The interaction of a constitutively active arrestin with the arrestin-insensitive 5-HT2A receptor induces agonist-independent internalization

Molecular Pharmacology

Volumn 63, Issue 5, 2003, Pages 961-972

  Gray, John A ^a   Bhatnagar, Anushree ^a   Gurevich, Vsevolod V ^b   Roth, Bryan L ^a  

^a CASE WESTERN RESERVE UNIVERSITY SCHOOL OF MEDICINE   (United States)

^b VANDERBILT UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

3,3' DITHIOBIS(SUCCINIMIDYL PROPIONATE); 4 IODO 2,5 DIMETHOXYAMPHETAMINE; CLOZAPINE; G PROTEIN COUPLED RECEPTOR; INOSITOL; KETANSERIN; MUTANT PROTEIN; PHENOXYBENZAMINE; PHOSPHATIDYLINOSITIDE; QUIPAZINE; RADIOLIGAND; RETINA S ANTIGEN; RITANSERIN; SEROTONIN; SEROTONIN 2A AGONIST; SEROTONIN 2A RECEPTOR; SPIPERONE;

ARTICLE; CELL CULTURE; CONFOCAL MICROSCOPY; CONTROLLED STUDY; CROSS LINKING; DRUG RECEPTOR BINDING; GENETIC TRANSFECTION; HUMAN; HUMAN CELL; HYDROLYSIS; IMMUNOCYTOCHEMISTRY; INTERNALIZATION; PRIORITY JOURNAL; PROTEIN PHOSPHORYLATION; RECEPTOR AFFINITY; RECEPTOR DOWN REGULATION; RECEPTOR UPREGULATION; WESTERN BLOTTING;

AMINO ACID SUBSTITUTION; ARRESTINS; CELLS, CULTURED; GLUTAMIC ACID; HUMANS; HYDROLYSIS; NEURONS; PHOSPHOPROTEINS; PHOSPHORYLATION; PROTEIN CONFORMATION; RECEPTOR, SEROTONIN, 5-HT2A; RECEPTORS, SEROTONIN; TRANSFECTION; TYROSINE;

EID: 0037847585     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.63.5.961     Document Type: Article

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