메뉴 건너뛰기




Volumn 56, Issue 1, 2003, Pages 101-110

Potential of carrageenans to protect drugs from polymorphic transformation

Author keywords

Carrageenan; Dehydration; Excipient; FT Raman spectroscopy; Indomethacin; Polymorphic transition; Recrystallisation; Tableting; Theophylline; Three dimensional modelling

Indexed keywords

CALCIUM PHOSPHATE DIBASIC; CARRAGEENAN; HYDROXYPROPYLMETHYLCELLULOSE; INDOMETACIN; MICROCRYSTALLINE CELLULOSE; THEOPHYLLINE;

EID: 0038015537     PISSN: 09396411     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0939-6411(03)00037-7     Document Type: Article
Times cited : (53)

References (41)
  • 1
    • 0026086152 scopus 로고
    • Review on crystal polymorphism of substances in the European Pharmacopeia
    • Borka L. Review on crystal polymorphism of substances in the European Pharmacopeia. Pharm. Acta Helv. 66:(1):1991;16-22.
    • (1991) Pharm. Acta Helv. , vol.66 , Issue.1 , pp. 16-22
    • Borka, L.1
  • 2
    • 0002435409 scopus 로고    scopus 로고
    • Effects of pharmaceutical processing on drug polymorphs and solvates
    • H.G. Brittain. New York, Basel: Marcel Dekker Inc
    • Brittain H.G., Fiese E.F. Effects of pharmaceutical processing on drug polymorphs and solvates. Brittain H.G. Polymorphism in Pharmaceutical Solids. 1999;348-361 Marcel Dekker Inc, New York, Basel.
    • (1999) Polymorphism in Pharmaceutical Solids , pp. 348-361
    • Brittain, H.G.1    Fiese, E.F.2
  • 3
    • 0017599379 scopus 로고
    • Polymorphism of phenylbutazone: Properties and compressional behavior of crystal
    • Ibrahim H.G., Pisano F., Bruno A. Polymorphism of phenylbutazone: properties and compressional behavior of crystal. J. Pharm. Sci. 66:(5):1977;669-673.
    • (1977) J. Pharm. Sci. , vol.66 , Issue.5 , pp. 669-673
    • Ibrahim, H.G.1    Pisano, F.2    Bruno, A.3
  • 4
    • 0020333255 scopus 로고
    • Zur Zeitabhängigkeit der Modifikationsumwandlung des Sulfanilamids bei der Tablettenkompression
    • Kala H., Traue J., Haack U., Moldenhauer H., Kedvessy G., Selmeczi B. Zur Zeitabhängigkeit der Modifikationsumwandlung des Sulfanilamids bei der Tablettenkompression. Pharmazie. 37:(9):1982;674-675.
    • (1982) Pharmazie , vol.37 , Issue.9 , pp. 674-675
    • Kala, H.1    Traue, J.2    Haack, U.3    Moldenhauer, H.4    Kedvessy, G.5    Selmeczi, B.6
  • 5
    • 0021797481 scopus 로고
    • Polymorphic transformation of some drugs under compression
    • Chan H.K., Doelker E. Polymorphic transformation of some drugs under compression. Drug Dev. Ind. Pharm. 11:(2/3):1985;315-332.
    • (1985) Drug Dev. Ind. Pharm. , vol.11 , Issue.2-3 , pp. 315-332
    • Chan, H.K.1    Doelker, E.2
  • 6
    • 0001647274 scopus 로고
    • Polymorphism: Pharmaceutical aspects
    • J. Swarbrick, & J.C. Boylan. New York, Basel, Hong-Kong: Marcel-Decker Inc
    • Otsuka M., Matsuda Y. Polymorphism: pharmaceutical aspects. Swarbrick J., Boylan J.C. Encyclopedia of Pharmaceutical Technology. 1988;305-326 Marcel-Decker Inc, New York, Basel, Hong-Kong.
