-
1
-
-
0028222149
-
-
(a) Vacca, J. P.; Dorsey, B. D.; Schleif, W. A.; Levin, R. B.; McDaniel, S. L.; Darke, P. L.; Zugay, J.; Quintero, J. C.; Blanhy, O. M.; Roth, E.; Sardana, V. V.; Schlabach, A. J.; Graham, P. I.; Condra, J. H.; Gotlib, L.; Holloway, M. K.; Lin, J.; Chen, I.-W.; Vastag, K.; Ostovic, D.; Anderson, P. S. ; Emini, E. A.; Huff, J. R. Proc. Natl. Sci. U.S.A. 1994, 91, 4096-4100.
-
(1994)
Proc. Natl. Sci. U.S.A.
, vol.91
, pp. 4096-4100
-
-
Vacca, J.P.1
Dorsey, B.D.2
Schleif, W.A.3
Levin, R.B.4
McDaniel, S.L.5
Darke, P.L.6
Zugay, J.7
Quintero, J.C.8
Blanhy, O.M.9
Roth, E.10
Sardana, V.V.11
Schlabach, A.J.12
Graham, P.I.13
Condra, J.H.14
Gotlib, L.15
Holloway, M.K.16
Lin, J.17
Chen, I.-W.18
Vastag, K.19
Ostovic, D.20
Anderson, P.S.21
Emini, E.A.22
Huff, J.R.23
more..
-
2
-
-
0141449192
-
-
(b) Ravina, E.; Casariego, I.; Masguer, C. f.; Fontenla, J. A.; Montenegro, G. Y.; Rivas, M. E.; Loza, M. I.; Enguix, M. J.; Villazon, M.; Cadavid, M. I.; Demontis, G. C. J. Med. Chem. 2000, 43, 4673-4693.
-
(2000)
Med. Chem.
, vol.43
, pp. 4673-4693
-
-
Ravina, E.1
Casariego, I.2
Masguer, C.F.3
Fontenla, J.A.4
Montenegro, G.Y.5
Rivas, M.E.6
Loza, M.I.7
Enguix, M.J.8
Villazon, M.9
Cadavid, M.I.10
Demontis, G.C.J.11
-
3
-
-
0032576635
-
-
(c) Rival, V.; Hoffmann, R.; Didier, B.; Rybaltchenko, V.; Bouruignon, J.-J.; Wermuth, C. G.; J. Med. Chem. 1998, 41, 311-317.
-
(1998)
J. Med. Chem.
, vol.41
, pp. 311-317
-
-
Rival, V.1
Hoffmann, R.2
Didier, B.3
Rybaltchenko, V.4
Bouruignon, J.-J.5
Wermuth, C.G.6
-
4
-
-
0027291048
-
-
(d) Naylor, A.; Judd, D. B.; Lloyd, J. E.; Scopes, D. I.; Hayes, A. G.; Birch, P. J. J. Med. Chem. 1993, 36, 2075-2083.
-
(1993)
Med. Chem.
, vol.36
, pp. 2075-2083
-
-
Naylor, A.1
Judd, D.B.2
Lloyd, J.E.3
Scopes, D.I.4
Hayes, A.G.5
Birch, P.J.J.6
-
5
-
-
0025739032
-
-
(e) Karton, Y.; Bradbury, B. J.; Baumgold, J.; Paek, R.; Jacobson, K. A. J. Med. Chem. 1991, 34, 2133-2145.
-
(1991)
J. Med. Chem.
, vol.34
, pp. 2133-2145
-
-
Karton, Y.1
Bradbury, B.J.2
Baumgold, J.3
Paek, R.4
Jacobson, K.A.5
-
6
-
-
0141672158
-
-
(f) McMillian, K.; Adler, M.; Auld, D. S.; Baldwin, J. J.; Blasko, E.; Browne, L. J.; Chelsky, D.; Davey, D.; Dolle, R. E.; Eagen, K. A.; Erickson, S. ; Feldman, R. I.; Glaser, C. B.; Mallari, C.; Morrissey, M. M.; Ohlmeyer, M. H. J.; Pan, G.; Parkinson, J. F.; Phillips, G. B.; Polokoff, M. A.; Sigal, N. H.; Vergona, R.; Whitlow, M.; Young, T. A.; Devlin, J. J. Proc. Natl. Acad. Sci. U.S.A. 2000, 6, 3943-3957.
