메뉴 건너뛰기




Volumn 98, Issue 3, 2003, Pages 741-747

The role of 5-HT1A/B autoreceptors in the antinociceptive effect of systemic administration of acetaminophen

Author keywords

[No Author keywords available]

Indexed keywords

2 DIPROPYLAMINO 8 HYDROXYTETRALIN; 3 (1,2,5,6 TETRAHYDRO 4 PYRIDYL)PYRROLO[3,2 B]PYRIDIN 5 ONE; N 3 [3 (DIMETHYLAMINOETHOXY) 4 METHOXYPHENYL] 2' METHYL 4' (5 METHYL 1,2,4 OXADIAZOL 3 YL) 1,1' BIPHENYL 4 CARBOXAMIDE; N [2 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL]ETHYL] N (2 PYRIDYL)CYCLOHEXANECARBOXAMIDE; PARACETAMOL; SB 216641; SEROTONIN 1A ANTAGONIST; SEROTONIN 1A RECEPTOR; SEROTONIN 1B AGONIST; SEROTONIN 1B RECEPTOR; SODIUM CHLORIDE; UNCLASSIFIED DRUG; 3 (1,2,5,6 TETRAHYDROPYRID 4 YL)PYRROLO(3,2 B)PYRID 5 ONE; 3-(1,2,5,6-TETRAHYDROPYRID-4-YL)PYRROLO(3,2-B)PYRID-5-ONE; ANALGESIC AGENT; AUTORECEPTOR; BENZAMIDE DERIVATIVE; N (3 (2 DIMETHYLAMINO)ETHOXY 4 METHOXYPHENYL) 2' METHYL 4' (5 METHYL 1,2,4 OXADIAZOL 3 YL) (1,1' BIPHENYL) 4 CARBOXAMIDE; N-(3-(2-DIMETHYLAMINO)ETHOXY-4-METHOXYPHENYL)-2'-METHYL-4'-(5-METHYL-1,2,4-OXADIAZOL-3-YL)-(1,1'-BIPHENYL)-4-CARBOXAMIDE; OXADIAZOLE DERIVATIVE; PYRIDINE DERIVATIVE; PYRROLE DERIVATIVE; SEROTONIN 1 RECEPTOR; SEROTONIN RECEPTOR;

EID: 0037370477     PISSN: 00033022     EISSN: None     Source Type: Journal    
DOI: 10.1097/00000542-200303000-00025     Document Type: Article
Times cited : (27)

References (43)
  • 1
    • 0028830040 scopus 로고
    • Central antinociceptive effects of non-steroidal anti-inflammatory drugs and paracetamol: Experimental studies in rat
    • Bjorkman R: Central antinociceptive effects of non-steroidal anti-inflammatory drugs and paracetamol: Experimental studies in rat. Acta Anaesthesiol Scand 1995; 103:1-44
    • (1995) Acta Anaesthesiol Scand , vol.103 , pp. 1-44
    • Bjorkman, R.1
  • 3
    • 0021288912 scopus 로고
    • Endogenous pain control system: Brainstem spinal pathways and endorphin circuitry
    • Basbaum A, Fields H: Endogenous pain control system: Brainstem spinal pathways and endorphin circuitry. Annu Rev Neurosci 1984; 7:309-38
    • (1984) Annu Rev Neurosci , vol.7 , pp. 309-338
    • Basbaum, A.1    Fields, H.2
  • 4
    • 0028276669 scopus 로고
    • The dorsal raphe: An important nucleus in pain modulation
    • Wang Q, Nakai Y: The dorsal raphe: An important nucleus in pain modulation. Brain Res Bull 1994; 34:575-85
    • (1994) Brain Res Bull , vol.34 , pp. 575-585
    • Wang, Q.1    Nakai, Y.2
  • 5
    • 0025309380 scopus 로고
    • Role of serotonergic systems in morphine-induced antinociception
    • Edited by Besson J. La-Roque-Gageac, France, Elsevier
    • Hammond D: Role of serotonergic systems in morphine-induced antinociception, Serotonin and Pain. Edited by Besson J. La-Roque-Gageac, France, Elsevier, 1990, pp 251-61
    • (1990) Serotonin and Pain , pp. 251-261
    • Hammond, D.1
  • 6
    • 0033178543 scopus 로고    scopus 로고
    • Central mechanisms of pain modulation
    • Mason P: Central mechanisms of pain modulation. Curr Opin Neurobiol 1999; 9:436-41
    • (1999) Curr Opin Neurobiol , vol.9 , pp. 436-441
    • Mason, P.1
  • 8
    • 0034307766 scopus 로고    scopus 로고
    • Control of dorsal raphe 5-HT function by multiple 5-HT(1) autoreceptors: Parallel purposes or pointless plurality?
