Semi-synthetic glycopeptide antibacterials

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 23, 2003, Pages 4165-4168

  Judice, J Kevin ^a,c   Pace, John L ^a,b  

^a THERAVANCE INC   (United States)

^b Genentech Inc ^*  (United States)

^c GENENTECH INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANTIINFECTIVE AGENT; DALBAVANCIN; GLYCOPEPTIDE; ORITAVANCIN; TELAVANCIN; THRX 689909; UNCLASSIFIED DRUG; VANCOMYCIN;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIBACTERIAL ACTIVITY; ARTICLE; BACTERIAL INFECTION; CLINICAL TRIAL; CONTROLLED CLINICAL TRIAL; CONTROLLED STUDY; DRUG ACTIVITY; DRUG DISTRIBUTION; DRUG EFFICACY; DRUG HALF LIFE; HUMAN; MOUSE; NEPHROTOXICITY; NONHUMAN; PHASE 1 CLINICAL TRIAL; PHASE 2 CLINICAL TRIAL; PHASE 3 CLINICAL TRIAL;

EID: 0242653645     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2003.08.067     Document Type: Article

References (56)

1. Witte W.J. Antimicrob. Chemother. 44:1999;1.
2. Moellering R.C. Jr. Clin. Infect. Dis. 27:1998;S135.
3. Chambers H.F. Clin. Microbiol. Rev. 10:1997;781.
4. Malabarba A., Nicas T., Ciabatti R. Eur. J. Med. Chem. 32:1997;459.
5. Ziglam H.M., Finch R.G. Clin. Microb. Infect. 7:2001;S53.
6. Smith T.L., Pearson M.L., Wilcox K.R., Cruz C., Lancaster M.V., Robinson-Dunn B., Tenover F.C., Zervos M.J., Band J.D., White E., Jarvis W.R. N. Engl. J. Med. 340:1999;493.
7. Hiramatsu K., Aritaka N., Hanaki H., Kawasaki Hosoda Y., Hori S., Fukuchi Y., Kobayashi I. Lancet. 350:1997;1670.
8. MMWR. 51:2002;565.
9. MMWR. 51:2002;902.
10. JAMA. 288:2002;2116.
11. Chang S., Sievert D.M., Hageman J.C., Boulton M.L., Tenover F.C., Downes F.P., Shah S., Rudrik J.T., Pupp G.R., Brown W.J., Cardo D., Fridkin S.K. N. Engl. J. Med. 348:2003;1342.
12. Leclerq R., Derlot E., Duval J., Courvalin P. N. Engl. J. Med. 319:1988;157.
13. Uttley A.H.C., Collins C.H., Naidoo J., George R.C. Lancet. 1988:1988;1. 57.
14. Bozdogan, B.; Chaitram, J.; Appelbaum, P. C.; Whitener, C.; Browne, F. A.; Tenover, F. C. Abstracts of Papers, 103rd Amer. Soc. for Microbiology Annual Meet., May 18-22, 2003; Amer. Soc. for Microbiology: Washington, DC, 2003; A-075.
15. Nagarajan R. J. Antibiot. 46:1993;1181.
16. Nagarajan R. Nagarajan R. Glycopeptide Antibiotics. 1994;195 Marcel Dekker, New York.
17. Nicas T.I., Allen N.E. Nagarajan R. Glycopeptide Antibiotics. 1994;219 Marcel Dekker, New York.
18. Nicas T.I., Mullen D.L., Flokowitsch J.E., Preston D.A., Snyder N.J., Zweifel M.J., Wilkie S.C., Rodriguez M.J., Thompson R.C., Cooper R.D. Antimicrob. Agents Chemother. 40:1996;2194.
19. Ge M., Chen Z., Onishi H.R., Kohler J., Silver L.L., Kerns R., Fukuzawa S., Thompson C., Kahne D. Science. 284:1999;507.
20. Chen L., Walker D., Sun B., Hu Y., Walker S., Kahne D. Proc. Natl. Acad. Sci. U.S.A. 100:2003;5658.
