Phosphinic acid-based MMP-13 inhibitors that spare MMP-1 and MMP-3

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 14, 2003, Pages 2331-2336

  Reiter, Lawrence A ^a   Mitchell, Peter G ^a   Martinelli, Gary J ^a   Lopresti Morrow, Lori L ^a   Yocum, Sue A ^a   Eskra, James D ^a  

^a PFIZER INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BENZYL DERIVATIVE; COLLAGENASE 3; INTERSTITIAL COLLAGENASE; MATRIX METALLOPROTEINASE INHIBITOR; PHOSPHINIC ACID DERIVATIVE; STROMELYSIN;

ANALYTICAL PARAMETERS; ARTICLE; CHEMICAL PARAMETERS; DRUG POTENCY; DRUG SELECTIVITY; DRUG SYNTHESIS; ENZYME INHIBITION; IC 50; MOLECULAR MECHANICS;

EID: 0038680537     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(03)00413-X     Document Type: Article

References (37)

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