    • Stamford JA, Davidson C, McLaughlin DP, Hopwood SE: Control of dorsal raphe 5-HT function by multiple 5-HT(1) autoreceptors: Parallel purposes or pointless plurality? Trends Neurosci 2000; 23:459-65
    • (2000) Trends Neurosci , vol.23 , pp. 459-465
    • Stamford, J.A.1    Davidson, C.2    McLaughlin, D.P.3    Hopwood, S.E.4
  • 10
    • 0029665352 scopus 로고    scopus 로고
    • 1A autoreceptors and the mode of action of selective serotonin reuptake inhibitors (SSRI)
    • 1A autoreceptors and the mode of action of selective serotonin reuptake inhibitors (SSRI). Behav Brain Res 1996; 73:281-3
    • (1996) Behav Brain Res , vol.73 , pp. 281-283
    • Hjorth, S.1    Auerbach, S.B.2
  • 11
    • 0029892782 scopus 로고    scopus 로고
    • 1D autoreceptors on the modulation of 5-HT release in guinea-pig mesencephalic raphe, hippocampus and frontal cortex
    • 1D autoreceptors on the modulation of 5-HT release in guinea-pig mesencephalic raphe, hippocampus and frontal cortex. Br J Pharmacol 1996; 118:681-9
    • (1996) Br J Pharmacol , vol.118 , pp. 681-689
    • El Mansari, M.1    Blier, P.2
  • 13
    • 0034333003 scopus 로고    scopus 로고
    • Pindolol, a beta-adrenoceptor blocker/5-hydroxytryptamine 1A/1B antagonist, enhances the analgesic effect of tramadol
    • Rojas-Corrales M, Ortega-Álvaro A, Gibert-Rahola J, Roca-Vinardell A, Micó J: Pindolol, a beta-adrenoceptor blocker/5-hydroxytryptamine 1A/1B antagonist, enhances the analgesic effect of tramadol. Pain 2000; 88:119-24
    • (2000) Pain , vol.88 , pp. 119-124
    • Rojas-Corrales, M.1    Ortega-Álvaro, A.2    Gibert-Rahola, J.3    Roca-Vinardell, A.4    Micó, J.5
  • 14
    • 0035085494 scopus 로고    scopus 로고
    • Potentiation of the antinociceptive effect of clomipramine by a 5-HT(1A) antagonist in neuropathic pain in rats
    • Ardid D, Alloui A, Brousse G, Jourdan D, Picard P, Dubray C, Eschalier A: Potentiation of the antinociceptive effect of clomipramine by a 5-HT(1A) antagonist in neuropathic pain in rats. Br J Pharmacol 2001; 132:1118-26
    • (2001) Br J Pharmacol , vol.132 , pp. 1118-1126
    • Ardid, D.1    Alloui, A.2    Brousse, G.3    Jourdan, D.4    Picard, P.5    Dubray, C.6    Eschalier, A.7
  • 15
    • 0025845133 scopus 로고
    • 1A agonists attenuate morphine-induced antinociception in mice in a competitive-like manner
    • 1A agonists attenuate morphine-induced antinociception in mice in a competitive-like manner. J Pharmacol Exp Ther 1991; 256:983-92
    • (1991) J Pharmacol Exp Ther , vol.256 , pp. 983-992
    • Millan, M.J.1    Colpaert, F.C.2
  • 16
    • 0020525719 scopus 로고
    • Ethical guidelines for investigations of experimental pain in conscious animals
    • IASP: Ethical guidelines for investigations of experimental pain in conscious animals. Pain 1980; 16:109-10
    • (1980) Pain , vol.16 , pp. 109-110
  • 17
    • 0000811019 scopus 로고
    • The evaluation of the analgesic action of pethidine hydrochloride
    • Woolfe H, MacDonald A: The evaluation of the analgesic action of pethidine hydrochloride. J Pharmacol Exp Ther 1944; 80:300-7
    • (1944) J Pharmacol Exp Ther , vol.80 , pp. 300-307
    • Woolfe, H.1    MacDonald, A.2
  • 18
    • 0038899949 scopus 로고    scopus 로고
