effect of bombesin, gastrin releasing peptide and various fragments in the rat stomach strip. Eur J Pharmacol 102: 489-497, 1984.
    • (1984) Eur. J. Pharmacol. , vol.102 , pp. 489-497
    • Girard, F.1    Bachelard, H.2    St-Pierre, S.3    Rioux, F.4
  • 126
    • 0025606853 scopus 로고
    • Cloning and functional characterization of a complementary DNA encoding the murine fibroblast bombesin/gastrin releasing peptide receptor
    • Spindel ER, Giladi E, Brehm P, Goodman RH and Segerson TP: Cloning and functional characterization of a complementary DNA encoding the murine fibroblast bombesin/gastrin releasing peptide receptor. Mol Endocrinol 4: 1956-1963, 1990.
    • (1990) Mol. Endocrinol. , vol.4 , pp. 1956-1963
    • Spindel, E.R.1    Giladi, E.2    Brehm, P.3    Goodman, R.H.4    Segerson, T.P.5
  • 130
    • 0023833532 scopus 로고
    • The bombesin receptor is coupled to a guanine nucleotide-binding protein which is insensitive to pertussis and cholera toxins
    • Fischer JB and Schonbrunn A: The bombesin receptor is coupled to a guanine nucleotide-binding protein which is insensitive to pertussis and cholera toxins. J Biol Chem 263: 2808-2816, 1988.
    • (1988) J. Biol. Chem. , vol.263 , pp. 2808-2816
    • Fischer, J.B.1    Schonbrunn, A.2
  • 131
    • 0033104343 scopus 로고    scopus 로고
    • Gastrin releasing peptide receptors in the human prostate: Relation to neoplastic transformation
    • Markwalder R and Reubi JC: Gastrin releasing peptide receptors in the human prostate: relation to neoplastic transformation. Cancer Res 59: 1152-1159, 1999.
    • (1999) Cancer Res. , vol.59 , pp. 1152-1159
    • Markwalder, R.1    Reubi, J.C.2
  • 132
    • 0033953894 scopus 로고    scopus 로고
    • Presence of receptors for bombesin/gastrin-releasing peptide and mRNA for three receptor subtypes in human prostate cancers
    • Sun B, Halmos G, Schally AV, Wang X and Martinez M: Presence of receptors for bombesin/gastrin-releasing peptide and mRNA for three receptor subtypes in human prostate cancers. Prostate 42: 295-303, 2000.
    • (2000) Prostate , vol.42 , pp. 295-303
    • Sun, B.1    Halmos, G.2    Schally, A.V.3    Wang, X.4    Martinez, M.5
  • 133
    • 0028894264 scopus 로고
    • Characterization of bombesin/gastrin-releasing peptide receptors in human breast cancer and their relationship to steroid receptor expression
    • Halmos G, Wittliff JL and Schally AV: Characterization of bombesin/gastrin-releasing peptide receptors in human breast cancer and their relationship to steroid receptor expression. Cancer Res 55: 280-287, 1995.
    • (1995) Cancer Res. , vol.55 , pp. 280-287
    • Halmos, G.1    Wittliff, J.L.2    Schally, A.V.3
  • 134
    • 0032804044 scopus 로고    scopus 로고
    • Gastrin-releasing peptide receptors in non-neoplastic and neoplastic human breast
    • Gugger M and Reubi JC: Gastrin-releasing peptide receptors in non-neoplastic and neoplastic human breast. Am J Pathol 155: 2067-2076, 1999.
    • (1999) Am. J. Pathol. , vol.155 , pp. 2067-2076
    • Gugger, M.1    Reubi, J.C.2
  • 135
    • 0030298095 scopus 로고    scopus 로고
    • Clinical correlates of bombesin-like peptide receptor subtype expression in human lung cancer cells
    • Toi-Scott M, Jones CL and Kane MA: Clinical correlates of bombesin-like peptide receptor subtype expression in human lung cancer cells. Lung Cancer 15: 341-354, 1996.
    • (1996) Lung Cancer , vol.15 , pp. 341-354
    • Toi-Scott, M.1    Jones, C.L.2    Kane, M.A.3
  • 136
    • 0032032589 scopus 로고    scopus 로고
    • Design, synthesis, and initial evaluation of high-affinity technetium bombesin analogues
    • Baidoo KE, Lin K-S, Zhan Y, Finley P, Scheffel U and Wagner HN: Design, synthesis, and initial evaluation of high-affinity technetium bombesin analogues. Bioconj Chem 9: 218-225, 1998.
