Highly potent non-peptidic inhibitors of the HCV NS3/NS4A serine protease

Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 21, 2002, Pages 3129-3133

  Sperandio, David ^a   Gangloff, Anthony R ^a   Litvak, Joane ^a   Goldsmith, Richard ^a   Hataye, Jason M ^a   Wang, Vivian R ^a   Shelton, Emma J ^a   Elrod, Kyle ^a   Janc, James W ^a   Clark, James M ^a   Rice, Ken ^a   Weinheimer, Steve ^b   Yeung, Kap Sun ^b   Meanwell, Nicholas A ^b   Hernandez, Dennis ^b   Staab, Andrew J ^b   Venables, Brian L ^b   Spencer, Jeffrey R ^a  

^a Bristol Myers Squibb Pharmaceutical Research Institute ^*  (United States)

^b BRISTOL MYERS SQUIBB   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

EDETIC ACID; PIBENZIMOL; SERINE PROTEINASE; SERINE PROTEINASE INHIBITOR; VIRUS ENZYME; ZINC ION;

ARTICLE; BINDING AFFINITY; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; ENZYME BINDING; HEPATITIS C VIRUS; PROTEINASE INHIBITION; STRUCTURE ACTIVITY RELATION;

BENZIMIDAZOLES; EDETIC ACID; HEPACIVIRUS; INDICATORS AND REAGENTS; PEPTIDES; RNA, VIRAL; SERINE PROTEINASE INHIBITORS; STRUCTURE-ACTIVITY RELATIONSHIP; VIRAL NONSTRUCTURAL PROTEINS; ZINC;

HEPATITIS C VIRUS;

EID: 0037020737     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(02)00680-7     Document Type: Article

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