Synthesis and binding studies of some epibatidine analogues

Bioorganic and Medicinal Chemistry Letters

Volumn 10, Issue 1, 2000, Pages 55-58

  Rádl, Stanislav ^a   Hezký, Petr ^a   Hafner, Wieland ^a   Buděšínský, Miloš ^b   Hejnová, Lucie ^a  

^a Research Institute of Pharmacy and Biochemistry Prague   (Czech Republic)

^b INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY   (Czech Republic)

Author keywords

[No Author keywords available]

Indexed keywords

CHOLINERGIC RECEPTOR; EPIBATIDINE;

ALZHEIMER DISEASE; ARTICLE; BINDING AFFINITY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; ISOMER; LIGAND BINDING; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY;

ANALGESICS, NON-NARCOTIC; ANIMALS; BICYCLO COMPOUNDS, HETEROCYCLIC; BINDING, COMPETITIVE; BRAIN; HEART ATRIA; INHIBITORY CONCENTRATION 50; ISOMERISM; KINETICS; NICOTINIC AGONISTS; PYRIDINES; RADIOLIGAND ASSAY; RATS; RECEPTOR, MUSCARINIC M1; RECEPTOR, MUSCARINIC M2; RECEPTOR, SEROTONIN, 5-HT1B; RECEPTORS, MUSCARINIC; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT1;

EID: 0342948833     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(99)00575-2     Document Type: Article

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