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Volumn 55, Issue 2, 2002, Pages 104-117

KMUP 880708: A vanyllilamide-based β1-adrenoceptor antagonist with α-adrenoceptor blocking and potassium channel opening activities

(3) Praveen Rao, P N a Habeeb, Amgad G a Knaus, Edward E a

a UNIVERSITY OF ALBERTA (Canada)

Author keywords

adrenoceptor blockade; Capsaicin analogue; K+ channels; Radioligand binding assay; Vasorelaxant activity

Indexed keywords

1H 1,2,4 OXADIAZOLO[4,3 A]QUINOXALIN 1 ONE; 4 (3 TERT BUTYLAMINO 2 HYDROXYPROPOXY) 2 BENZIMIDAZOLONE; 4 AMINOPYRIDINE; APAMIN; ATENOLOL; BETA 1 ADRENERGIC RECEPTOR BLOCKING AGENT; CHARYBDOTOXIN; GLIBENCLAMIDE; INDOMETACIN; ISOPRENALINE; KMUP 880708; LABETALOL; METHYLENE BLUE; N [4 [2 HYDROXY 3 (2 METHOXY 1 OXYETHYLAMINOBENZENE)PROPOXY] 3 METHOXYBENZYL]HEXANAMIDE; N(G) NITROARGININE METHYL ESTER; PHENOBARBITAL; PHENYLEPHRINE; POTASSIUM CHANNEL; PRAZOSIN; PROPANOLAMINE DERIVATIVE; PROPRANOLOL; RADIOLIGAND; TETRYLAMMONIUM; UNCLASSIFIED DRUG; VANILLIN DERIVATIVE;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ARTERIAL PRESSURE; ARTICLE; BINDING ASSAY; BRADYCARDIA; BRAIN MEMBRANE; CHRONOTROPISM; CONTROLLED STUDY; DOSE RESPONSE; DRUG ANTAGONISM; DRUG EFFECT; DRUG POTENCY; DRUG SELECTIVITY; FAST MUSCLE; GUINEA PIG; HEART CONTRACTION; HEART MUSCLE RELAXATION; HEART RIGHT ATRIUM; INOTROPISM; NONHUMAN; RAT; SMOOTH MUSCLE RELAXATION; TACHYCARDIA; VASCULAR ENDOTHELIUM; VASCULAR SMOOTH MUSCLE; VASODILATATION;

EID: 0036239393 PISSN: 02724391 EISSN: None Source Type: Journal
DOI: 10.1002/ddr.10043 Document Type: Article

Times cited : (5)

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