    • (1988) Encyclopedia of Pharmaceutical Technology , pp. 305-326
    • Otsuka, M.1    Matsuda, Y.2
  • 7
    • 0026759756 scopus 로고
    • Effect of compressional forces on piroxicam polymorphs
    • Ghan G.A., Lalla J.K. Effect of compressional forces on piroxicam polymorphs. J. Pharm. Pharmacol. 44:1992;678-681.
    • (1992) J. Pharm. Pharmacol. , vol.44 , pp. 678-681
    • Ghan, G.A.1    Lalla, J.K.2
  • 8
    • 0027194157 scopus 로고
    • Effects of grinding and compression on crystal structure of anhydrous caffeine
    • Pirttimäki J., Laine E., Ketolainen J., Paronen P. Effects of grinding and compression on crystal structure of anhydrous caffeine. Int. J. Pharm. 95:1993;93-99.
    • (1993) Int. J. Pharm. , vol.95 , pp. 93-99
    • Pirttimäki, J.1    Laine, E.2    Ketolainen, J.3    Paronen, P.4
  • 9
    • 0028300988 scopus 로고
    • Relation between polymorphic transformation pathway during grinding and the physicochemical properties of bulk powders for pharmaceutical preparations
    • Otsuka M., Otsuka K., Kaneniwa N. Relation between polymorphic transformation pathway during grinding and the physicochemical properties of bulk powders for pharmaceutical preparations. Drug Dev. Ind. Pharm. 20:(9):1994;1649-1660.
    • (1994) Drug Dev. Ind. Pharm. , vol.20 , Issue.9 , pp. 1649-1660
    • Otsuka, M.1    Otsuka, K.2    Kaneniwa, N.3
  • 10
    • 0038370669 scopus 로고    scopus 로고
    • Phase purity and impact of polymorphism on the material properties of caffeine
    • Hellemann M., Griesser U.J., Abberger T., Schlocker W., Burger A. Phase purity and impact of polymorphism on the material properties of caffeine. PharmSci. 2:(4):2000;3091.
    • (2000) PharmSci. , vol.2 , Issue.4 , pp. 3091
    • Hellemann, M.1    Griesser, U.J.2    Abberger, T.3    Schlocker, W.4    Burger, A.5
  • 11
    • 1142303337 scopus 로고    scopus 로고
    • What is the true solubility advantage for amorphous pharmaceuticals?
    • Hancock B.C., Parks M. What is the true solubility advantage for amorphous pharmaceuticals? Pharm. Res. 17:(4):2000;397-404.
    • (2000) Pharm. Res. , vol.17 , Issue.4 , pp. 397-404
    • Hancock, B.C.1    Parks, M.2
  • 12
    • 0002611989 scopus 로고
    • Molekulargalenik als Grundlage moderner Arzneiformung
    • Hüttenrauch R. Molekulargalenik als Grundlage moderner Arzneiformung. Acta. Pharm. Technol. 6:1978;55-127.
    • (1978) Acta. Pharm. Technol. , vol.6 , pp. 55-127
    • Hüttenrauch, R.1
  • 13
    • 0036188050 scopus 로고    scopus 로고
    • Influence of tableting on the enzymatic activity of different α-amylases by using various excipients
    • Picker K.M. Influence of tableting on the enzymatic activity of different α-amylases by using various excipients. Eur. J. Pharm. Biopharm. 53:2002;181-185.
    • (2002) Eur. J. Pharm. Biopharm. , vol.53 , pp. 181-185
    • Picker, K.M.1
  • 14
    • 0033014978 scopus 로고    scopus 로고
    • Matrix tablets of carrageenans I. a compaction study
    • Picker K.M. Matrix tablets of carrageenans I. a compaction study. Drug Dev. Ind. Pharm. 25:(3):1999;329-337.
    • (1999) Drug Dev. Ind. Pharm. , vol.25 , Issue.3 , pp. 329-337
    • Picker, K.M.1
  • 15
    • 0033059323 scopus 로고    scopus 로고
    • The use of carrageenan in mixture with microcrystalline cellulose and its functionality for making tablets
    • Picker K.M. The use of carrageenan in mixture with microcrystalline cellulose and its functionality for making tablets. Eur. J. Pharm. Biopharm. 48:1999;27-36.
