Synthesis and structural studies of a novel scaffold for drug discovery: A 4,5-dihydro-3H-spiro[1,5-benzoxazepine-2,4′-piperidine]

Tetrahedron Letters

Volumn 45, Issue 5, 2004, Pages 1051-1054

  Willand, Nicolas ^a   Beghyn, Terence ^a   Nowogrocki, Guy ^b   Gesquiere, Jean Claude ^a   Deprez, Benoit ^a  

^a UNIV LILLE   (France)

^b CNRS   (France)

Author keywords

Benzoxazepine; Piperidine; Privileged structures; Scaffold; X ray

Indexed keywords

4,5 DIHYDRO 3H SPIRO[1,5 BENZOXAZEPINE 2,4' PIPERIDINE]; ACETOPHENONE DERIVATIVE; PIPERIDINE DERIVATIVE; PIPERIDONE DERIVATIVE; UNCLASSIFIED DRUG;

AQUEOUS SOLUTION; ARTICLE; CHEMICAL ANALYSIS; CHEMICAL STRUCTURE; DRUG DESIGN; NUCLEAR MAGNETIC RESONANCE; NUCLEAR OVERHAUSER EFFECT; STRUCTURE ANALYSIS; X RAY DIFFRACTION;

EID: 0347022273     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tetlet.2003.11.079     Document Type: Article

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