    • (1998) Bioconj. Chem. , vol.9 , pp. 218-225
    • Baidoo, K.E.1    Lin, K.-S.2    Zhan, Y.3    Finley, P.4    Scheffel, U.5    Wagner, H.N.6
  • 148
    • 0023609864 scopus 로고
    • Influence of stereochemistry of the sequence Arg-Gly-Asp-Xaa on binding specificity in cell adhesion
    • Pierschbacher MD and Ruoslahti E: Influence of stereochemistry of the sequence Arg-Gly-Asp-Xaa on binding specificity in cell adhesion. J Biol Chem 262: 17294-17298, 1987.
    • (1987) J. Biol. Chem. , vol.262 , pp. 17294-17298
    • Pierschbacher, M.D.1    Ruoslahti, E.2
  • 149
    • 0037131442 scopus 로고    scopus 로고
    • The structures of integrins and integrin-ligand complexes: Implications for drug design and signal transduction
    • Gottschalk K and Kessler H: The structures of integrins and integrin-ligand complexes: implications for drug design and signal transduction. Angew Chem Int Ed 41: 3767-3774, 2002.
    • (2002) Angew Chem. Int. Ed. , vol.41 , pp. 3767-3774
    • Gottschalk, K.1    Kessler, H.2
  • 150
    • 0035957050 scopus 로고    scopus 로고
    • Solution structures and integrin binding activities of an RGD peptide with two isomers
    • Assa-Munt N, Jia X, Laakkonen P and Ruoslahti E: Solution structures and integrin binding activities of an RGD peptide with two isomers. Biochemistry 40: 2373-2378, 2001.
    • (2001) Biochemistry , vol.40 , pp. 2373-2378
    • Assa-Munt, N.1    Jia, X.2    Laakkonen, P.3    Ruoslahti, E.4
  • 152
    • 2342439574 scopus 로고    scopus 로고
    • Radiolabeled tracers for imaging of tumor angiogenesis and evaluation of anti-angiogenic therapies
    • Haubner R and Wester HJ: Radiolabeled tracers for imaging of tumor angiogenesis and evaluation of anti-angiogenic therapies. Curr Pharm Des 10: 1439-1455, 2004.
    • (2004) Curr. Pharm. Des. , vol.10 , pp. 1439-1455
    • Haubner, R.1    Wester, H.J.2
  • 161
    • 0001859580 scopus 로고
    • Vasoactive intestinal polypeptide and related peptides
    • (Walsh JH and Dockray GJ, eds.) New York, Raven Press
    • Dockray GJ: Vasoactive intestinal polypeptide and related peptides. In: Gut Peptides (Walsh JH and Dockray GJ, eds.) New York, Raven Press, 1994, pp 447-472.
    • (1994) Gut Peptides , pp. 447-472
    • Dockray, G.J.1
  • 163
    • 18144453553 scopus 로고    scopus 로고
    • Vasoactive intestinal peptide/pituitary adenylate cyclase-activating peptide receptor subtypes in human tumors and their tissues of origin
    • Reubi JC, Laderach U, Waser B, Gebbers J, Robberecht P and Laissue JA: Vasoactive intestinal peptide/pituitary adenylate cyclase-activating peptide receptor subtypes in human tumors and their tissues of origin. Cancer Res 60: 3105-3112, 2000.
    • (2000) Cancer Res. , vol.60 , pp. 3105-3112
    • Reubi, J.C.1    Laderach, U.2    Waser, B.3    Gebbers, J.4    Robberecht, P.5    Laissue, J.A.6
  • 166
    • 0030773660 scopus 로고    scopus 로고
    • Receptor nuclear medicine: Vasointestinal peptide and somatostatin receptor scintigraphy for diagnosis and treatment of tumor patients
    • Virgolini I: Receptor nuclear medicine: vasointestinal peptide and somatostatin receptor scintigraphy for diagnosis and treatment of tumor patients. Eur J Clin Invest 27: 793-800, 1997.
    • (1997) Eur. J. Clin. Invest. , vol.27 , pp. 793-800
    • Virgolini, I.1
  • 174
    • 0024407943 scopus 로고
    • Characterization of receptors for alpha-melanocyte-stimulating hormone on human melanoma cells
    • Siegrist W, Solca F, Stutz S, Giuffre L, Carrel S, Girard J and Eberle AN: Characterization of receptors for alpha-melanocyte-stimulating hormone on human melanoma cells. Cancer Res 49: 6352-6358, 1989.
