Loperamide (ADL 2-1294), an opioid antihyperalgesic agent with peripheral selectivity

Journal of Pharmacology and Experimental Therapeutics

Volumn 289, Issue 1, 1999, Pages 494-502

  Dehaven Hudkins, D L ^a   Cortes Burgos, L ^a   Cassel, J A ^a   Daubert, J D ^a   Dehaven, R N ^a   Mansson, E ^a   Nagasaka, H ^b,c   Yu, G ^a   Yaksh, T ^b  

^a ADOLOR CORPORATION   (United States)

^b University of California   (United States)

^c SAITAMA MEDICAL UNIVERSITY   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

LOPERAMIDE;

ANALGESIC ACTIVITY; ANIMAL EXPERIMENT; ANTINOCICEPTION; ARTICLE; DRUG EFFECT; DRUG EFFICACY; DRUG MECHANISM; DRUG POTENCY; HYPERALGESIA; MALE; NONHUMAN; PRIORITY JOURNAL; RAT;

ANALGESICS, OPIOID; ANIMALS; ANTIDIARRHEALS; CLONING, MOLECULAR; CRICETINAE; CYCLIC AMP; FORSKOLIN; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); HUMANS; HYPERALGESIA; INFLAMMATION; LOPERAMIDE; MALE; MICE; MICE, INBRED ICR; PAIN MEASUREMENT; PERIPHERAL NERVOUS SYSTEM; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, OPIOID; RECEPTORS, OPIOID, DELTA; RECEPTORS, OPIOID, KAPPA; RECEPTORS, OPIOID, MU;

EID: 0344609779     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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