Parallel bioassay of 39 tachykinins on 11 smooth muscle preparations. Structure and receptor selectivity/affinity relationship

Peptides

Volumn 21, Issue 11, 2000, Pages 1587-1595

  Severini, Cinzia ^a,c   Salvadori, Severo ^b   Guerrini, Remo ^b   Falconieri Erspamer, Giuliana ^c   Mignogna, Giuseppina ^c   Erspamer, Vittorio ^c  

^a CNR   (Italy)

^b Ferrara   (Italy)

^c SAPIENZA UNIVERSITY OF ROME   (Italy)

Author keywords

Parallel bioassay; Smooth muscle preparations; Structure Receptor selectivity relationship; Tachykinins

Indexed keywords

ALIPHATIC AMINE; NEUROKININ; TACHYKININ; TRIPEPTIDE;

AMINO ACID SEQUENCE; AMINO ACID SUBSTITUTION; ARTICLE; BINDING AFFINITY; CARBOXY TERMINAL SEQUENCE; PRIORITY JOURNAL; RECEPTOR AFFINITY; RECEPTOR BINDING; SMOOTH MUSCLE; STRUCTURE ACTIVITY RELATION;

ANIMALS; BIOLOGICAL ASSAY; GUINEA PIGS; ISOLEUCINE; MALE; MICE; MUSCLE, SMOOTH; PHENYLALANINE; PROLINE; PROTEIN BINDING; RABBITS; RATS; RATS, WISTAR; RECEPTORS, NEUROKININ-1; RECEPTORS, NEUROKININ-2; RECEPTORS, NEUROKININ-3; RECEPTORS, TACHYKININ; TACHYKININS; TYROSINE;

EID: 0033725188     PISSN: 01969781     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0196-9781(00)00290-4     Document Type: Article

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32. Historical notes
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