Technetium-99m labelled integrated tropane-BAT as a potential dopamine transporter tracer

Bioorganic and Medicinal Chemistry

Volumn 13, Issue 4, 2005, Pages 1053-1058

  Cleynhens, Bernard J ^a   De Groot, Tjibbe J ^a   Vanbilloen, Hubert P ^a   Kieffer, Davy ^a   Mortelmans, Luc ^a   Bormans, Guy M ^a   Verbruggen, Alfons M ^a  

^a UNIVERSITY HOSPITALS LEUVEN   (Belgium)

Author keywords

[No Author keywords available]

Indexed keywords

[2 [[2 [[[3 (4 CHLOROPHENYL) 8 METHYL 8 AZABICYCLO[3.2.1]OCT 2 YL]METHYL](2 MERCAPTOETHYL)AMINO]ETHYL]AMINO]ETHANETHIOLATO]OXOTECHNETIUM TC 99M; DOPAMINE TRANSPORTER; N (2' MERCAPTOETHYL) 3 BETA (4 CHLOROPHENYL) 2 BETA [N (2' MERCAPTOETHYLAMINO)METHYLENE]NORTROPANE TC 99M; RADIOPHARMACEUTICAL AGENT; TRACER; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL ANALYSIS; CHEMICAL REACTION; CHEMICAL STRUCTURE; CONTROLLED STUDY; DRUG DISTRIBUTION; DRUG UPTAKE; ISOTOPE LABELING; NONHUMAN; RAT; REACTION ANALYSIS; SYNTHESIS; TISSUE DISTRIBUTION;

ANIMALS; CHROMATOGRAPHY, LIQUID; DOPAMINE PLASMA MEMBRANE TRANSPORT PROTEINS; MAGNETIC RESONANCE SPECTROSCOPY; MEMBRANE GLYCOPROTEINS; MEMBRANE TRANSPORT PROTEINS; NERVE TISSUE PROTEINS; ORGANOTECHNETIUM COMPOUNDS; RADIOMETRY; RATS; SPECTROMETRY, MASS, ELECTROSPRAY IONIZATION; TROPANES;

EID: 12844268649     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2004.11.036     Document Type: Article

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