    • The antinociceptive action of paracetamol is associated with changes in the serotonergic system in the rat brain
    • Pini L, Sandrini M, Vitale G: The antinociceptive action of paracetamol is associated with changes in the serotonergic system in the rat brain. Eur J Pharmacol 1996; 308:31-40
    • (1996) Eur J Pharmacol , vol.308 , pp. 31-40
    • Pini, L.1    Sandrini, M.2    Vitale, G.3
  • 19
    • 0030898943 scopus 로고    scopus 로고
    • Naloxone-reversible antinociception by paracetamol in the rat
    • Pini L, Vitale G, Ottani A, Sandrini M: Naloxone-reversible antinociception by paracetamol in the rat. J Pharmacol Exp Ther 1997; 280:934-40
    • (1997) J Pharmacol Exp Ther , vol.280 , pp. 934-940
    • Pini, L.1    Vitale, G.2    Ottani, A.3    Sandrini, M.4
  • 21
    • 0033024898 scopus 로고    scopus 로고
    • The potentiation of analgesic activity of paracetamol plus morphine involves the serotonergic system in rat brain
    • Sandrini M, Vitale G, Ottani A, Pini L: The potentiation of analgesic activity of paracetamol plus morphine involves the serotonergic system in rat brain. Inflamm Res 1999; 48:120-7
    • (1999) Inflamm Res , vol.48 , pp. 120-127
    • Sandrini, M.1    Vitale, G.2    Ottani, A.3    Pini, L.4
  • 22
    • 0034936102 scopus 로고    scopus 로고
    • The influence of divalent cations on the analgesic effect of opioid and non-opioid drugs
    • Assi AA: The influence of divalent cations on the analgesic effect of opioid and non-opioid drugs. Pharmacol Res 2001; 43:521-9
    • (2001) Pharmacol Res , vol.43 , pp. 521-529
    • Assi, A.A.1
  • 23
    • 0037052047 scopus 로고    scopus 로고
    • Synthesis and pharmacological properties of benzisothiazole/benzimidazole derivates with acidic groups
    • Vincini P, Incerti M, Amoretti L, Ballabeni V, Tognolini M, Barocelli E: Synthesis and pharmacological properties of benzisothiazole/benzimidazole derivates with acidic groups. Il Farmaco 2002; 57:363-7
    • (2002) Il Farmaco , vol.57 , pp. 363-367
    • Vincini, P.1    Incerti, M.2    Amoretti, L.3    Ballabeni, V.4    Tognolini, M.5    Barocelli, E.6
  • 24
    • 0026022639 scopus 로고
    • Antinociceptive effect of paracetamol in rats is partly dependent on spinal serotonergic systems
    • Tjolsen A, Lund A, Hole K: Antinociceptive effect of paracetamol in rats is partly dependent on spinal serotonergic systems. Eur J Pharmacol 1991; 193:193-201
    • (1991) Eur J Pharmacol , vol.193 , pp. 193-201
    • Tjolsen, A.1    Lund, A.2    Hole, K.3
  • 25
    • 0033017947 scopus 로고    scopus 로고
    • Acetaminophen-induced antinociception via central 5-HT(2A) receptors
    • Srikiatkhachorn A, Tarasub N, Govitrapong P: Acetaminophen-induced antinociception via central 5-HT(2A) receptors. Neurochem Int 1999; 34:491-8
    • (1999) Neurochem Int , vol.34 , pp. 491-498
    • Srikiatkhachorn, A.1    Tarasub, N.2    Govitrapong, P.3
  • 26
    • 0033990859 scopus 로고    scopus 로고
    • 1B and 5-HT1D autoreceptors in rat dorsal raphe nucleus
    • 1B and 5-HT1D autoreceptors in rat dorsal raphe nucleus. Neurochem Int 2000; 36:91-6
    • (2000) Neurochem Int , vol.36 , pp. 91-96
    • Davidson, C.1    Stamford, J.A.2
  • 27
    • 0034099924 scopus 로고    scopus 로고
