Quantitative structure-activity relationship study on some benzodiazepine derivatives as anti-Alzheimer agents

Journal of Molecular Modeling

Volumn 10, Issue 5-6, 2004, Pages 328-334

  Debnath, Bikash ^a   Gayen, Shovanlal ^a   Basu, Anindya ^a   Srikanth, Kolluru ^b   Jha, Tarun ^a  

^a JADAVPUR UNIVERSITY   (India)

^b UNIVERSITY OF MINNESOTA   (United States)

Author keywords

secretase; Alzheimer's disease; Benzodiazepine; ETSA index; QSAR

Indexed keywords

BENZODIAZEPINE DERIVATIVE; BENZODIAZEPINE RECEPTOR; BENZODIAZEPINE RECEPTOR BLOCKING AGENT; FLUORINE DERIVATIVE; GAMMA SECRETASE; GAMMA SECRETASE INHIBITOR;

ALZHEIMER DISEASE; ARTICLE; DRUG ACTIVITY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; ENZYME INHIBITION; PHARMACOPHORE; PRIORITY JOURNAL; QUANTITATIVE STRUCTURE ACTIVITY RELATION; SUBSTITUTION REACTION;

ALZHEIMER DISEASE; AMYLOID PRECURSOR PROTEIN SECRETASES; BENZODIAZEPINES; ENDOPEPTIDASES; MODELS, MOLECULAR; MOLECULAR STRUCTURE; PROTEASE INHIBITORS; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 10944265512     PISSN: 16102940     EISSN: None     Source Type: Journal    
DOI: 10.1007/s00894-004-0199-4     Document Type: Article

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