-
(2000)
Proc. Natl. Acad. Sci. U.S.A.
, vol.6
, pp. 3943-3957
-
-
McMillian, K.1
Adler, M.2
Auld, D.S.3
Baldwin, J.J.4
Blasko, E.5
Browne, L.J.6
Chelsky, D.7
Davey, D.8
Dolle, R.E.9
Eagen, K.A.10
Erickson, S.11
Feldman, R.I.12
Glaser, C.B.13
Mallari, C.14
Morrissey, M.M.15
Ohlmeyer, M.H.J.16
Pan, G.17
Parkinson, J.F.18
Phillips, G.B.19
Polokoff, M.A.20
Sigal, N.H.21
Vergona, R.22
Whitlow, M.23
Young, T.A.24
Devlin, J.J.25
more..
-
7
-
-
0034268096
-
-
(g) Cheng, Y.; Lu, Z.; Chapman, K. T.; Tata, J. R. J. Comb. Chem. 2000, 2, 445-446.
-
(2000)
J. Comb. Chem.
, vol.2
, pp. 445-446
-
-
Cheng, Y.1
Lu, Z.2
Chapman, K.T.3
Tata, J.R.4
-
8
-
-
0024239320
-
-
Evans, B. E.; Rittle, K. E.; Bock, M. G.; DiPardo, R. M.; Freidinger, R. M.; Whitter, W. L.; Lundell, G. F.; Veber, D. F.; Anderson, P. S.; Chang, R. S. L.; Lotti, V. J.; Cerino, D. J.; Chen, T. B.; Kling, P. J.; Kunkel, K. A.; Springer, J. P.; Hirshfield, J. J. Med. Chem., 1988, 31, 2235-2246.
-
(1988)
J. Med. Chem.
, vol.31
, pp. 2235-2246
-
-
Evans, B.E.1
Rittle, K.E.2
Bock, M.G.3
DiPardo, R.M.4
Freidinger, R.M.5
Whitter, W.L.6
Lundell, G.F.7
Veber, D.F.8
Anderson, P.S.9
Chang, R.S.L.10
Lotti, V.J.11
Cerino, D.J.12
Chen, T.B.13
Kling, P.J.14
Kunkel, K.A.15
Springer, J.P.16
Hirshfield, J.17
-
14
-
-
0030857041
-
-
(f) Cuny, G. D.; Cao, J.; Hanske, J. R. Tetrahedron Lett. 1997, 38, 5237-5240.
-
(1997)
Tetrahedron Lett.
, vol.38
, pp. 5237-5240
-
-
Cuny, G.D.1
Cao, J.2
Hanske, J.R.3
-
15
-
-
0032474714
-
-
(g) Hoemann, M. Z.; Melikan-Badalian, M.; Kumaravel, G.; Hauske, J. Tetrahedron Lett. 1998, 39, 4749-4752.
-
(1998)
Tetrahedron Lett.
, vol.39
, pp. 4749-4752
-
-
Hoemann, M.Z.1
Melikan-Badalian, M.2
Kumaravel, G.3
Hauske, J.4
-
17
-
-
0030921936
-
-
(a) Brown, A. R.; Rees, D. C.; Rankovic, Z.; Morphy, J. R. J. Am. Chem. Soc. 1997, 119, 3288-3295.
-
(1997)
J. Am. Chem. Soc.
, vol.119
, pp. 3288-3295
-
-
Brown, A.R.1
Rees, D.C.2
Rankovic, Z.3
Morphy, J.R.4
-
18
-
-
0035511874
-
-
(b) Barn, D.; Caulfield, W.; Cowley, P.; Dickens, R.; Iwema Bakker, W.; McGuire, R.; Morphy, J. R.; Rankovic, Z.; Thorn, M. J. Comb. Chem. 2001, 3, 534-541.
