5-N-Substituted-2-(substituted benzenesulphonyl) glutamines as antitumor agents. Part II: Synthesis, biological activity and QSAR study

Bioorganic and Medicinal Chemistry

Volumn 12, Issue 6, 2004, Pages 1413-1423

  Samanta, Soma ^a,b   Srikanth, K ^a,c   Banerjee, Suchandra ^a   Debnath, Bikash ^a   Gayen, Shovanlal ^a   Jha, Tarun ^a  

^a JADAVPUR UNIVERSITY   (India)

^b UNIVERSITY OF MINNESOTA   (United States)

^c INDIAN INSTITUTE OF CHEMICAL BIOLOGY   (India)

Author keywords

Anticancer activity; Cell count inhibition; Glutamine analogues; QSAR study; Synthesis

Indexed keywords

ANTINEOPLASTIC AGENT; BENZENE DERIVATIVE; GLUTAMIC ACID DERIVATIVE; GLUTAMINE DERIVATIVE; SULFUR DERIVATIVE;

AMINO ACID SUBSTITUTION; ANTINEOPLASTIC ACTIVITY; ARTICLE; BIOSYNTHESIS; CANCER INHIBITION; DRUG ACTIVITY; DRUG DESIGN; DRUG EFFICACY; DRUG SCREENING; DRUG SYNTHESIS; PHYSICAL CHEMISTRY; QUANTITATIVE STRUCTURE ACTIVITY RELATION; STEREOCHEMISTRY; TUMOR CELL;

ANIMALS; ANTINEOPLASTIC AGENTS; CARCINOMA, EHRLICH TUMOR; DRUG SCREENING ASSAYS, ANTITUMOR; FEMALE; GLUTAMINE; HUMANS; MICE; MOLECULAR STRUCTURE; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; TUMOR CELLS, CULTURED;

EID: 1542361437     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2004.01.006     Document Type: Article

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