    • (1999) Eur. J. Pharm. Biopharm. , vol.48 , pp. 27-36
    • Picker, K.M.1
  • 16
    • 0014228967 scopus 로고
    • 1-Acyl-indoles. II A new synthesis of 1-(p-chlorobenzoyl)-5-methoxy-3-indolylacid and its polymorphism
    • Yamamoto H. 1-Acyl-indoles. II A new synthesis of 1-(p-chlorobenzoyl)-5-methoxy-3-indolylacid and its polymorphism. Chem. Pharm. Bull. 16:1968;17-19.
    • (1968) Chem. Pharm. Bull. , vol.16 , pp. 17-19
    • Yamamoto, H.1
  • 17
    • 0017388614 scopus 로고
    • Polymorphism of indomethacin Part I. Preparation of polymorphic forms of indomethacin
    • Pakula R., Pichnej L., Spychala S., Butkiewicz K. Polymorphism of indomethacin Part I. Preparation of polymorphic forms of indomethacin. Pol. J. Pharmacol. Pharm. 29:1977;151-156.
    • (1977) Pol. J. Pharmacol. Pharm. , vol.29 , pp. 151-156
    • Pakula, R.1    Pichnej, L.2    Spychala, S.3    Butkiewicz, K.4
  • 18
    • 0017395498 scopus 로고
    • Polymorphism of indomethacin Part II. identification and rapid determination of polymorphic forms of indomethacin by IR spectrometry
    • Spychala S., Butkiewicz K., Pakula R., Pichnej L. Polymorphism of indomethacin Part II. identification and rapid determination of polymorphic forms of indomethacin by IR spectrometry. Pol. J. Pharmacol. Pharm. 29:1977;157-161.
    • (1977) Pol. J. Pharmacol. Pharm. , vol.29 , pp. 157-161
    • Spychala, S.1    Butkiewicz, K.2    Pakula, R.3    Pichnej, L.4
  • 19
    • 0026705833 scopus 로고
    • Isolation and solid-state characteristics of a new crystal form of indomethacin
    • Lin S.-Y. Isolation and solid-state characteristics of a new crystal form of indomethacin. J. Pharm. Sci. 81:(6):1992;572-576.
    • (1992) J. Pharm. Sci. , vol.81 , Issue.6 , pp. 572-576
    • Lin, S.-Y.1
  • 20
    • 0028597539 scopus 로고
    • Crystallization of indomethacin from the amorphous state below and above its glass transition temperature
    • Yoshioka M., Hancock B.C., Zografi G. Crystallization of indomethacin from the amorphous state below and above its glass transition temperature. J. Pharm. Sci. 83:(12):1994;1700-1705.
    • (1994) J. Pharm. Sci. , vol.83 , Issue.12 , pp. 1700-1705
    • Yoshioka, M.1    Hancock, B.C.2    Zografi, G.3
  • 22
    • 0031750863 scopus 로고    scopus 로고
    • The quantitative analysis of crystallinity using FT-Raman spectroscopy
    • Taylor L.S., Zografi G. The quantitative analysis of crystallinity using FT-Raman spectroscopy. Pharm. Res. 15:(5):1998;755-761.
    • (1998) Pharm. Res. , vol.15 , Issue.5 , pp. 755-761
    • Taylor, L.S.1    Zografi, G.2
  • 23
    • 0033780815 scopus 로고    scopus 로고
    • Evaluation of solid-state forms present in tablets by Raman-spectroscopy
    • Taylor L.S., Langkilde F.W. Evaluation of solid-state forms present in tablets by Raman-spectroscopy. J. Pharm. Sci. 89:(10):2000;1342-1353.
    • (2000) J. Pharm. Sci. , vol.89 , Issue.10 , pp. 1342-1353
    • Taylor, L.S.1    Langkilde, F.W.2
  • 24
    • 0032756138 scopus 로고    scopus 로고
    • Physical properities of solid molecular dispersions of indomethacin with poly(vinylpyrrolidone) and poly(vinylpyrrolidone-co-vinylacetate) in relation to indomethacin crystallisation
    • Matsumoto T., Zografi G. Physical properities of solid molecular dispersions of indomethacin with poly(vinylpyrrolidone) and poly(vinylpyrrolidone-co-vinylacetate) in relation to indomethacin crystallisation. Pharm. Res. 16:(11):1999;1722-1728.
