Quantitative structure-activity analyses of bufokinin and other tachykinins at bufokinin (bNK1) receptors of the small intestine of the cane toad, Bufo marinus

Biochemical Pharmacology

Volumn 69, Issue 2, 2005, Pages 329-338

  Liu, Lu ^a   Murray, Michael ^b   Conlon, J Michael ^c   Burcher, Elizabeth ^a  

^a UNIVERSITY OF NEW SOUTH WALES   (Australia)

^b UNIVERSITY OF SYDNEY   (Australia)

^c UNITED ARAB EMIRATES UNIVERSITY   (United Arab Emirates)

Author keywords

Amphibian; Binding; Bufokinin; Functional; Intestine; Non mammalian; QSAR; Structure activity; Substance P; Tachykinin receptors; Tachykinins

Indexed keywords

BUFOKININ; KININ; PHYSALAEMIN; RANATACHYKININ; SUBSTANCE P; TACHYKININ; TACHYKININ DERIVATIVE; TACHYKININ RECEPTOR; UNCLASSIFIED DRUG; NEUROKININ 1 RECEPTOR; SIGNAL PEPTIDE;

AMINO ACID SEQUENCE; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BINDING COMPETITION; CARBOXY TERMINAL SEQUENCE; CONTROLLED STUDY; DRUG EFFECT; DRUG MECHANISM; MATHEMATICAL ANALYSIS; NONHUMAN; PRIORITY JOURNAL; PROTEIN BINDING; QUANTITATIVE STRUCTURE ACTIVITY RELATION; SMALL INTESTINE; STRUCTURE ACTIVITY RELATION; TOAD; AMINO ACID SUBSTITUTION; ANIMAL; CHEMISTRY; COMPARATIVE STUDY; DOSE RESPONSE; DRUG POTENTIATION; GENETICS; INTESTINE MUCOSA; METABOLISM; PHYSIOLOGY;

AMINO ACID SUBSTITUTION; ANIMALS; BUFO MARINUS; DOSE-RESPONSE RELATIONSHIP, DRUG; INTERCELLULAR SIGNALING PEPTIDES AND PROTEINS; INTESTINAL MUCOSA; INTESTINE, SMALL; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; RECEPTORS, NEUROKININ-1; TACHYKININS;

EID: 13844256868     PISSN: 00062952     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bcp.2004.09.023     Document Type: Article

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