3,5-Di-(tert-Butyl)-6-fluoro-cycloSal-d4TMP - A Pronucleotide with a Considerably Improved Masking Group

European Journal of Organic Chemistry

Volumn , Issue 24, 2003, Pages 4786-4791

  Ducho, Christian ^a   Wendicke, Silke ^a   Görbig, Ulf ^a   Balzarini, Jan ^b   Meier, Chris ^a  

^a UNIVERSITY OF HAMBURG   (Germany)

^b REGA INSTITUTE FOR MEDICAL RESEARCH   (Belgium)

Author keywords

Antiviral agents; DNA; Nucleosides

Indexed keywords

3,5 DI(TERT BUTYL) 6 FLUOROCYCLOSALICYL ALCOHOL 2',3' DIDEOXY 2',3' DIDEHYDROTHYMIDINE; ANTI HUMAN IMMUNODEFICIENCY VIRUS AGENT; CHOLINESTERASE; FLUORINE DERIVATIVE; NUCLEOTIDE DERIVATIVE; THYMIDINE KINASE; UNCLASSIFIED DRUG;

ANTIVIRAL ACTIVITY; ARTICLE; DRUG HALF LIFE; DRUG POTENCY; DRUG SELECTIVITY; ENZYME INHIBITION; REACTION ANALYSIS; STRUCTURE ACTIVITY RELATION;

EID: 0346732153     PISSN: 1434193X     EISSN: None     Source Type: Journal    
DOI: 10.1002/ejoc.200300537     Document Type: Article

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