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Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 1, 2002, Pages 101-104

Potent P1′ biphenylmethyl substituted aggrecanase inhibitors

(9) Yao, Wenqing a Chao, Michael a Wasserman, Zelda R a Liu, Rui Qin a Covington, Maryanne B a Newton, Robert a Christ, David a Wexler, Ruth R a Decicco, Carl P a

a BRISTOL MYERS SQUIBB (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AGGRECANASE; BIPHENYL; ENZYME INHIBITOR; GELATINASE A; GELATINASE B; INTERSTITIAL COLLAGENASE; ANTIRHEUMATIC AGENT; BIPHENYL DERIVATIVE; METALLOPROTEINASE; PROTEINASE; PROTEINASE INHIBITOR;

ARTICLE; DRUG BINDING; DRUG CONFORMATION; DRUG POTENCY; DRUG SELECTIVITY; DRUG SYNTHESIS; IC 50; OSTEOARTHRITIS; STRUCTURE ACTIVITY RELATION; CHEMISTRY; DRUG DESIGN; DRUG SCREENING; ENZYME ACTIVE SITE; ENZYME SPECIFICITY; HUMAN; METABOLISM; SYNTHESIS;

ANTIRHEUMATIC AGENTS; BIPHENYL COMPOUNDS; CATALYTIC DOMAIN; DRUG DESIGN; DRUG EVALUATION, PRECLINICAL; ENDOPEPTIDASES; HUMAN; INHIBITORY CONCENTRATION 50; METALLOENDOPEPTIDASES; PROTEASE INHIBITORS; STRUCTURE-ACTIVITY RELATIONSHIP; SUBSTRATE SPECIFICITY;

EID: 0037033136 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/S0960-894X(01)00704-1 Document Type: Article

Times cited : (33)

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