Searching for allosteric effects via QSAR. Part II

Bioorganic and Medicinal Chemistry

Volumn 11, Issue 4, 2002, Pages 621-628

  Garg, Rajni ^a   Kurup, Alka ^a   Mekapati, Suresh B ^a   Hansch, Corwin ^a  

^a POMONA COLLEGE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANTIINFECTIVE AGENT; CARBANILAMIDE DERIVATIVE; CARBOXYPEPTIDASE A; CYCLIC AMP; DOPAMINE RECEPTOR; ENZYME INHIBITOR; EPIDERMAL GROWTH FACTOR RECEPTOR; EPOXIDE HYDROLASE; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); LEUKOCYTE ELASTASE INHIBITOR; METABOTROPIC RECEPTOR; MUSCARINIC AGENT; MUSCARINIC M3 RECEPTOR; SERINE PROTEINASE INHIBITOR; SEROTONIN 1D RECEPTOR; SULFUR 35; THROMBIN INHIBITOR; THROMBIN RECEPTOR; TYROSINE KINASE RECEPTOR;

ALLOSTERISM; ANTIMICROBIAL ACTIVITY; ARTICLE; AUTOPHOSPHORYLATION; BACTERIAL GROWTH; CALCULATION; CELL TYPE; DNA CLEAVAGE; DRUG EFFECT; ENZYME INHIBITION; HUMAN; HYDROLYSIS; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; QUANTITATIVE STRUCTURE ACTIVITY RELATION; X RAY CRYSTALLOGRAPHY;

ALGORITHMS; ANIMALS; CARBOXYPEPTIDASES; CARBOXYPEPTIDASES A; CHO CELLS; CRICETINAE; DNA TOPOISOMERASES, TYPE II; DRUG DESIGN; ENZYME INHIBITORS; EPOXIDE HYDROLASES; ESCHERICHIA COLI; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); GUINEA PIGS; HUMANS; ILEUM; LEUKOCYTE ELASTASE; LIGANDS; MICE; MICROBIAL SENSITIVITY TESTS; MUSCLE CONTRACTION; MUSCLE, SMOOTH; QUANTITATIVE STRUCTURE-ACTIVITY RELATIONSHIP; RATS; RECEPTOR, EPIDERMAL GROWTH FACTOR; RECEPTOR, MUSCARINIC M3; RECEPTORS, DRUG; RECEPTORS, METABOTROPIC GLUTAMATE; RECEPTORS, MUSCARINIC; SERINE PROTEINASE INHIBITORS; THROMBIN;

EID: 0037252016     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0968-0896(02)00382-6     Document Type: Article

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