-
(2001)
J. Comb. Chem.
, vol.3
, pp. 534-541
-
-
Barn, D.1
Caulfield, W.2
Cowley, P.3
Dickens, R.4
Iwema Bakker, W.5
McGuire, R.6
Morphy, J.R.7
Rankovic, Z.8
Thorn, M.9
-
19
-
-
0034709661
-
-
(a) Schlienger, N.; Bryce, M. R.; Hansen, T. K. Tetrahedron Lett. 2000, 41, 5147-5150.
-
(2000)
Tetrahedron Lett.
, vol.41
, pp. 5147-5150
-
-
Schlienger, N.1
Bryce, M.R.2
Hansen, T.K.3
-
20
-
-
0034670582
-
-
(b) Schlienger, N.; Bryce, M. R.; Hansen, T. K. Tetrahedron 2000, 56, 10023-10030.
-
(2000)
Tetrahedron
, vol.56
, pp. 10023-10030
-
-
Schlienger, N.1
Bryce, M.R.2
Hansen, T.K.3
-
21
-
-
0001252095
-
-
Lane, C. L. Chem. Rev. 1976, 76, 6 (6), 773-799
-
(1976)
Chem. Rev.
, vol.6
, Issue.6
, pp. 773-799
-
-
Lane, C.L.1
-
22
-
-
0001242088
-
-
Salvino, J. M.; Kumar, N. V.; Orton, E.; Airey, J.; Kiesow, T.; Crawford, K.; Mathew, R.; Krolikowski, P.; Drew, M.; Engers, D.; Krolinkowski, D.; Herpin, T.; Gardyan, M.; McGeehan, G.; Labaudiniere, R. J. Comb. Chem. 2000, 2, 691-697.
-
(2000)
J. Comb. Chem.
, vol.2
, pp. 691-697
-
-
Salvino, J.M.1
Kumar, N.V.2
Orton, E.3
Airey, J.4
Kiesow, T.5
Crawford, K.6
Mathew, R.7
Krolikowski, P.8
Drew, M.9
Engers, D.10
Krolinkowski, D.11
Herpin, T.12
Gardyan, M.13
McGeehan, G.14
Labaudiniere, R.15
-
24
-
-
0033525195
-
-
(a) Hall, D. G.; Laplante, C.; Manku, S.; Nagendran, J. J. Org. Chem. 1999, 64, 698-699.
-
(1999)
J. Org. Chem.
, vol.64
, pp. 698-699
-
-
Hall, D.G.1
Laplante, C.2
Manku, S.3
Nagendran, J.4
-
25
-
-
0001758406
-
-
(b) Nefzi, A.; Ostresh, J. M.; Giulianotti, M.; Houghten, R. A. J. Comb. Chem. 1999, 1, 195-198.
-
(1999)
J. Comb. Chem.
, vol.1
, pp. 195-198
-
-
Nefzi, A.1
Ostresh, J.M.2
Giulianotti, M.3
Houghten, R.A.4
-
26
-
-
0035830582
-
-
(c) Manku, S.; Laplante, C.; Kopac, D.; Chan, T.; Hall, D. G. J. Org. Chem. 2001, 66, 874-885.
-
(2001)
J. Org. Chem.
, vol.66
, pp. 874-885
-
-
Manku, S.1
Laplante, C.2
Kopac, D.3
Chan, T.4
Hall, D.G.5
-
27
-
-
0141449191
-
-
Argonaut Technologies, Foster City, CA 94404
-
Argonaut Technologies, Foster City, CA 94404
-
-
-
-
28
-
-
0034658164
-
-
Gong, Y.; Becker, M.; Choi-Sledeski, Y. M.; Davis, R. S.; Salvino, J. M. ; Chu, V.; Brown, K. D.; Pauls, H. W. Bioorg. Med. Chem. Lett. 2000, 10, 1033-1036.
-
(2000)
Bioorg. Med. Chem. Lett.
, vol.10
, pp. 1033-1036
-
-
Gong, Y.1
Becker, M.2
Choi-Sledeski, Y.M.3
Davis, R.S.4
Salvino, J.M.5
Chu, V.6
Brown, K.D.7
Pauls, H.W.8
-
29
-
-
0141560713
-
-
note
-
Reaction of polymeric TFP-4-acetylamino-benzenesulfonic acid ester (7b) with 2-methylbenzylamine overnight gave equivalent loading results compared to reaction after 3 h.
-
-
-
|