21. Leadbetter, M. R.; Linsell, M.; Fatheree, P.; Trapp, S.; Lam, B.; Nodwell, M.; Shaw, J.; Pace, J.; Judice, K. Abstracts of Papers, 42nd ICAAC, San Diego, CA, Sept. 27-30, 2002; Am. Soc. Microbiol.: Washington, DC, 2002; F-367.
22. Blizzard T.A., Kim R.M., Morgan J.D. II, Chang J., Kohler J., Kilburn R., Chapman K., Hammond M.L. Biorg. Med. Chem. Lett. 12:2002;849.
23. Yoshida O., Yasukata T., Sumino Y., Munekage T., Narukawa Y., Nishitani Y. Bioorg. Med. Chem. Lett. 12:2002;3027.
24. Allen N.E., Nicas T.I. FEMS Microbiol. Rev. 26:2002;511.
25. Rodriguez M.J., Snyder N.J., Zweifel M.J., Wilkie S.C., Stack D.R., Cooper R.D.G., Nicas T.I., Mullen D.L., Butler T.F., Thompson R.C. J. Antibiotics. 51:1998;560.
26. Nagarajan R., Schabel A.A., Occolowitz J.L., Counter F.T., Ott J.L., Felty-Duckworth A.M. J. Antibiotics. 42:1989;63.
27. Pavlov A.Y., Lazhko E.I., Preobrazhenskaya M.N. J. Antibiotics. 50:1997;509.
28. Debabov, D., Pace, J.; Kaniga, K.; Nodwell, M.; Farrington, L.; Campbell, B.; Karr, D.; Leadbetter, M.: Linsell, M.; Wu, T.; Krause, K.; Johnston, D.; Lane, C.; Quast, K.; Bazzini, B.; Phi, B.; Schmidt, D.; White, L.; Higgins, D.; Christensen, B.; Judice, K. Abstracts of Papers, 42nd ICAAC, San Diego, CA, Sept. 27-30, 2002. Am. Soc. Microbiol.: Washington, DC, 2002; F-364.
29. Pace, J. L. Abstracts of Papers, 42nd ICAAC, San Diego, CA, Sept. 27-30, 2002; Am. Soc. Microbiol.: Washington, DC, 2002; p 614.
30. Bugg T.D.H., Wright G.D., Dutka-Malen S.S., Arthur M., Courvalin P., Walsh C.T. Biochemistry. 30:1991;10408.
31. Nieto M., Perkins R., Reynolds P.E. Biochem. J. 126:1972;139.
32. Gerhard U., Mackay J.P., Maplestone R.A., Williams D.H. J. Am. Chem. Soc. 115:1993;232.
33. Sharman G.J., Williams D.H. Chem. Commun. 7:1997;723.
34. Rao J., Lahiri J., Issacs L., Weis R.M., Whitesides G.M. Science. 280:1998;708.
35. Beauregard D.A., Williams D.H., Gwynn M.N., Knowles D.J. Antimicrob. Agents Chemother. 39:1995;781.
36. Goldstein B.P., Rosina R., Parenti F. Nagarajan R. Glycopeptide Antibiotics. 1994;273 Marcel Dekker, New York.
37. Allen N.E., leTourneau D.L., Hobbs J.N. Jr., Thompson R.C. Antimicrob. Agents Chemother. 46:2002;2344.
38. Pace, J.; Quast, K.; Chen, Q.; Linsell, M.; Krause, K.; Farrington, L.; Nodwell, M.; Leadbetter, M.; Schmidt, D.; Mabery, E.; Soriano, E.; Fatheree, P. ; Bazzini, B.; Bao, J.; Gao, D.; Higgins, D.; Griffin, J.; Karr, D.; Christensen, B.; Judice, K. Abstracts of Papers, 12th ECCMID, Milan, Italy, April 24-27, 2002; ESCMID: Basel, Switzerland, 2002; O134.
39. Pace, J.; Judice, K.; Hegde, S.; Leadbetter, M.; Linsell, M.; Kaniga, K. ; Reyes, N.; Farrington, L.; Debabov, D.; Nodwell, M.; Christensen, B. Abstracts of Papers, 10th International Symposium Staphylococci and Staphylococcal Infection, Tsukuba, Japan, Oct. 16-19, 2002; Japanese Symposium on Staphylococci and Staphylococcal Infections: Tokyo, Japan, 2002; 265-01.