    • 1B/1D receptors on the modulation of acute fluoxetine-induced changes in extracellular 5-HT: The mechanism of action of (±)pindolol
    • 1B/1D receptors on the modulation of acute fluoxetine-induced changes in extracellular 5-HT: The mechanism of action of (±)pindolol. Neuropharmacology 2000; 39:1044-52
    • (2000) Neuropharmacology , vol.39 , pp. 1044-1052
    • Dawson, L.1    Nguyen, H.2
  • 28
    • 0032905345 scopus 로고    scopus 로고
    • Pindolol and mianserin augment the antidepressant activity of fluoxetine in hospitalized major depressed patients, including those with treatment resistance
    • Maes M, Libbrecht I, van Hunsel F, Campens D, Meltzer HY: Pindolol and mianserin augment the antidepressant activity of fluoxetine in hospitalized major depressed patients, including those with treatment resistance. J Clin Psychopharmacol 1999; 19:177-82
    • (1999) J Clin Psychopharmacol , vol.19 , pp. 177-182
    • Maes, M.1    Libbrecht, I.2    Van Hunsel, F.3    Campens, D.4    Meltzer, H.Y.5
  • 29
    • 0035141862 scopus 로고    scopus 로고
    • Augmentation of fluoxetine's antidepressant action by pindolol: Analysis of clinical, pharmacokinetic, and methodologic factors
    • Perez V, Puiigdemont D, Gilaberte I, Alvarez E, Artigas F: Augmentation of fluoxetine's antidepressant action by pindolol: Analysis of clinical, pharmacokinetic, and methodologic factors. J Clin Psychopharmacol 2001; 21:36-45
    • (2001) J Clin Psychopharmacol , vol.21 , pp. 36-45
    • Perez, V.1    Puiigdemont, D.2    Gilaberte, I.3    Alvarez, E.4    Artigas, F.5
  • 30
    • 0032509709 scopus 로고    scopus 로고
    • WAY 100,635 enhances both the "antidepressant" actions of duloxetine and its influence on dialysate levels of serotonin in frontal cortex
    • Millan MJ, Brocco M, Veiga S, Cistarelli L, Melon C, Gobert A: WAY 100,635 enhances both the "antidepressant" actions of duloxetine and its influence on dialysate levels of serotonin in frontal cortex. Eur J Pharmacol 1998; 341:165-7
    • (1998) Eur J Pharmacol , vol.341 , pp. 165-167
    • Millan, M.J.1    Brocco, M.2    Veiga, S.3    Cistarelli, L.4    Melon, C.5    Gobert, A.6
  • 32
    • 0030056145 scopus 로고    scopus 로고
    • Neuronal release of serotonin in the cerebellum of behaving rats: An in vivo microdialysis study
    • Mendlin A, Martin FJ, Rueter LE, Jacobs BL: Neuronal release of serotonin in the cerebellum of behaving rats: An in vivo microdialysis study. J Neurochem 1996; 67:617-22
    • (1996) J Neurochem , vol.67 , pp. 617-622
    • Mendlin, A.1    Martin, F.J.2    Rueter, L.E.3    Jacobs, B.L.4
  • 33
    • 0021690107 scopus 로고
    • Rapid agonist-induced decrease of 125I-pindolol binding to beta-adrenergic receptors: Relationship to desensitization of cyclic AMP accumulation in intact heart cells
    • Linden J, Patel A, Spanier AM, Weglicki WB: Rapid agonist-induced decrease of 125I-pindolol binding to beta-adrenergic receptors: Relationship to desensitization of cyclic AMP accumulation in intact heart cells. J Biol Chem 1984; 259:15115-22
    • (1984) J Biol Chem , vol.259 , pp. 15115-15122
    • Linden, J.1    Patel, A.2    Spanier, A.M.3    Weglicki, W.B.4
  • 35
    • 0035823421 scopus 로고    scopus 로고
    • 1B binding sites after intra-hippocampal ibotenic acid injections in the rat
