Influence of hydroxypropyl-β-cyclodextrin complexation on piroxicam release from buccoadhesive tablets

European Journal of Pharmaceutical Sciences

Volumn 21, Issue 2-3, 2004, Pages 251-260

  Jug, Mario ^a   Bećirević Laćan, Mira ^a  

^a UNIVERSITY OF ZAGREB   (Croatia)

Author keywords

Buccal drug delivery; Cyclodextrin complexation; Mucoadhesion; Piroxicam

Indexed keywords

2 HYDROXYPROPYL BETA CYCLODEXTRIN; C 940; CARBOPOL 940; HYDROXYPROPYLMETHYLCELLULOSE; LACTOSE; MAGNESIUM STEARATE; PIROXICAM; POLYMER;

ADHESION; ARTICLE; COMPLEX FORMATION; COMPRESSION; CONTROLLED DRUG RELEASE; DIFFERENTIAL SCANNING CALORIMETRY; DISSOLUTION; DRUG DIFFUSION; DRUG INTERACTION; DRUG SOLUBILITY; DRUG SYNTHESIS; HYDRATION; HYDROPHILICITY; INFRARED SPECTROSCOPY; PRIORITY JOURNAL; SOLID STATE; STOICHIOMETRY; TABLET; WATER TRANSPORT; X RAY DIFFRACTION;

EID: 0742287066     PISSN: 09280987     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejps.2003.10.029     Document Type: Article

References (21)

1. Badawy S.I.F., Ghorab M.M., Adeyeye C.M. Bioavailability of danazol-hydroxypropil-β-cyclodextrin complex by different routes of administration. Int. J. Pharm. 145:1996;137-143.
2. Bottenberg P., Cleymaet R., DeMuyuck C., Remon J.P., Coomans D., Michotte Y., Slop D. Development and testing of bioadhesive, fluoride containing flow-release tablets for oral use. J. Pharm. Pharmacol. 43:1991;457-464.
3. Doliwa A., Santoyo S., Ygartna P. Influence of piroxicam: hydroxypropyl-beta-cyclodextrin complexation on the in vitro permeation and skin retention of piroxicam. Skin Pharmacol. Appl. Skin Physiol. 14:2001;97-107.
4. Higuchi T., Connors K. Phase solubility techniques. Adv. Anal. Chem. Instrum. 7:1965;117-212.
5. Korsmeyer R.W., Guruy R., Doelker E., Buri P., Peppas N.A. Mechanism of solute release from porous polymers. Int. J. Pharm. 15:1983;25-35.
6. Lee V.H.L., Yamamoto A., Kompella M.B. Mucosal penetration enhancers for facilitation of peptide and protein drug absorption. Crit. Dev. Ther. Drug Carrier Syst. 8:1991;91-92.
7. Loftsson T., Brewster M.E. Pharmaceutical applications of cyclodextrins. I. Drug solubilisation and stabilisation. J. Pharm. Sci. 85:1996;1012-1025.
8. McEwen J. Clinical pharmacology of piroxicam-β-cyclodextrin. Clin. Drug Invest. 19:2000;27-31.
9. Park C.R., Munday D.L. Development and evaluation of a biphasic buccal adhesive tablet for nicotine replacement therapy. Int. J. Pharm. 237:2002;215-226.
10. Perez-Marcos B., Ford J.L., Armstrong D.J., Elliott P.N.C., Rostrom C., Hogan J.E. Influence of pH on the release of propranolol hydrochloride from matrices containing hydroxypropyl-methylcellulose K4M and Carbopol 974. J. Pharm. Sci. 85:1996;330-334.
11. Pitha J., Harman S.M., Michel M.E. Hydrophylic cyclodextrin derivatives enable effective oral administration of steroidal hormones. J. Pharm. Sci. 75:1986;165-167.
12. Ponchel G., Tonchard F., Duchene D., Peppas N.A. Bioadhesive analysis of controlled release systems. I. Fracture and inter penetration analysis in poly(acrylic acid) containing system. J. Control. Release. 5:1987;129-141.
13. Rajewski R.A., Stella V.J. Pharmaceutical applications of cyclodextrins 2. In vivo drug delivery. J. Pharm. Sci. 85:1996;1142-1169.
14. Redenti E., Peveri T., Zanol M., Ventura P., Gnappi G., Montenero A. A study on the differentiation between amorphous piroxicam: β cyclodextrin complex and a mixture of the two amorphous components. Int. J. Pharm. 129:1996;289-294.
15. Ritger P.L., Peppas A. A simple equation for description of solute release. II. Fickian and anomalous release from swellable devices. J. Controll. Rel. 5:1987;37-42.
16. Senel S., Capan Y., Sargon M.F., Giray C.B., Hincal A.A. Histological bioadhesion studies on buccal and bioadhesive tablets containing a penetration enhancer sodium glycodeoxycholate. Int. J. Pharm. 170:1998;239-245.
17. Senel S., Hincal A.A. Drug permeation enhancement via buccal route: possibilities and limitations. J. Control. Release. 72:2001;133-144.
18. Singh B., Ahuja N. Development of controlled-release buccoadhesive hydrophilic matrices of diltiazem hydrochloride. Optimisation of bioadhesion, dissolution, and diffusion parameters. Drug Develop. Ind. Pharm. 28:2002;431-442.
19. Sridevi S., Divan P.V.R. Optimized transdermal delivery of ketoprofen using pH and hydroxypropyl-β-cyclodextrin as co-enhancers. Eur. J. Pharm. Biopharm. 54:2002;151-154.
20. Voorspoels J., Remon J., Eechante W., De Sy W. Buccal absorption of testosterone and its esters using a bioadhesive tablet in dogs. Pharm. Res. 13:1996;1228-1232.
21. Vrecer F., Vrbinc M., Meden A. Characterisation of piroxicam crystal modification. Int. J. Pharm. 256:2003;3-15.