    • (1989) Cancer Res. , vol.49 , pp. 6352-6358
    • Siegrist, W.1    Solca, F.2    Stutz, S.3    Giuffre, L.4    Carrel, S.5    Girard, J.6    Eberle, A.N.7
  • 176
    • 0000448866 scopus 로고
    • 4-Norleucine, 7-D-phenylalanine- alpha-melanocyte-stimulating hormone: A highly potent alpha-melanotropin with ultralong biological activity
    • Sawyer TK, Sanfilippo PJ, Hruby VJ, Engel MH, Heward CB, Burnett JB and Hadley ME: 4-Norleucine, 7-D-phenylalanine-alpha- melanocyte-stimulating hormone: a highly potent alpha-melanotropin with ultralong biological activity. Proc Natl Acad Sci USA 77: 5754-5758, 1980.
    • (1980) Proc. Natl. Acad. Sci. USA , vol.77 , pp. 5754-5758
    • Sawyer, T.K.1    Sanfilippo, P.J.2    Hruby, V.J.3    Engel, M.H.4    Heward, C.B.5    Burnett, J.B.6    Hadley, M.E.7
  • 177
    • 0025694915 scopus 로고
    • A chelating derivative of alpha-melanocyte stimulating hormone as a potential imaging agent for malignant melanoma
    • Bard DR, Knight CG and Page-Thomas DP: A chelating derivative of alpha-melanocyte stimulating hormone as a potential imaging agent for malignant melanoma. Br J Cancer 62: 919-922, 1990.
    • (1990) Br. J. Cancer , vol.62 , pp. 919-922
    • Bard, D.R.1    Knight, C.G.2    Page-Thomas, D.P.3
  • 178
    • 0026504777 scopus 로고
    • The use of a chelating derivative of alpha melanocyte stimulating hormone for the clinical imaging of malignant melanoma
    • Wraight EP, Bard DR, Maughan TS, Knight CG and Page-Thomas DP: The use of a chelating derivative of alpha melanocyte stimulating hormone for the clinical imaging of malignant melanoma. Br J Radiol 65 112-118, 1992.
    • (1992) Br. J. Radiol. , vol.65 , pp. 112-118
    • Wraight, E.P.1    Bard, D.R.2    Maughan, T.S.3    Knight, C.G.4    Page-Thomas, D.P.5
  • 179
    • 0023606861 scopus 로고
    • Specific receptors for α-melanocyte-stimulating hormone are widely distributed in tissues of rodents
    • Tatro JB and Reichlin S: Specific receptors for α-melanocyte-stimulating hormone are widely distributed in tissues of rodents. Endocrinol 121: 1900-1907, 1987.
    • (1987) Endocrinol. , vol.121 , pp. 1900-1907
    • Tatro, J.B.1    Reichlin, S.2
  • 180
    • 0030091928 scopus 로고    scopus 로고
    • Enhanced binding and inertness to dehalogenation of α-melanotropic peptides labeled using N-Succinimidyl 3-iodobenzoate
    • Garg PK, Alston KL, Welsh PC and Zalutsky MR: Enhanced binding and inertness to dehalogenation of α-melanotropic peptides labeled using N-Succinimidyl 3-iodobenzoate. Bioconj Chem 7: 233-239, 1996.
    • (1996) Bioconj. Chem. , vol.7 , pp. 233-239
    • Garg, P.K.1    Alston, K.L.2    Welsh, P.C.3    Zalutsky, M.R.4
  • 181
    • 0036900073 scopus 로고    scopus 로고
    • A novel DOTA-α-melanocyte-stimulating hormone analog for metastatic melanoma diagnosis
    • Froidevaux S, Calame-Christe M, Tanner H, Sumanovski L and Eberle AN: A novel DOTA-α-melanocyte-stimulating hormone analog for metastatic melanoma diagnosis. J Nucl Med 43: 1699-1706, 2002.
    • (2002) J. Nucl. Med. , vol.43 , pp. 1699-1706
    • Froidevaux, S.1    Calame-Christe, M.2    Tanner, H.3    Sumanovski, L.4    Eberle, A.N.5
  • 185
    • 0345357056 scopus 로고    scopus 로고
    • Evaluation of the human melanoma targeting properties of radiolabeled α-stimulating hormone peptide analogues
    • Miao Y, Whitener D, Feng W, Owen NK, Chen J and Quinn TP: Evaluation of the human melanoma targeting properties of radiolabeled α-stimulating hormone peptide analogues. Bioconj Chem 14: 1177-1184, 2003.
    • (2003) Bioconj. Chem. , vol.14 , pp. 1177-1184
    • Miao, Y.1    Whitener, D.2    Feng, W.3    Owen, N.K.4    Chen, J.5    Quinn, T.P.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.