    • 1B binding sites after intra-hippocampal ibotenic acid injections in the rat. Neurosci Lett 2001; 310:25-8
    • (2001) Neurosci Lett , vol.310 , pp. 25-28
    • Ait Amara, D.1    Segu, L.2    Buhot, M.C.3
  • 36
    • 0028240934 scopus 로고
    • Serotonin receptor subtypes in spinal antinociception in the rat
    • Xu W, Qiu XC, Han JS: Serotonin receptor subtypes in spinal antinociception in the rat. J Pharmacol Exp Ther 1994; 269:1182-9
    • (1994) J Pharmacol Exp Ther , vol.269 , pp. 1182-1189
    • Xu, W.1    Qiu, X.C.2    Han, J.S.3
  • 37
    • 0035976823 scopus 로고    scopus 로고
    • 5-HT receptor subtypes involved in the spinal antinociceptive effect of acetaminophen in rats
    • Courade JP, Chassaing C, Bardin L, Alloui A, Eschalier A: 5-HT receptor subtypes involved in the spinal antinociceptive effect of acetaminophen in rats. Eur J Pharmacol 2001; 432:1-7
    • (2001) Eur J Pharmacol , vol.432 , pp. 1-7
    • Courade, J.P.1    Chassaing, C.2    Bardin, L.3    Alloui, A.4    Eschalier, A.5
  • 38
    • 0027524905 scopus 로고
    • In vivo microdialysis evidence for central serotonin1A and serotonin1B autoreceptor blocking properties of the beta adrenoceptor antagonist (-)penbutolol
    • Hjorth S, Sharp T: In vivo microdialysis evidence for central serotonin1A and serotonin1B autoreceptor blocking properties of the beta adrenoceptor antagonist (-)penbutolol. J Pharmacol Exp Ther 1993; 265:707-12
    • (1993) J Pharmacol Exp Ther , vol.265 , pp. 707-712
    • Hjorth, S.1    Sharp, T.2
  • 39
    • 0030011682 scopus 로고    scopus 로고
    • Lack of binding of acetaminophen to 5-HT receptor or uptake sites (or eleven other binding/uptake assays)
    • Raffa R, Codd E: Lack of binding of acetaminophen to 5-HT receptor or uptake sites (or eleven other binding/uptake assays). Life Sci 1996; 59:37-40
    • (1996) Life Sci , vol.59 , pp. 37-40
    • Raffa, R.1    Codd, E.2
  • 40
    • 0028940655 scopus 로고
    • Involvement of brain serotonergic system in the antinociceptive action of acetylsalicylic acid in the rat
    • Pini L, Sandrini M, Vitale G: Involvement of brain serotonergic system in the antinociceptive action of acetylsalicylic acid in the rat. Inflamm Res 1995; 44:30-5
    • (1995) Inflamm Res , vol.44 , pp. 30-35
    • Pini, L.1    Sandrini, M.2    Vitale, G.3
  • 41
    • 0029787774 scopus 로고    scopus 로고
    • Analgesic efficacy and safety of paracetamol-codeine combinations versus paracetamol alone: A systematic review
    • de Craen A, Di Giulio G, Lampe-Schoenmaeckers J, Kessels A, Kleijnen J: Analgesic efficacy and safety of paracetamol-codeine combinations versus paracetamol alone: A systematic review. BMJ 1996; 313:321-5
    • (1996) BMJ , vol.313 , pp. 321-325
    • De Craen, A.1    Di Giulio, G.2    Lampe-Schoenmaeckers, J.3    Kessels, A.4    Kleijnen, J.5
  • 42
    • 0033834590 scopus 로고    scopus 로고
    • Ibuprofen plus caffeine in the treatment of tension-type headache
    • Diamond S, Balm TK, Freitag FG: Ibuprofen plus caffeine in the treatment of tension-type headache. Clin Pharmacol Ther 2000; 68:312-9
    • (2000) Clin Pharmacol Ther , vol.68 , pp. 312-319
    • Diamond, S.1    Balm, T.K.2    Freitag, F.G.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.