40. King, A.; Phillips, I.; Farrington, L.; Pace, J.; Kaniga, K. Abstracts of Papers, 13th ECCMID, Glasgow, Scotland, May 10-13, 2003; ESCMID: Basel, Switzerland, 2003; p 799.
41. Jones R.N., Barrett M.S., Erwin M.E. Antimicrob. Agents Chemother. 41:1996;488.
42. Karlowsky, J. A.; Loutit, J.; Porter, S. B.; Blosser-Middleton, R. S.; Jones, M. E.; Thornsberry, C.; Sahm, D. Abstract of Papers, 13th ECCMID, Glasgow, Scotland, May 10-13, 2003. ESCMID: Basel, Switzerland, 2003; p 801.
43. Reynolds, P. Abstracts of Papers, 37th ICAAC, Toronto, CN, Sept. 28-Oct. 1, 1997; Am. Soc. Microbiol.: Washington, DC, 1997; C-165.
44. Weigel, L. M., McDougal, L. K.; Clark, N.; Killgore, G.; Tenover, F. C.; Appelbaum, P. C.; Bozdogan, B. Abstracts of Papers, 103rd Am. Soc. for Microbiology Annual Meet., May 18-22, 2003; Am. Soc. for Microbiology: Washington, DC, 2003; A-111.
45. Jones, R. N.; Biedenbach, D. J.; Johnson, D. M.; Pfaller, M. A. Abstracts of Papers, 42nd ICAAC, San Diego, CA, Sept. 27-30, 2002; Am. Soc. Microbiol.: Washington, DC, 2002; p 2276.
46. Patel R., Rouse M.S., Piper K.E., Cockerill F.R., Steckelberg J.M. Diagn. Microbiol. Infect. Dis. 30:1998;89.
47. Coyle E.A., Rybak M.J. Antimicrob. Agents Chemother. 45:2001;706.
48. Garcia-Garrote F., Cercenado E., Alcala L., Bouza E. Antimicrob. Agents Chemother. 42:1998;2452.
49. Zeckel M.L.D., Preston D.A., Allen B.S. Antimicrob. Agents Chemother. 44:2000;1370.
50. Gomez, M.; Hackbarth, C. J.; Lopez, S.; Trias, J.; White, R. 101st Am. Soc. Microbiol. Gen. Meet., Orlando, FL, May 20-24, 2001; Am. Soc. Microbiol.: Washington, DC, 2001; A-4.
51. Barriere, S.; Shaw, J. P.; Seroogy, J.; Kaniga, K.; Pace, J.; Judice, K. ; Mant, T. Abstracts of Papers, 13th ECCMID, Glasgow, Scotland, May 10-13, 2003; ESCMID: Basel, Switzerland, 2003; P1214.
52. Barriere, S.; Genter, F.; Spencer, E.; Kitt, M.; Hoelscher, D.; Morganroth, J. Abstracts of Papers, 13th ECCMID, Glasgow, Scotland, May 10-13, 2003; ESCMID: Basel, Switzerland, 2003; O144.
53. Leighton, A., White, R.; Chaudhari, U.; Van Saders, C.; Baylor, M.; Perry, M.; Henkel, T.; Kelly, E.; Campbell, K. C. M. Abstracts of Papers, 41st ICAAC, Chicago, IL Dec. 7-11, 2001; Am. Soc. Microbiol.: Washington, DC, 2001; 2192.
54. Dowell, J. A.; Gottlieb, A. B.; Van Saders, C.; Dorr, M. B.; Leighton, A.; Cavaleri, M.; Guanci, M.; Colombo, L. 2002. Abstracts of Papers, 42nd ICAAC, San Diego, CA, Sept. 27-30, 2002; Am. Soc. Microbiol.: Washington, DC, 2001; p 1386.
55. White, R. J.; Brown, G. L.; Cavellero, M.; Romano, G. Abstracts of Papers, 40th ICAAC, Toronto, Canada, Sept. 17-20, 2000; Am. Soc. Microbiol.: Washington, DC, 2000; p 2196.
56. Candiani G., Abbondi M., Borogonovi M., Romano G., Parenti F.J. Antimicrob. Chemother. 44:1999;179.