    • (1999) Pharm. Res. , vol.16 , Issue.11 , pp. 1722-1728
    • Matsumoto, T.1    Zografi, G.2
  • 25
    • 0029056118 scopus 로고
    • Inhibition of indomethacin crystallization in poly(vinylpyrrolidone) coprecipitates
    • Yoshioka M., Hancock B.C., Zografi G. Inhibition of indomethacin crystallization in poly(vinylpyrrolidone) coprecipitates. J. Pharm. Sci. 84:(8):1995;983-986.
    • (1995) J. Pharm. Sci. , vol.84 , Issue.8 , pp. 983-986
    • Yoshioka, M.1    Hancock, B.C.2    Zografi, G.3
  • 26
    • 0037694529 scopus 로고
    • Untersuchungen zur Arzneistofffreigabe aus Matrixtabletten und deren Beeinflussung am Beispiel eines Antasthmatikums
    • Universität Halle-Wittenberg
    • G. Zessin, Untersuchungen zur Arzneistofffreigabe aus Matrixtabletten und deren Beeinflussung am Beispiel eines Antasthmatikums, Habilitationsschrift, Universität Halle-Wittenberg, 1976.
    • (1976) Habilitationsschrift
    • Zessin, G.1
  • 27
    • 0035123570 scopus 로고    scopus 로고
    • Time dependence of elastic recovery of characterization of tableting materials
    • Picker K.M. Time dependence of elastic recovery of characterization of tableting materials. Pharm. Dev. Technol. 6:2001;61-70.
    • (2001) Pharm. Dev. Technol. , vol.6 , pp. 61-70
    • Picker, K.M.1
  • 28
    • 0031423468 scopus 로고    scopus 로고
    • Spectroscopic characterization of interactions between PVP and indomethacin in amorphous molecular dispersions
    • Taylor L.S., Zografi G. Spectroscopic characterization of interactions between PVP and indomethacin in amorphous molecular dispersions. Pharm. Res. 14:(12):1997;1691-1698.
    • (1997) Pharm. Res. , vol.14 , Issue.12 , pp. 1691-1698
    • Taylor, L.S.1    Zografi, G.2
  • 29
    • 0000292691 scopus 로고
    • Density-pressure relationships in powder compaction
    • Heckel R.W. Density-pressure relationships in powder compaction. Trans. Metal. Soc. AIME. 221:(8):1961;671-675.
    • (1961) Trans. Metal. Soc. AIME , vol.221 , Issue.8 , pp. 671-675
    • Heckel, R.W.1
  • 30
    • 0000693333 scopus 로고
    • An analysis of powder compaction phenomena
    • Heckel R.W. An analysis of powder compaction phenomena. Trans. Metal. Soc. AIME. 221:(10):1961;1001-1008.
    • (1961) Trans. Metal. Soc. AIME , vol.221 , Issue.10 , pp. 1001-1008
    • Heckel, R.W.1
  • 31
    • 0034595280 scopus 로고    scopus 로고
    • A new theoretical model to characterize the densification behavior of tableting materials
    • Picker K.M. A new theoretical model to characterize the densification behavior of tableting materials. Eur. J. Pharm. Biopharm. 49:2000;267-273.
    • (2000) Eur. J. Pharm. Biopharm. , vol.49 , pp. 267-273
    • Picker, K.M.1
  • 32
    • 0030695783 scopus 로고    scopus 로고
    • Use of Raman spectroscopy for the quantitative analysis of calcium oxalate hydrate: Applications for the analysis of urinary stones
    • Kontoyannis C.G., Bouropoulos N.C., Koutsoukos P.G. Use of Raman spectroscopy for the quantitative analysis of calcium oxalate hydrate: applications for the analysis of urinary stones. Appl. Spectrosc. 51:(1):1997;64-67.
