Solid-phase synthesis of substituted 3-aminothiophenes and 2-methylene-2,3-dihydrothiazoles

Tetrahedron Letters

Volumn 37, Issue 34, 1996, Pages 6213-6216

  Zaragoza, Florencio ^a  

^a NOVO NORDISK A S   (Denmark)

Author keywords

[No Author keywords available]

Indexed keywords

ACETAMIDE DERIVATIVE; THIAZOLE DERIVATIVE; THIOPHENE DERIVATIVE;

ARTICLE; CHEMICAL REACTION; DRUG DETERMINATION; DRUG STRUCTURE; DRUG SYNTHESIS; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY;

EID: 0030593632     PISSN: 00404039     EISSN: None     Source Type: Journal    
DOI: 10.1016/0040-4039(96)01326-3     Document Type: Article

References (14)

1. 1. Zaragoza, F.; Petersen, S. V. Tetrahedron 1996, 52, 5999-6002; Zaragoza, F. Tetrahedron Lett. 1995, 36, 8677-8678.
2. 1. Zaragoza, F.; Petersen, S. V. Tetrahedron 1996, 52, 5999-6002; Zaragoza, F. Tetrahedron Lett. 1995, 36, 8677-8678.
3. 2. Laliberté, R.; Médawar, G. Can. J. Chem. 1970, 48, 2709-2717; Laliberté, R.; Warwick, H.; Médawar, G. Can. J. Chem. 1968, 46, 3643-3648.
4. 2. Laliberté, R.; Médawar, G. Can. J. Chem. 1970, 48, 2709-2717; Laliberté, R.; Warwick, H.; Médawar, G. Can. J. Chem. 1968, 46, 3643-3648.
5. 3. Thompson, L. A.; Ellman, J. A. Chem. Rev. 1996, 96, 555-600; Terrett, N. K.; Gardner, M.; Gordon, D. W.; Kobylecki, R. J.; Steele, J. Tetrahedron 1995, 51, 8135-8173.
6. 3. Thompson, L. A.; Ellman, J. A. Chem. Rev. 1996, 96, 555-600; Terrett, N. K.; Gardner, M.; Gordon, D. W.; Kobylecki, R. J.; Steele, J. Tetrahedron 1995, 51, 8135-8173.
7. 4. Other relevant references: Mohareb, R. M.; Sherif, S. M. Arch. Pharm. (Weinheim) 1991, 324, 469-471; Mohareb, R. M.; Sherif, S. M.; Abdel-Aal, F. A. M.; Sayed, N. I. A. Liebigs Ann. Chem. 1990, 1143-1146; Gewald, K.; Hain, U.; Schmidt, M. J. Prakt. Chem. 1986, 328, 459-464; Chiba, T.; Sato, H.; Kato, T. Chem. Pharm. Bull. 1982, 30, 3548-3554; Augustin, M.; Dölling, W. J. Prakt. Chem. 1982, 324, 322-328; Augustin, M.; Rudorf, W.-D.; Schmidt, U. Tetrahedron 1976, 32, 3055-3061.
8. 4. Other relevant references: Mohareb, R. M.; Sherif, S. M. Arch. Pharm. (Weinheim) 1991, 324, 469-471; Mohareb, R. M.; Sherif, S. M.; Abdel-Aal, F. A. M.; Sayed, N. I. A. Liebigs Ann. Chem. 1990, 1143-1146; Gewald, K.; Hain, U.; Schmidt, M. J. Prakt. Chem. 1986, 328, 459-464; Chiba, T.; Sato, H.; Kato, T. Chem. Pharm. Bull. 1982, 30, 3548-3554; Augustin, M.; Dölling, W. J. Prakt. Chem. 1982, 324, 322-328; Augustin, M.; Rudorf, W.-D.; Schmidt, U. Tetrahedron 1976, 32, 3055-3061.
9. 4. Other relevant references: Mohareb, R. M.; Sherif, S. M. Arch. Pharm. (Weinheim) 1991, 324, 469-471; Mohareb, R. M.; Sherif, S. M.; Abdel-Aal, F. A. M.; Sayed, N. I. A. Liebigs Ann. Chem. 1990, 1143-1146; Gewald, K.; Hain, U.; Schmidt, M. J. Prakt. Chem. 1986, 328, 459-464; Chiba, T.; Sato, H.; Kato, T. Chem. Pharm. Bull. 1982, 30, 3548-3554; Augustin, M.; Dölling, W. J. Prakt. Chem. 1982, 324, 322-328; Augustin, M.; Rudorf, W.-D.; Schmidt, U. Tetrahedron 1976, 32, 3055-3061.
10. 4. Other relevant references: Mohareb, R. M.; Sherif, S. M. Arch. Pharm. (Weinheim) 1991, 324, 469-471; Mohareb, R. M.; Sherif, S. M.; Abdel-Aal, F. A. M.; Sayed, N. I. A. Liebigs Ann. Chem. 1990, 1143-1146; Gewald, K.; Hain, U.; Schmidt, M. J. Prakt. Chem. 1986, 328, 459-464; Chiba, T.; Sato, H.; Kato, T. Chem. Pharm. Bull. 1982, 30, 3548-3554; Augustin, M.; Dölling, W. J. Prakt. Chem. 1982, 324, 322-328; Augustin, M.; Rudorf, W.-D.; Schmidt, U. Tetrahedron 1976, 32, 3055-3061.
11. 4. Other relevant references: Mohareb, R. M.; Sherif, S. M. Arch. Pharm. (Weinheim) 1991, 324, 469-471; Mohareb, R. M.; Sherif, S. M.; Abdel-Aal, F. A. M.; Sayed, N. I. A. Liebigs Ann. Chem. 1990, 1143-1146; Gewald, K.; Hain, U.; Schmidt, M. J. Prakt. Chem. 1986, 328, 459-464; Chiba, T.; Sato, H.; Kato, T. Chem. Pharm. Bull. 1982, 30, 3548-3554; Augustin, M.; Dölling, W. J. Prakt. Chem. 1982, 324, 322-328; Augustin, M.; Rudorf, W.-D.; Schmidt, U. Tetrahedron 1976, 32, 3055-3061.
12. 4. Other relevant references: Mohareb, R. M.; Sherif, S. M. Arch. Pharm. (Weinheim) 1991, 324, 469-471; Mohareb, R. M.; Sherif, S. M.; Abdel-Aal, F. A. M.; Sayed, N. I. A. Liebigs Ann. Chem. 1990, 1143-1146; Gewald, K.; Hain, U.; Schmidt, M. J. Prakt. Chem. 1986, 328, 459-464; Chiba, T.; Sato, H.; Kato, T. Chem. Pharm. Bull. 1982, 30, 3548-3554; Augustin, M.; Dölling, W. J. Prakt. Chem. 1982, 324, 322-328; Augustin, M.; Rudorf, W.-D.; Schmidt, U. Tetrahedron 1976, 32, 3055-3061.
13. 13C NMR, MS and IR spectral data.
14. 2 was observed.