Parallel solution- and solid-phase synthesis of spirohydantoin derivatives as neurokinin-1 receptor ligands

Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 18, 2002, Pages 2519-2522

  Bleicher, Konrad H ^a   Wüthrich, Yves ^a   De Boni, Maxime ^a   Kolczewski, Sabine ^a   Hoffmann, Torsten ^a   Sleight, Andrew J ^a  

^a F HOFFMANN LA ROCHE LTD   (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

BENZENE DERIVATIVE; G PROTEIN COUPLED RECEPTOR; HYDANTOIN DERIVATIVE; LIGAND; NEUROKININ 1 RECEPTOR;

ARTICLE; BINDING AFFINITY; DRUG ACTIVITY; DRUG SYNTHESIS; METHODOLOGY; SOLID; STEREOCHEMISTRY; STRUCTURE ACTIVITY RELATION;

COMBINATORIAL CHEMISTRY TECHNIQUES; LIGANDS; RECEPTORS, NEUROKININ-1; SPIRO COMPOUNDS;

EID: 0037119745     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(02)00488-2     Document Type: Article

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