In vitro metabolic characteristics of cytochrome P-450 2A6 in Chinese liver microsomes

Acta Pharmacologica Sinica

Volumn 23, Issue 5, 2002, Pages 471-476

  Xia, Xue Yan ^a   Peng, Ren Xiu ^a   Yu, Jie Ping ^b   Wang, Hui ^a   Wang, Jun ^a  

^a WUHAN UNIVERSITY   (China)

^b RENMIN HOSPITAL OF WUHAN UNIVERSITY   (China)

Author keywords

Coumarins; Cytochrome P 450 CYP2A6; Glucuronosyltransferase; Liver microsomes; Rifampicin

Indexed keywords

ALPHA NAPHTHOFLAVONE; AZITHROMYCIN; COUMARIN 7 HYDROXYLASE; CYTOCHROME P450; CYTOCHROME P450 2A6; DIETHYLDITHIOCARBAMIC ACID; ENZYME INHIBITOR; PILOCARPINE; RIFAMPICIN; SULFAPHENAZOLE; TROLEANDOMYCIN; XENOBIOTIC AGENT; COUMARIN 7-HYDROXYLASE; GLUCURONOSYLTRANSFERASE; MIXED FUNCTION OXIDASE; UNSPECIFIC MONOOXYGENASE;

ARTICLE; BIOCHEMISTRY; ENZYME ACTIVITY; ENZYME INHIBITION; ENZYME KINETICS; HUMAN; HUMAN TISSUE; HYDROXYLATION; IC 50; LIVER METABOLISM; LIVER MICROSOME; REACTION ANALYSIS; XENOBIOTIC METABOLISM; ADULT; ASIAN; DRUG ANTAGONISM; ENZYMOLOGY; MALE; METABOLISM; MIDDLE AGED;

ADULT; ARYL HYDROCARBON HYDROXYLASES; ASIAN CONTINENTAL ANCESTRY GROUP; ENZYME INHIBITORS; GLUCURONOSYLTRANSFERASE; HUMANS; MALE; MICROSOMES, LIVER; MIDDLE AGED; MIXED FUNCTION OXYGENASES; PILOCARPINE; RIFAMPIN;

EID: 0036252316     PISSN: 16714083     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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