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Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 1, 2002, Pages 5-8

Phthalazine PDE4 inhibitors. Part 3: The synthesis and in vitro evaluation of derivatives with a hydrogen bond acceptor

(8) Napoletano, Mauro a Norcini, Gabriele c Pellacini, Franco a Marchini, Francesco b Morazzoni, Gabriele a Fattori, Raimondo a Ferlenga, Pierpaolo b Pradella, Lorenzo b

a Zambon Group (Switzerland)

b Zambon Group SpA (Italy)

c Lamberti SpA (Italy)

Author keywords

[No Author keywords available]

Indexed keywords

CILOMILAST; GW 3600; PHOSPHODIESTERASE IV INHIBITOR; PHTHALAZINE DERIVATIVE; PICLAMILAST; ROLIPRAM; UNCLASSIFIED DRUG;

ARTICLE; DRUG BINDING SITE; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; ENZYME INHIBITION; HUMAN; HYDROGEN BOND; STRUCTURE ACTIVITY RELATION;

3',5'-CYCLIC-NUCLEOTIDE PHOSPHODIESTERASE; BINDING SITES; DRUG DESIGN; DRUG EVALUATION, PRECLINICAL; HUMANS; HYDROGEN BONDING; NEUTROPHILS; PHOSPHODIESTERASE INHIBITORS; PHTHALAZINES; ROLIPRAM; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0037033177 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/S0960-894X(01)00668-0 Document Type: Article

Times cited : (21)

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