    • (1997) Appl. Spectrosc. , vol.51 , Issue.1 , pp. 64-67
    • Kontoyannis, C.G.1    Bouropoulos, N.C.2    Koutsoukos, P.G.3
  • 33
    • 0031056536 scopus 로고    scopus 로고
    • Effects of sorbed water on the crystallization of indomethacin from the amorphous state
    • Andronis V., Yoshioka M., Zografi G. Effects of sorbed water on the crystallization of indomethacin from the amorphous state. J. Pharm. Sci. 86:(3):1997;346-351.
    • (1997) J. Pharm. Sci. , vol.86 , Issue.3 , pp. 346-351
    • Andronis, V.1    Yoshioka, M.2    Zografi, G.3
  • 34
    • 0022601812 scopus 로고
    • Effect of environmental temperature on polymorphic solid-state transformation of indomethacin during grinding
    • Otsuka M., Matsumoto T., Kaneniwa N. Effect of environmental temperature on polymorphic solid-state transformation of indomethacin during grinding. Chem. Pharm. Bull. 34:(4):1986;1784-1793.
    • (1986) Chem. Pharm. Bull. , vol.34 , Issue.4 , pp. 1784-1793
    • Otsuka, M.1    Matsumoto, T.2    Kaneniwa, N.3
  • 35
    • 0031782493 scopus 로고    scopus 로고
    • The molecular mobility of supercooled amorphous indomethacin as a function of temperature and relative humidity
    • Andronis V., Zografi G. The molecular mobility of supercooled amorphous indomethacin as a function of temperature and relative humidity. Pharm. Res. 15:(6):1998;835-843.
    • (1998) Pharm. Res. , vol.15 , Issue.6 , pp. 835-843
    • Andronis, V.1    Zografi, G.2
  • 36
    • 0030724408 scopus 로고    scopus 로고
    • Polymorphism in anhydrous theophylline-implications on the dissolution rate of theophylline tablets
    • Phadnis N.V., Suryanarayanan R. Polymorphism in anhydrous theophylline-implications on the dissolution rate of theophylline tablets. J. Pharm. Sci. 86:(11):1997;1256-1263.
    • (1997) J. Pharm. Sci. , vol.86 , Issue.11 , pp. 1256-1263
    • Phadnis, N.V.1    Suryanarayanan, R.2
  • 38
    • 0024560872 scopus 로고
    • Thermochemical study of theophylline and its hydrate
    • Suzuki E., Shimomura K., Sekiguchi K. Thermochemical study of theophylline and its hydrate. Chem. Pharm. Bull. 37:(2):1989;493-497.
    • (1989) Chem. Pharm. Bull. , vol.37 , Issue.2 , pp. 493-497
    • Suzuki, E.1    Shimomura, K.2    Sekiguchi, K.3
  • 39
    • 0015620251 scopus 로고
    • Dehydration of crystalline theophylline monohydrate and ampicillin trihydrate
    • Shefter E., Fung H.-L. Dehydration of crystalline theophylline monohydrate and ampicillin trihydrate. J. Pharm. Sci. 62:(5):1973;791-794.
    • (1973) J. Pharm. Sci. , vol.62 , Issue.5 , pp. 791-794
    • Shefter, E.1    Fung, H.-L.2
  • 40
    • 0028273709 scopus 로고
    • Dehydration of theophylline monohydrate - Effects of particle size and sample weight
    • Agbade C.O., York P. Dehydration of theophylline monohydrate - effects of particle size and sample weight. Int. J. Pharm. 106:1994;33-40.
    • (1994) Int. J. Pharm. , vol.106 , pp. 33-40
    • Agbade, C.O.1    York, P.2
  • 41
    • 0024241277 scopus 로고
    • The dehydration kinetics of theophylline monohydrate - Powder and tablet
    • Otsuka M., Kaneniwa N. The dehydration kinetics of theophylline monohydrate - powder and tablet. Chem. Pharm. Bull. 36:(12):1988;4914-4920.
    • (1988) Chem. Pharm. Bull. , vol.36 , Issue.12 , pp. 4914-4920
    • Otsuka, M.1    Kaneniwa, N.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.