6-(2-Furanyl)-9H-purin-2-amine derivatives as A2A adenosine antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 8, 2005, Pages 2119-2122

  Kiselgof, Eugenia ^a   Tulshian, Deen B ^a   Arik, Leyla ^a   Zhang, Hongtao ^a   Fawzi, Ahmad ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

Author keywords

2 Furanyl; 9 H Purin; Adenosine receptor; Antagonist

Indexed keywords

2 AMINO 6 (2 FURANYL)PURINE; 5 AMINO 2 (2 FURYL) 7 (2 PHENYLETHYL)PYRAZOLO[4,3 E][1,2,4]TRIAZOLO[1,5 C]PYRIMIDINE; ADENOSINE A2A RECEPTOR ANTAGONIST; AMINE; PURINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; DRUG IDENTIFICATION; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; DRUG STRUCTURE; RECEPTOR AFFINITY; STRUCTURE ACTIVITY RELATION; SUBSTITUTION REACTION;

EID: 15944380474     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.02.031     Document Type: Article

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